Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50009625
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085756BDBM50085756(cyclo(1,1'-3)Ac-D-Asp (Gly)-D-Cpa-D-Lys-Ser-Tyr-D-...)
Affinity DataKi:  0.140nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085742BDBM50085742(cyclo(1,1'-3)Ac-D-Asp (beta-Ala)-D-Cpa-D-Orn-Ser-T...)
Affinity DataKi:  0.170nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085761BDBM50085761(cyclo(1,1'-3)Ac-D-Asp (Gaba)-D-Cpa-D-Dpr-Ser-Tyr-D...)
Affinity DataKi:  0.180nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085753BDBM50085753(cyclo(1-3)Ac-D-Glu-D-Cpa-D-Dbu-Ser-Tyr-D-Nal-Leu-A...)
Affinity DataKi:  0.310nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085757BDBM50085757(cyclo(1,1'-3)Ac-D-Asp (beta-Ala)-D-Cpa-D-Dbu-Ser-T...)
Affinity DataKi:  0.320nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085746BDBM50085746(cyclo(1,1'-3)Ac-D-Asp (Gly)-D-Cpa-D-Orn-Ser-Tyr-D-...)
Affinity DataKi:  0.340nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085751BDBM50085751(cyclo(1,1'-3)Ac-D-Asp (beta-Ala)-D-Cpa-D-Dpr-Ser-T...)
Affinity DataKi:  0.350nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085748BDBM50085748(cyclo(1-3)Ac-D-Glu-D-Cpa-D-Lys-Ser-Tyr-D-Nal-Leu-A...)
Affinity DataKi:  0.470nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085763BDBM50085763(cyclo(1-3)Ac-D-Asp (D-Ala)-D-Cpa-D-Dbu-Ser-Tyr-D-N...)
Affinity DataKi:  0.570nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085752BDBM50085752(cyclo(1,1'-3)Ac-D-Asp (Gly)-D-Cpa-D-Dbu-Ser-Tyr-D-...)
Affinity DataKi:  0.700nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085760BDBM50085760(cyclo(1-3)Ac-D-Asp-D-Cpa-D-Lys-Ser-Tyr-D-Nal-Leu-A...)
Affinity DataKi:  0.820nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085744BDBM50085744(dicyclo(1-3, 4-10)Ac-D-Asp-D-Cpa-D-Lys-Asp-Tyr-D-N...)
Affinity DataKi:  1.20nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085758BDBM50085758(cyclo(1,1'-3)Ac-D-Glu (Gly)-D-Cpa-D-Lys-Ser-Tyr-D-...)
Affinity DataKi:  1.5nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085750BDBM50085750(cyclo(1-3)Ac-D-Asp-D-Cpa-D-Orn-Ser-Tyr-D-Nal-Leu-A...)
Affinity DataKi:  1.60nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085759BDBM50085759(cyclo(1-3)Ac-D-Dpr-D-Cpa-D-Asp-Ser-Tyr-D-Nal-Leu-A...)
Affinity DataKi:  1.70nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085767BDBM50085767(cyclo(1,1'-3)Ac-D-Asp (Ala)-D-Cpa-D-Dbu-Ser-Tyr-D-...)
Affinity DataKi:  1.80nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085741BDBM50085741(cyclo(1,1'-3)Ac-D-Glu (beta-Ala)-D-Cpa-D-Lys-Ser-T...)
Affinity DataKi:  2.20nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085743BDBM50085743(cyclo(1,1'-3)Ac-D-Orn (beta-Ala)-D-Cpa-D-Asp-Ser-T...)
Affinity DataKi:  2.20nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085755BDBM50085755(cyclo(1,1'-3)Ac-D-Asp (D-Ala)-D-Cpa-D-Orn-Ser-Tyr-...)
Affinity DataKi:  2.40nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085749BDBM50085749(cyclo(1,1'-3)Ac-D-Asp (Ala)-D-Cpa-D-Orn-Ser-Tyr-D-...)
Affinity DataKi:  3.30nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085765BDBM50085765(cyclo(1,1'-3)Ac-D-Glu-D-Cpa-D-Orn-Ser-Tyr-D-Nal-Le...)
Affinity DataKi:  4.20nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085762BDBM50085762(tricyclo(1-3/4-10/5-8)Ac-D-Glu-D-Cpa-D-Lys-Asp-Glu...)
Affinity DataKi:  4.60nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085766BDBM50085766(cyclo(1-3)Ac-D-Glu-D-Cpa-D-Orn-Ser-Tyr-D-Nal-Leu-A...)
Affinity DataKi:  5.20nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085764BDBM50085764(cyclo(1,1'-3)Ac-D-Glu (Gly)-D-Cpa-D-Dbu-Ser-Tyr-D-...)
Affinity DataKi:  20.3nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085747BDBM50085747(cyclo(1-3)Ac-D-Glu-D-Cpa-D-Dbu-Ser-Tyr-D-Arg-Leu-A...)
Affinity DataKi:  31nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085745BDBM50085745(cyclo(1-3)Ac-Asp-D-Cpa-Dpr-Ser-Tyr-D-Nal-Leu-Arg-P...)
Affinity DataKi:  31nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50085754BDBM50085754(cyclo(1,1'-3)Ac-D-Asp (Ala)-D-Cpa-D-Orn-Ser-Tyr-D-...)
Affinity DataKi:  350nMAssay Description:Competitive radioligand binding assay for rat Gonadotropin-releasing hormone receptor cells stably transfected in human HEK293More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed