Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50010592
TargetProtein kinase C alpha type(Human)
Institute of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50057509(8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1-methyl-...)
Affinity DataKi:  15nMAssay Description:Displacement phorbol 12,13-dibutyrate(PDBU) binding from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Institute of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50096601(8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-7-methoxy...)
Affinity DataKi:  46nMAssay Description:Displacement phorbol 12,13-dibutyrate(PDBU) binding from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C delta type(Human)
Institute of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50096601(8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-7-methoxy...)
Affinity DataKi:  91nMAssay Description:Binding affinity for protein kinase C deltaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C epsilon type(Human)
Institute of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50096601(8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-7-methoxy...)
Affinity DataKi:  121nMAssay Description:Binding affinity for protein kinase C epsilonMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Institute of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50057513(benzolactam-V8 | (2S,5S)-5-Hydroxymethyl-2-isoprop...)
Affinity DataKi:  334nMAssay Description:Displacement phorbol 12,13-dibutyrate(PDBU) binding from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Institute of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50096602((2S,5S)-5-Hydroxymethyl-2-isopropyl-7-methoxy-1-me...)
Affinity DataKi:  7.16E+3nMAssay Description:Displacement phorbol 12,13-dibutyrate(PDBU) binding from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed