Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50036808
TargetIntegrase(Human immunodeficiency virus type 1)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065793(8-Hydroxy-2-[(E)-2-(3,4,5-trihydroxy-phenyl)-vinyl...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human immunodeficiency virus-1 (HIV-1) integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein(RSV-Pr-C)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065793(8-Hydroxy-2-[(E)-2-(3,4,5-trihydroxy-phenyl)-vinyl...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein(RSV-Pr-C)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065796(2-[2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-quino...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065796(2-[2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-quino...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human immunodeficiency virus-1 (HIV-1) integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065790(2-[2-(2,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-quino...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human immunodeficiency virus-1 (HIV-1) integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065788(2-(3-carboxy-4-hydroxystyryl)-8-hydroxyquinoline-7...)
Affinity DataIC50: 2.70E+3nMAssay Description:Compound was tested in vitro to inhibit human immuno virus-1 (HIV-1) using enzymatic disintegration assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50087421(8-hydroxy-2-styrylquinoline-7-carboxylic acid | 8-...)
Affinity DataIC50: 3.40E+3nMAssay Description:Compound was tested in vitro to inhibit human immuno virus-1 (HIV-1) using enzymatic disintegration assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50087435(8-hydroxy-2-(4-hydroxystyryl)quinoline-7-carboxyli...)
Affinity DataIC50: 4.20E+3nMAssay Description:Compound was tested in vitro to inhibit human immuno virus-1 (HIV-1) using enzymatic disintegration assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein(RSV-Pr-C)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065788(2-(3-carboxy-4-hydroxystyryl)-8-hydroxyquinoline-7...)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein(RSV-Pr-C)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50087421(8-hydroxy-2-styrylquinoline-7-carboxylic acid | 8-...)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein(RSV-Pr-C)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50087435(8-hydroxy-2-(4-hydroxystyryl)quinoline-7-carboxyli...)
Affinity DataIC50: 2.09E+4nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein(RSV-Pr-C)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065786(2-[2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-quino...)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein(RSV-Pr-C)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065790(2-[2-(2,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-quino...)
Affinity DataIC50: 3.83E+4nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein(RSV-Pr-C)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065787(4-(2-(8-hydroxyquinolin-2-yl)vinyl)benzene-1,2-dio...)
Affinity DataIC50: 6.51E+4nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein(RSV-Pr-C)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065800((E)-3-(3,4-Dihydroxy-phenyl)-acrylic acid 2-methyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein(RSV-Pr-C)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065789(2-Styryl-quinolin-8-ol | 2-Styrylquinolin-8-ol | 2...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065789(2-Styryl-quinolin-8-ol | 2-Styrylquinolin-8-ol | 2...)
Affinity DataIC50: 1.00E+5nMAssay Description:Compound was tested in vitro to inhibit human immuno virus-1 (HIV-1) using enzymatic disintegration assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065784(4-[(E)-2-(8-Nitro-quinolin-2-yl)-vinyl]-benzene-1,...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human immunodeficiency virus-1 (HIV-1) integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065791(4-[(E)-2-(8-Amino-quinolin-2-yl)-vinyl]-benzene-1,...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human immunodeficiency virus-1 (HIV-1) integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065800((E)-3-(3,4-Dihydroxy-phenyl)-acrylic acid 2-methyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human immunodeficiency virus-1 (HIV-1) integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein(RSV-Pr-C)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065784(4-[(E)-2-(8-Nitro-quinolin-2-yl)-vinyl]-benzene-1,...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065798(Acetic acid 2-((E)-styryl)-quinolin-8-yl ester | A...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human immunodeficiency virus-1 (HIV-1) integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein(RSV-Pr-C)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065802(Acetic acid 2-acetoxy-5-[2-(8-acetoxy-quinolin-2-y...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein(RSV-Pr-C)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065791(4-[(E)-2-(8-Amino-quinolin-2-yl)-vinyl]-benzene-1,...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065802(Acetic acid 2-acetoxy-5-[2-(8-acetoxy-quinolin-2-y...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human immunodeficiency virus-1 (HIV-1) integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed
TargetGag-Pol polyprotein(RSV-Pr-C)
Cnrs Umr 8532

Curated by ChEMBL
LigandPNGBDBM50065798(Acetic acid 2-((E)-styryl)-quinolin-8-yl ester | A...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/14/2012
Entry Details Article
PubMed