Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 50004708
TargetMultidrug resistance-associated protein 1(Human)
Queen'S University

Curated by ChEMBL
LigandPNGBDBM50420244(CHEMBL1628111)
Affinity DataKi:  380nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetMultidrug resistance-associated protein 1(Human)
Queen'S University

Curated by ChEMBL
LigandPNGBDBM50366524(Estrone Sulphate | ESTRONE | ESTROPIPATE | Estrone...)
Affinity DataKi:  450nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in membrane vesicle from MRP1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed