Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50010079
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090718(N-(1-{1-[1-Carboxy-2-(1H-indol-3-yl)-ethylcarbamoy...)
Affinity DataKi:  230nMAssay Description:Inhibition constant for the displacement of specific binding of [125I][D-Lys6]-GnRH (Kd=177 pM) bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090717(15,18-Di-sec-butyl-9,12-bis-(1H-indol-3-ylmethyl)-...)
Affinity DataKi:  320nMAssay Description:Inhibition constant for the displacement of specific binding of [125I][D-Lys6]-GnRH (Kd=177 pM) bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090721(2-{2-[2-[2-[2-(2-Amino-3-methyl-pentanoylamino)-3-...)
Affinity DataKi:  500nMAssay Description:Inhibition constant for the displacement of specific binding of [125I][D-Lys6]-GnRH (Kd=177 pM) bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090712(2-{2-[2-[2-[2-(2-Amino-3-methyl-pentanoylamino)-3-...)
Affinity DataKi:  700nMAssay Description:Inhibition constant for the displacement of specific binding of [125I][D-Lys6]-GnRH (Kd=177 pM) bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090722([5,8-Di-sec-butyl-11,14-bis-(1H-indol-3-ylmethyl)-...)
Affinity DataKi:  700nMAssay Description:Inhibition constant for the displacement of specific binding of [125I][D-Lys6]-GnRH (Kd=177 pM) bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50001220(CHEMBL317064 | 3-{2-[2-Acetylamino-3-(1H-indol-3-y...)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition constant for the displacement of specific binding of [125I][D-Lys6]-GnRH (Kd=177 pM) bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090719(2-{2-[2-(2-{2-[2-Acetylamino-3-(1H-indol-3-yl)-pro...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition constant for the displacement of specific binding of [125I][D-Lys6]-GnRH (Kd=177 pM) bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090716(2-{2-[2-[2-[2-(2-Amino-3-methyl-pentanoylamino)-3-...)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition constant for the displacement of specific binding of [125I][D-Lys6]-GnRH (Kd=177 pM) bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090715(3-{2-[2-Amino-3-(1H-indol-3-yl)-propionylamino]-4-...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition constant for the displacement of specific binding of [125I][D-Lys6]-GnRH (Kd=177 pM) bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090720(2-(2-{2-[2-[2-(2-Amino-3-methyl-pentanoylamino)-3-...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition constant for the displacement of specific binding of [125I][D-Lys6]-GnRH (Kd=177 pM) bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Institute of Science

Curated by ChEMBL
LigandPNGBDBM50090714(2-(2-{2-[2-[2-(2-Amino-3-methyl-pentanoylamino)-3-...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition constant for the displacement of specific binding of [125I][D-Lys6]-GnRH (Kd=177 pM) bound to rat pituitary membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed