Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 50009702
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  0.470nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086855(Cyclohexanecarboxylic acid ((S)-1-phenethyl-pyrrol...)
Affinity DataKi:  0.490nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM21395(3-(2-{4-[(4-fluorophenyl)carbonyl]piperidin-1-yl}e...)
Affinity DataKi:  0.660nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity for Dopamine receptor D2 by displacement of [3H]-spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086861(3-Methylsulfanyl-N-((S)-1-phenethyl-pyrrolidin-2-y...)
Affinity DataKi:  4.30nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086856(N-((S)-1-Phenethyl-pyrrolidin-2-ylmethyl)-benzamid...)
Affinity DataKi:  4.60nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086857(5-Methylsulfanyl-2,3-dihydro-benzofuran-7-carboxyl...)
Affinity DataKi:  6.70nMAssay Description:Binding affinity for Dopamine receptor D2 by displacement of [3H]-spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086858(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  10nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086852(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  12nMAssay Description:Binding affinity for Dopamine receptor D2 by displacement of [3H]-spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086854(5-Methoxy-2,3-dihydro-benzofuran-7-carboxylic acid...)
Affinity DataKi:  21nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086851(2-Methoxy-5-methylsulfanyl-N-((S)-1-phenethyl-pyrr...)
Affinity DataKi:  24nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086852(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  34nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086862(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  35nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  43nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086862(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  57nMAssay Description:Binding affinity for Dopamine receptor D2 by displacement of [3H]-spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086863(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  86nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086857(5-Methylsulfanyl-2,3-dihydro-benzofuran-7-carboxyl...)
Affinity DataKi:  100nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086860(3-Methylsulfanyl-N-((R)-1-phenethyl-pyrrolidin-2-y...)
Affinity DataKi:  110nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086854(5-Methoxy-2,3-dihydro-benzofuran-7-carboxylic acid...)
Affinity DataKi:  120nMAssay Description:Binding affinity for Dopamine receptor D2 by displacement of [3H]-spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086861(3-Methylsulfanyl-N-((S)-1-phenethyl-pyrrolidin-2-y...)
Affinity DataKi:  160nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086851(2-Methoxy-5-methylsulfanyl-N-((S)-1-phenethyl-pyrr...)
Affinity DataKi:  170nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086853(Cyclohexanecarboxylic acid ((R)-1-phenethyl-pyrrol...)
Affinity DataKi:  190nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086855(Cyclohexanecarboxylic acid ((S)-1-phenethyl-pyrrol...)
Affinity DataKi:  240nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM21395(3-(2-{4-[(4-fluorophenyl)carbonyl]piperidin-1-yl}e...)
Affinity DataKi:  240nMAssay Description:Binding affinity for Dopamine receptor D2 by displacement of [3H]-spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086858(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  280nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086852(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  300nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086857(5-Methylsulfanyl-2,3-dihydro-benzofuran-7-carboxyl...)
Affinity DataKi:  430nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086856(N-((S)-1-Phenethyl-pyrrolidin-2-ylmethyl)-benzamid...)
Affinity DataKi:  430nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086863(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  430nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086851(2-Methoxy-5-methylsulfanyl-N-((S)-1-phenethyl-pyrr...)
Affinity DataKi:  460nMAssay Description:Binding affinity for Dopamine receptor D2 by displacement of [3H]-spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086863(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  630nMAssay Description:Binding affinity for Dopamine receptor D2 by displacement of [3H]-spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086854(5-Methoxy-2,3-dihydro-benzofuran-7-carboxylic acid...)
Affinity DataKi:  660nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086858(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataKi:  800nMAssay Description:Binding affinity for Dopamine receptor D2 by displacement of [3H]-spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086853(Cyclohexanecarboxylic acid ((R)-1-phenethyl-pyrrol...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against binding of Dopamine receptor D2 by displacement of [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086855(Cyclohexanecarboxylic acid ((S)-1-phenethyl-pyrrol...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against binding of Dopamine receptor D2 by displacement of [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086859(N-((R)-1-Phenethyl-pyrrolidin-2-ylmethyl)-benzamid...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]-ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086861(3-Methylsulfanyl-N-((S)-1-phenethyl-pyrrolidin-2-y...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against binding of Dopamine receptor D2 by displacement of [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086859(N-((R)-1-Phenethyl-pyrrolidin-2-ylmethyl)-benzamid...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM21395(3-(2-{4-[(4-fluorophenyl)carbonyl]piperidin-1-yl}e...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 1A receptor from striata of male Wistar rats by displacement of [3H]8-OH-DPATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against binding of Dopamine receptor D2 by displacement of [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086853(Cyclohexanecarboxylic acid ((R)-1-phenethyl-pyrrol...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]-ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086860(3-Methylsulfanyl-N-((R)-1-phenethyl-pyrrolidin-2-y...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against binding of Dopamine receptor D2 by displacement of [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]-ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086859(N-((R)-1-Phenethyl-pyrrolidin-2-ylmethyl)-benzamid...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against binding of Dopamine receptor D2 by displacement of [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086862(6-Chloro-4-methyl-3,4-dihydro-2H-benzo[1,4]oxazine...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]-ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086856(N-((S)-1-Phenethyl-pyrrolidin-2-ylmethyl)-benzamid...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against binding of Dopamine receptor D2 by displacement of [3H]spiperoneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerotonin 2 (5-HT2) receptor(Rat)
Yoshitomi Pharmaceutical Industries

Curated by ChEMBL
LigandPNGBDBM50086860(3-Methylsulfanyl-N-((R)-1-phenethyl-pyrrolidin-2-y...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory concentration against binding of 5-hydroxytryptamine 2 receptor from striata of male Wistar rats by displacement of [3H]-ketanserinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed