Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50035193
TargetProtein Rev(Human immunodeficiency virus type 1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097336(Pyrene-1-carboxylic acid [(4R,5S,6S)-5-amino-6-((2...)
Affinity DataKd:  240nMAssay Description:Dissociation constant was determined in presence of Rev Response Element RNA IIBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097337(Neamine derivative | CHEMBL349996)
Affinity DataKd:  30nMAssay Description:Dissociation constant for TAR RNAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097336(Pyrene-1-carboxylic acid [(4R,5S,6S)-5-amino-6-((2...)
Affinity DataKd:  290nMAssay Description:Dissociation constant for TAR RNAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097338(Neamine derivative | CHEMBL408877)
Affinity DataKd:  25nMAssay Description:Dissociation constant for TAR RNAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetProtein Rev(Human immunodeficiency virus type 1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097339(Neamine derivative | CHEMBL415806)
Affinity DataKd:  3.40nMAssay Description:Dissociation constant was determined for Rev Response Element RNA IIBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetProtein Rev(Human immunodeficiency virus type 1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097337(Neamine derivative | CHEMBL349996)
Affinity DataKd:  8.5nMAssay Description:Dissociation constant was determined for Rev Response Element RNA IIBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097337(Neamine derivative | CHEMBL349996)
Affinity DataIC50: 28nMAssay Description:Inhibition of Tat peptide binding to HIV-1 TAR RNAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetProtein Rev(Human immunodeficiency virus type 1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097337(Neamine derivative | CHEMBL349996)
Affinity DataIC50: 350nMAssay Description:Inhibitory activity against peptide binding to the Rev Response Element RNA IIB was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetProtein Rev(Human immunodeficiency virus type 1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097335(2-Amino-5-guanidino-pentanoic acid [(4R,5S,6S)-5-a...)
Affinity DataIC50: 460nMAssay Description:Inhibitory activity against peptide binding to the RRE RNA was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097335(2-Amino-5-guanidino-pentanoic acid [(4R,5S,6S)-5-a...)
Affinity DataIC50: 600nMAssay Description:Inhibition of Tat peptide binding to HIV-1 TAR RNAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097336(Pyrene-1-carboxylic acid [(4R,5S,6S)-5-amino-6-((2...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of Tat peptide binding to HIV-1 TAR RNAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetProtein Rev(Human immunodeficiency virus type 1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM50097336(Pyrene-1-carboxylic acid [(4R,5S,6S)-5-amino-6-((2...)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibitory activity against peptide binding to the RRE RNA was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetProtein Rev(Human immunodeficiency virus type 1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM8580((2R,3S,4R,5R,6R)-5-amino-2-(aminomethyl)-6-{[(1R,2...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibitory activity against peptide binding to the RRE RNA was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetProtein Tat(HIV-1)
Graduate School of Bioscience and Biotechnology

Curated by ChEMBL
LigandPNGBDBM8580((2R,3S,4R,5R,6R)-5-amino-2-(aminomethyl)-6-{[(1R,2...)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibition of Tat peptide binding to HIV-1 TAR RNAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed