Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50010646
LigandPNGBDBM50081217(4-{5-[(S)-2-Butyl-4-(2,3-dimethyl-phenyl)-5-oxo-pi...)
Affinity DataIC50: 440nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant Ras-CVIM by human farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097070(4-{5-[(S)-2-Butyl-4-(2,3-dimethyl-phenyl)-6-oxo-pi...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant Ras-CVIM by human farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097071(4-{5-[4-(3-Chloro-phenyl)-3-oxo-piperazin-1-ylmeth...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant Ras-CVIM by human farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50097069(4-{5-[(S)-6-Butyl-4-(2,3-dimethyl-phenyl)-2,3-diox...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant Ras-CVIM by human farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097075(4-[5-(3-Oxo-4-phenyl-piperazin-1-ylmethyl)-imidazo...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant Ras-CVIM by human farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097075(4-[5-(3-Oxo-4-phenyl-piperazin-1-ylmethyl)-imidazo...)
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition of human geranylgeranyltransferase-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097073(4-{5-[4-(3-Chloro-phenyl)-2,3-dioxo-piperazin-1-yl...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant Ras-CVIM by human farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097074(4-{5-[4-(2,3-Dimethyl-phenyl)-3-oxo-piperazin-1-yl...)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant Ras-CVIM by human farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097076(4-[5-(2,3-Dioxo-4-phenyl-piperazin-1-ylmethyl)-imi...)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant Ras-CVIM by human farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097076(4-[5-(2,3-Dioxo-4-phenyl-piperazin-1-ylmethyl)-imi...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human geranylgeranyltransferase-1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097080(4-{5-[4-(2,3-Dimethyl-phenyl)-2,3-dioxo-piperazin-...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant Ras-CVIM by human farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097072(4-{5-[4-(3-Chloro-phenyl)-piperazine-1-carbonyl]-i...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant Ras-CVIM by human farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097078(4-{5-[4-(3-Chloro-phenyl)-3-oxo-piperazine-1-carbo...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant Ras-CVIM by human farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097081(4-{5-[4-(3-Chloro-phenyl)-2-oxo-piperazin-1-ylmeth...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant Ras-CVIM by human farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097079(4-{5-[4-(3-Chloro-phenyl)-piperazin-1-ylmethyl]-im...)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant Ras-CVIM by human farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50097077(4-[5-(2,5-Dioxo-4-phenyl-piperazin-1-ylmethyl)-imi...)
Affinity DataIC50: 9.50E+5nMAssay Description:Inhibition of [3H]FPP incorporation into recombinant Ras-CVIM by human farnesyl transferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed