Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50003560
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50472901(CHEMBL2111833)
Affinity DataIC50: 100nMAssay Description:Binding affinity against Src SH2 domain in competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50472902(CHEMBL2111834)
Affinity DataIC50: 200nMAssay Description:Binding affinity against Src SH2 domain in competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50472903(CHEMBL2112641)
Affinity DataIC50: 1.60E+3nMAssay Description:Binding affinity against Src SH2 domain in competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50097347(Phosphoric acid mono-(4-{2-acetylamino-2-[1-(3-car...)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity against Src SH2 domain in competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50101077((2S,3S)-2-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-phosphon...)
Affinity DataIC50: 5.60E+3nMAssay Description:Binding affinity against Src SH2 domain in competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50472904(CHEMBL2112639)
Affinity DataIC50: 8.10E+3nMAssay Description:Binding affinity against Src SH2 domain in competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Ariad Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50472905(CHEMBL2112638)
Affinity DataIC50: 3.20E+4nMAssay Description:Binding affinity against Src SH2 domain in competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed