Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 50010413
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094676(Diethyl-[2-(1H-indol-3-yl)-ethyl]-amine | N,N-diet...)
Affinity DataEC50:  5.37E+3nMAssay Description:Evaluated for the effective concentration at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094675(3-(2-Diethylamino-ethyl)-1H-indol-4-ol | CHEMBL143...)
Affinity DataEC50:  2.31E+3nMAssay Description:Evaluated for the effective concentration at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094672(Diethyl-[2-(6-fluoro-1H-indol-3-yl)-ethyl]-amine |...)
Affinity DataEC50:  3.70E+3nMAssay Description:EC50 for inhibition of 50 uM forskolin-stimulated cAMP accumulation against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094674([2-(4-Fluoro-5-methoxy-1H-indol-3-yl)-ethyl]-dimet...)
Affinity DataEC50:  1.81E+4nMAssay Description:Evaluated for the effective concentration at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094669([2-(6-Fluoro-5-methoxy-1H-indol-3-yl)-ethyl]-dimet...)
Affinity DataEC50:  7.90E+3nMAssay Description:Evaluated for the effective concentration at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094673(Diethyl-[2-(5-methoxy-1H-indol-3-yl)-ethyl]-amine ...)
Affinity DataEC50:  2.39E+3nMAssay Description:Evaluated for the effective concentration at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094672(Diethyl-[2-(6-fluoro-1H-indol-3-yl)-ethyl]-amine |...)
Affinity DataEC50:  3.39E+4nMAssay Description:Evaluated for the effective concentration at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094677(3-(2-Dimethylamino-ethyl)-7-fluoro-1H-indol-4-ol |...)
Affinity DataEC50:  4.92E+3nMAssay Description:Evaluated for the effective concentration at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094671(3-(2-Dimethylamino-ethyl)-6-fluoro-1H-indol-4-ol |...)
Affinity DataEC50:  2.60E+3nMAssay Description:Evaluated for the effective concentration at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataEC50:  5.82nMAssay Description:EC50 for inhibition of 50 uM forskolin-stimulated cAMP accumulation against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094676(Diethyl-[2-(1H-indol-3-yl)-ethyl]-amine | N,N-diet...)
Affinity DataEC50:  680nMAssay Description:EC50 for inhibition of 50 uM forskolin-stimulated cAMP accumulation against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataEC50:  0.130nMAssay Description:EC50 for inhibition of 50 uM forskolin-stimulated cAMP accumulation against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094673(Diethyl-[2-(5-methoxy-1H-indol-3-yl)-ethyl]-amine ...)
Affinity DataEC50:  22nMAssay Description:EC50 for inhibition of 50 uM forskolin-stimulated cAMP accumulation against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094674([2-(4-Fluoro-5-methoxy-1H-indol-3-yl)-ethyl]-dimet...)
Affinity DataEC50:  0.930nMAssay Description:EC50 for inhibition of 50 uM forskolin-stimulated cAMP accumulation against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094670(LY-293384 | LY 293284 | LY-293284 | CHEMBL276031 |...)
Affinity DataKi:  0.0880nMAssay Description:Inhibition constant of 50 uM forskolin-stimulated cAMP accumulation against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094673(Diethyl-[2-(5-methoxy-1H-indol-3-yl)-ethyl]-amine ...)
Affinity DataKi:  1.70nMAssay Description:Evaluated for the binding constant at [3H]8-OH-DPAT-labeled human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094677(3-(2-Dimethylamino-ethyl)-7-fluoro-1H-indol-4-ol |...)
Affinity DataKi:  5.40nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094671(3-(2-Dimethylamino-ethyl)-6-fluoro-1H-indol-4-ol |...)
Affinity DataKi:  7.40nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094675(3-(2-Diethylamino-ethyl)-1H-indol-4-ol | CHEMBL143...)
Affinity DataKi:  10nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094677(3-(2-Dimethylamino-ethyl)-7-fluoro-1H-indol-4-ol |...)
Affinity DataKi:  13nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094673(Diethyl-[2-(5-methoxy-1H-indol-3-yl)-ethyl]-amine ...)
Affinity DataKi:  16nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094669([2-(6-Fluoro-5-methoxy-1H-indol-3-yl)-ethyl]-dimet...)
Affinity DataKi:  19nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094675(3-(2-Diethylamino-ethyl)-1H-indol-4-ol | CHEMBL143...)
Affinity DataKi:  25nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094669([2-(6-Fluoro-5-methoxy-1H-indol-3-yl)-ethyl]-dimet...)
Affinity DataKi:  33nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094673(Diethyl-[2-(5-methoxy-1H-indol-3-yl)-ethyl]-amine ...)
Affinity DataKi:  42nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094676(Diethyl-[2-(1H-indol-3-yl)-ethyl]-amine | N,N-diet...)
Affinity DataKi:  47nMAssay Description:Evaluated for the binding constant at [3H]8-OH-DPAT-labeled human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094675(3-(2-Diethylamino-ethyl)-1H-indol-4-ol | CHEMBL143...)
Affinity DataKi:  49nMAssay Description:Evaluated for the binding constant at [3H]8-OH-DPAT-labeled human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094674([2-(4-Fluoro-5-methoxy-1H-indol-3-yl)-ethyl]-dimet...)
Affinity DataKi:  55nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094669([2-(6-Fluoro-5-methoxy-1H-indol-3-yl)-ethyl]-dimet...)
Affinity DataKi:  84.5nMAssay Description:Evaluated for the binding constant at [3H]8-OH-DPAT-labeled human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094676(Diethyl-[2-(1H-indol-3-yl)-ethyl]-amine | N,N-diet...)
Affinity DataKi:  104nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094671(3-(2-Dimethylamino-ethyl)-6-fluoro-1H-indol-4-ol |...)
Affinity DataKi:  114nMAssay Description:Evaluated for the binding constant at [3H]8-OH-DPAT-labeled human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094677(3-(2-Dimethylamino-ethyl)-7-fluoro-1H-indol-4-ol |...)
Affinity DataKi:  120nMAssay Description:Evaluated for the binding constant at [3H]8-OH-DPAT-labeled human 5-hydroxytryptamine 1A receptor receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094674([2-(4-Fluoro-5-methoxy-1H-indol-3-yl)-ethyl]-dimet...)
Affinity DataKi:  122nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094676(Diethyl-[2-(1H-indol-3-yl)-ethyl]-amine | N,N-diet...)
Affinity DataKi:  133nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094672(Diethyl-[2-(6-fluoro-1H-indol-3-yl)-ethyl]-amine |...)
Affinity DataKi:  145nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2C(Rat)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094672(Diethyl-[2-(6-fluoro-1H-indol-3-yl)-ethyl]-amine |...)
Affinity DataKi:  210nMAssay Description:Evaluated for the binding constant at [125I]-DOI-labeled rat 5-hydroxytryptamine 2C receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Purdue University

Curated by ChEMBL
LigandPNGBDBM50094672(Diethyl-[2-(6-fluoro-1H-indol-3-yl)-ethyl]-amine |...)
Affinity DataKi:  256nMAssay Description:Evaluated for the binding constant at [3H]8-OH-DPAT-labeled human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed