Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50010717
TargetSubstance-K receptor(Human)
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50097911(5-Fluoro-3-[3-(4-methoxy-4-(methylsulfinyl)benzene...)
Affinity DataIC50: 2.5nMAssay Description:Binding affinity for heterologously expressed human Tachykinin receptor 2 using [3H]-SR- 48968 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50097912(3-(1-{2-[(R)-4-Benzoyl-2-(3,4-difluoro-phenyl)-mor...)
Affinity DataIC50: 6nMAssay Description:Binding affinity for heterologously expressed human Tachykinin receptor 2 using [3H]-SR- 48968 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50097914(1-[3-(5-Fluoro-1H-indol-3-yl)-propyl]-4-(methylsul...)
Affinity DataIC50: 13nMAssay Description:Binding affinity for heterologously expressed human Tachykinin receptor 2 using [3H]-SR- 48968 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50097915(1-[3-(3,4-dichlorophenyl)-4-methyl(phenyl)carboxam...)
Affinity DataIC50: 14nMAssay Description:Binding affinity for heterologously expressed human Tachykinin receptor 2 using [3H]-SR- 48968 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50097909(4-(oxidosulfanyl)benzenemethyl-1-[2-(5-fluoro-1H-i...)
Affinity DataIC50: 22nMAssay Description:Binding affinity for heterologously expressed human Tachykinin receptor 2 using [3H]-SR- 48968 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50097913(4-((oxidosulfanyl)benzene-phenyl-methyl)-1-[2-(5-f...)
Affinity DataIC50: 111nMAssay Description:Binding affinity for heterologously expressed human Tachykinin receptor 2 using [3H]-SR- 48968 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50097910((2S,12bR)-2-Benzenesulfinylmethyl-9-fluoro-1,2,3,4...)
Affinity DataIC50: 2.53E+4nMAssay Description:Binding affinity for heterologously expressed human Tachykinin receptor 2 using [3H]-SR- 48968 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed