Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50036966
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095801(CHEMBL61545 | CHEMBL1204234 | 2-{4-[4-(2-Butoxy-ph...)
Affinity DataKi:  1.20nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095818(CHEMBL61250 | CHEMBL1204241 | 2-{4-[4-(3-Trifluoro...)
Affinity DataKi:  3.60nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095817(CHEMBL1204235 | CHEMBL61614 | 2-{4-[4-(1,3-Dioxo-t...)
Affinity DataKi:  3.70nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095800(CHEMBL1204239 | CHEMBL62017 | 2-{4-[4-(1,3-Dioxo-t...)
Affinity DataKi:  3.90nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095816(CHEMBL1204250 | CHEMBL59791 | 2-{4-[4-(3-Bromo-phe...)
Affinity DataKi:  4nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095829(CHEMBL1204254 | CHEMBL292315 | 2-{4-[4-(2-Butoxy-p...)
Affinity DataKi:  6.5nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095803(CHEMBL292279 | CHEMBL1204232 | 2-{4-[4-(2-Methoxy-...)
Affinity DataKi:  8.60nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095810(CHEMBL1204230 | CHEMBL60973 | 2-{3-[4-(2-Butoxy-ph...)
Affinity DataKi:  11nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095825(CHEMBL58006 | CHEMBL1204253 | 2-{4-[4-(1,4-Dioxo-o...)
Affinity DataKi:  14nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095806(CHEMBL1204237 | CHEMBL417381 | 2-[4-(4-o-Tolyl-pip...)
Affinity DataKi:  16nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL416266 | CHEMBL1204203 | Ethanesulfonic acid...)
Affinity DataKi:  22nMAssay Description:In vitro binding affinity towards D2 receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095808(CHEMBL1204236 | CHEMBL59282 | 2-{4-[4-(1,4-Dioxo-o...)
Affinity DataKi:  24nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL416266 | CHEMBL1204203 | Ethanesulfonic acid...)
Affinity DataKi:  27nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095807(CHEMBL59778 | CHEMBL1204258 | 2-[3-(4-o-Tolyl-pipe...)
Affinity DataKi:  27nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095822(CHEMBL1204240 | CHEMBL58702 | 2-[4-(4-o-Tolyl-pipe...)
Affinity DataKi:  27nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095805(CHEMBL1204238 | CHEMBL58850 | 2-{4-[3-(1,4-Dioxo-h...)
Affinity DataKi:  31nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095802(CHEMBL1204229 | CHEMBL57953 | 2-{4-[3-(1,3-Dioxo-h...)
Affinity DataKi:  33nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095815(CHEMBL1204244 | CHEMBL61473 | 2-{3-[4-(3-Bromo-phe...)
Affinity DataKi:  33nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095823(CHEMBL60078 | CHEMBL1204257 | 2-{4-[3-(1,4-Dioxo-h...)
Affinity DataKi:  44nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095811(CHEMBL1204248 | CHEMBL58197 | 2-{4-[3-(1,3-Dioxo-h...)
Affinity DataKi:  60nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095813(CHEMBL293365 | CHEMBL1204231 | 2-{4-[4-(3-Amino-ph...)
Affinity DataKi:  80nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50369259(CHEMBL1202594)
Affinity DataKi:  102nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095804(CHEMBL293488 | CHEMBL1204243 | 2-{3-[4-(2-Butoxy-p...)
Affinity DataKi:  110nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095799(CHEMBL1204246 | CHEMBL301637 | 2-{3-[4-(2-Methoxy-...)
Affinity DataKi:  126nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095828(CHEMBL417213 | CHEMBL1204245 | 2-[3-(4-o-Tolyl-pip...)
Affinity DataKi:  134nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095820(CHEMBL1204252 | CHEMBL61904 | N-(3-{4-[4-(1,4-Diox...)
Affinity DataKi:  169nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095809(CHEMBL1204255 | CHEMBL294837 | 2-{3-[4-(3-Trifluor...)
Affinity DataKi:  214nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095826(CHEMBL1204247 | CHEMBL58946 | N-(3-{4-[3-(1,4-Diox...)
Affinity DataKi:  326nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095821(CHEMBL59892 | CHEMBL1204233 | 2-{4-[4-(1,3-Dioxo-h...)
Affinity DataKi:  341nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095819(CHEMBL293048 | CHEMBL1204242 | 2-{4-[4-(1,4-Dioxo-...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095827(CHEMBL1204228 | CHEMBL59062 | N-(3-{4-[3-(1,3-Diox...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL416266 | CHEMBL1204203 | Ethanesulfonic acid...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 3 receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095812(CHEMBL59950 | CHEMBL1204249 | 2-{3-[4-(3-Amino-phe...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095824(CHEMBL418638 | CHEMBL1204251 | 2-{4-[3-(1,3-Dioxo-...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 4(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL416266 | CHEMBL1204203 | Ethanesulfonic acid...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity towards 5-HT4 receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL416266 | CHEMBL1204203 | Ethanesulfonic acid...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50095814(CHEMBL1204256 | CHEMBL60211 | 2-{4-[3-(1,4-Dioxo-o...)
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed