Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50036882
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094575(4-[(1R,2R,6R,7R,8R)-8-hydroxytricyclo[5.2.1.0^{2,6...)
Affinity DataKi:  450nMAssay Description:In vivo binding affinity fot cytosolic androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094570((3aS) -4-(5-Hydroxy-5-methyl-octahydro-4,7-methano...)
Affinity DataIC50: 1.20E+3nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50368314(ZANOTERONE)
Affinity DataKi:  2.20E+3nMAssay Description:In vivo binding affinity fot cytosolic androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094568(4-[(1S,2S,6S,7S,8S)-8-hydroxytricyclo[5.2.1.0^{2,6...)
Affinity DataIC50: 2.32E+3nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM18161(DHT | Dihydrotestosterone | [3H]DHT | (5alpha,17be...)
Affinity DataIC50: 3.20E+3nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094576(4-[(1R,2R,6R,7R,8S)-8-hydroxytricyclo[5.2.1.0^{2,6...)
Affinity DataIC50: 3.90E+3nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094579((3aS)-4-(5-Hydroxy-5-vinyl-octahydro-4,7-methano-i...)
Affinity DataIC50: 9.73E+3nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094578(4-[(1S,2S,6S,7S,8R)-8-hydroxytricyclo[5.2.1.0^{2,6...)
Affinity DataIC50: 1.04E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094580((3aS) -4-(5-Ethynyl-5-hydroxy-octahydro-4,7-methan...)
Affinity DataIC50: 1.35E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094572((3aS)-2-(4-Oxo-cyclohexylidene)-octahydro-4,7-meth...)
Affinity DataIC50: 1.42E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094574((3aS) -4-(5-Hydroxy-5-trifluoromethyl-octahydro-4,...)
Affinity DataIC50: 1.56E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094569(Cyproterone 17-O-acetate | cyproterone acetate | C...)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of [3H]-R-1881 binding to rat ventral prostrate cytosolic androgen receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094571((3aR)-4-(5-Hydroxy-5-methyl-octahydro-4,7-methano-...)
Affinity DataIC50: 2.74E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094566((3aR) -2-(4-Oxo-cyclohexylidene)-octahydro-4,7-met...)
Affinity DataIC50: 3.30E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094575(4-[(1R,2R,6R,7R,8R)-8-hydroxytricyclo[5.2.1.0^{2,6...)
Affinity DataIC50: 3.59E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094567((3aR)-4-(5-Hydroxy-5-trifluoromethyl-octahydro-4,7...)
Affinity DataIC50: 4.12E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094577((3aR)-4-(5-Ethynyl-5-hydroxy-octahydro-4,7-methano...)
Affinity DataIC50: 5.70E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetAndrogen receptor(Rat)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM50094581((3aR)-4-(5-Hydroxy-5-vinyl-octahydro-4,7-methano-i...)
Affinity DataIC50: 6.25E+4nMAssay Description:Ability to inhibit binding of [3H]R-1881 to rat ventral prostrate cytosolic androgen receptor was measured in a radioligand binding assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed