Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50010057
TargetD(2) dopamine receptor(Rat)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50090488(1-Benzyl-1,2,3,4-tetrahydro-isoquinoline-6,7-diol ...)
Affinity DataKi:  640nMAssay Description:The compound has been evaluated for its binding affinity towards Dopamine receptor D2 by displacing the radioligand [3H]YM-09151-2 (0.5 nM) in rat st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50017041(1,2,3,4-Tetrahydro-1-(phenylmethyl)isoquinoline | ...)
Affinity DataKi:  3.57E+3nMAssay Description:The compound has been evaluated for its binding affinity towards Dopamine receptor D2 by displacing the radioligand [3H]YM-09151-2 (0.5 nM) in rat st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50090489(4-(1,2,3,4-Tetrahydro-isoquinolin-1-ylmethyl)-benz...)
Affinity DataKi:  8.79E+3nMAssay Description:The compound has been evaluated for its binding affinity towards Dopamine receptor D2 by displacing the radioligand [3H]YM-09151-2 (0.5 nM) in rat st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50090488(1-Benzyl-1,2,3,4-tetrahydro-isoquinoline-6,7-diol ...)
Affinity DataKi:  9.27E+3nMAssay Description:The compound has been evaluated for its binding affinity towards Dopamine receptor D1 by displacing the radioligand [3H]SCH-23390 (1.5 nM) in rat str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50090489(4-(1,2,3,4-Tetrahydro-isoquinolin-1-ylmethyl)-benz...)
Affinity DataKi:  2.15E+4nMAssay Description:The compound has been evaluated for its binding affinity towards Dopamine transporter by displacing the radioligand [3H]GBR-12935 (1.0 nM) in rat str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50017041(1,2,3,4-Tetrahydro-1-(phenylmethyl)isoquinoline | ...)
Affinity DataKi:  3.66E+4nMAssay Description:The compound has been evaluated for its binding affinity towards Dopamine transporter by displacing the radioligand [3H]GBR-12935 (1.0 nM) in rat str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50090488(1-Benzyl-1,2,3,4-tetrahydro-isoquinoline-6,7-diol ...)
Affinity DataKi:  5.76E+4nMAssay Description:The compound has been evaluated for its binding affinity towards Dopamine transporter by displacing the radioligand [3H]GBR-12935 (1.0 nM) in rat str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50090489(4-(1,2,3,4-Tetrahydro-isoquinolin-1-ylmethyl)-benz...)
Affinity DataKi:  1.75E+5nMAssay Description:The compound has been evaluated for its binding affinity towards Dopamine receptor D1 by displacing the radioligand [3H]SCH-23390 (1.5 nM) in rat str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50017041(1,2,3,4-Tetrahydro-1-(phenylmethyl)isoquinoline | ...)
Affinity DataKi:  2.49E+5nMAssay Description:The compound has been evaluated for its binding affinity towards Dopamine receptor D1 by displacing the radioligand [3H]SCH-23390 (1.5 nM) in rat str...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed