Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 50010080
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50422274(Human gonadoliberin-i | GONADORELIN)
Affinity DataIC50: 2nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090745(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 7nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090748(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 11nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090736(1-{2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 14nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090732(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 16nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090724(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 17nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090730(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 20nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090734(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 23nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090723(1-{2-[2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 25nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090752(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 28nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090728(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 28nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090725(1-{2-[2-({2-[2-(2-Acetylamino-3-naphthalen-2-yl-pr...)
Affinity DataIC50: 31nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090737(1-[2-(3-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 38nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090727(1-{2-[(1-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pr...)
Affinity DataIC50: 42nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090747(1-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-propio...)
Affinity DataIC50: 45nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090744(1-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-propio...)
Affinity DataIC50: 70nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090750(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 72nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090739(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 74nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090733(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 81nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090746(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 88nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090738(Ac-D-Nal2-D-Cpa-D-Pal-Pro-Arg-Pro-D-Ala-NH2 | CHEM...)
Affinity DataIC50: 110nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090743(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 130nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090729(1-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-propio...)
Affinity DataIC50: 130nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090749(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-pro...)
Affinity DataIC50: 140nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090751(1-[2-(2-{2-[2-(2-Acetylamino-3-phenyl-propionylami...)
Affinity DataIC50: 230nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090753(1-[2-(2-{2-[2-(2-Amino-3-naphthalen-2-yl-propionyl...)
Affinity DataIC50: 280nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090735(1-[2-(2-{2-[2-(2-Acetylamino-3-naphthalen-1-yl-pro...)
Affinity DataIC50: 370nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090740(1-{2-[2-(2-{2-[2-Acetylamino-3-(1H-indol-3-yl)-pro...)
Affinity DataIC50: 450nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090742(1-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-propio...)
Affinity DataIC50: 550nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090726(1-(2-{2-[2-(2-Acetylamino-3-naphthalen-2-yl-propio...)
Affinity DataIC50: 1.50E+3nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090741([1-(1-{1-[({1-[2-(1-Carbamoyl-ethylcarbamoyl)-pyrr...)
Affinity DataIC50: 2.20E+3nMAssay Description:Concentration of the peptide which displaces 50% of 125 I-[D-Lys6] gonadotropin-releasing hormone bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed