Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50009917
TargetNeutrophil elastase(Human)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089098(Cys-Phe-Leu-Glu-Ala-Ile-Pro-Met-Asp-Ile-Pro-Pro-Gl...)
Affinity DataKi:  1.90E+4nMAssay Description:Competitive inhibition constant against Human neutrophil elastase using the reporter substrate MeO-AAPV-pNaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089095(Met-Phe-Leu-Glu-Ala-Ile-Pro-Met-Ser-Ile | CHEMBL21...)
Affinity DataKi:  2.70E+4nMAssay Description:Competitive inhibition constant against Human neutrophil elastase using the reporter substrate MeO-AAPV-pNaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089095(Met-Phe-Leu-Glu-Ala-Ile-Pro-Met-Ser-Ile | CHEMBL21...)
Affinity DataKi:  1.00E+5nMAssay Description:Peptide was tested for inhibition constant for competitive inhibition using Suc-AAPA-pNa and Pancreatic elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen A(Bovine)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089095(Met-Phe-Leu-Glu-Ala-Ile-Pro-Met-Ser-Ile | CHEMBL21...)
Affinity DataKi:  1.60E+5nMAssay Description:Competitive inhibition constant against Chymotrypsinogen using the reporter substrate Suc-AAPA-pNaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089098(Cys-Phe-Leu-Glu-Ala-Ile-Pro-Met-Asp-Ile-Pro-Pro-Gl...)
Affinity DataKi:  1.90E+5nMAssay Description:Peptide was tested for inhibition constant for competitive inhibition using Suc-AAPA-pNa and Pancreatic elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089094(Met-Phe-Leu-Glu-Ala-Ile-Pro-Met-Ser | CHEMBL414810)
Affinity DataKi:  1.90E+5nMAssay Description:Competitive inhibition constant against Human neutrophil elastase using the reporter substrate MeO-AAPV-pNaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen A(Bovine)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089098(Cys-Phe-Leu-Glu-Ala-Ile-Pro-Met-Asp-Ile-Pro-Pro-Gl...)
Affinity DataKi:  2.40E+5nMAssay Description:Competitive inhibition constant against Chymotrypsinogen using the reporter substrate Suc-AAPA-pNaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089096(ent-Met-Phe-Leu-Glu-Ala-Ile-Pro-Met | Met-Phe-Leu-...)
Affinity DataKi:  2.70E+5nMAssay Description:Competitive inhibition constant against Human neutrophil elastase using the reporter substrate MeO-AAPV-pNaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089097(Met-Phe-Leu-Glu-Ala-Ile-Pro-Lys | CHEMBL21028)
Affinity DataKi:  5.40E+5nMAssay Description:Competitive inhibition constant against trypsin using the reporter substrate Ac-R-pNaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen A(Bovine)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089094(Met-Phe-Leu-Glu-Ala-Ile-Pro-Met-Ser | CHEMBL414810)
Affinity DataKi:  3.10E+6nMAssay Description:Competitive inhibition constant against Chymotrypsinogen using the reporter substrate Suc-AAPA-pNaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089099((S)-2-{(S)-2-[(S)-2-((S)-2-Amino-4-methylsulfanyl-...)
Affinity DataKi:  1.10E+6nMAssay Description:Peptide was tested for inhibition constant for competitive inhibition using Suc-AAPA-pNa and Pancreatic elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen A(Bovine)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089096(ent-Met-Phe-Leu-Glu-Ala-Ile-Pro-Met | Met-Phe-Leu-...)
Affinity DataKi:  2.30E+6nMAssay Description:Competitive inhibition constant against Chymotrypsinogen using the reporter substrate Suc-AAPA-pNaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsin-like elastase family member 2A(Pig)
The Oxford Centre For Molecular Sciences

Curated by ChEMBL
LigandPNGBDBM50089094(Met-Phe-Leu-Glu-Ala-Ile-Pro-Met-Ser | CHEMBL414810)
Affinity DataKi:  5.80E+6nMAssay Description:Peptide was tested for inhibition constant for competitive inhibition using Suc-AAPA-pNa and Pancreatic elastaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed