Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 50009624
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085734(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  0.100nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085715(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  0.160nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085719(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  0.200nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085718(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  0.200nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085710(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  0.200nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085720(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  0.230nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085737(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  0.230nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085732(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  0.270nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085735(Cyclo (5-8) [Ac-D Nal, D Cpa, D Pal, Asp, Glu, D A...)
Affinity DataKi:  0.280nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085704(Cyclo (4-10) [Ac-D Nal, D Cpa, D Pal, Asp, Glu, D ...)
Affinity DataKi:  0.320nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085711(DiCyclo (4-10/5-8) [Ac-D Nal, D Cpa, D Trp, Asp, G...)
Affinity DataKi:  0.320nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085722(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  0.350nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085730(Cyclo (4-10) [Ac-D Nal, D Fpa, D Trp, Asp, Glu, D ...)
Affinity DataKi:  0.360nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085729(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  0.370nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085705(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  0.590nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085707(Cyclo (4-10) [Ac-Delta Pro, D Fpa, D Trp, Asp, MeT...)
Affinity DataKi:  0.740nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085725(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  0.75nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085709(Cyclo (5-8) [Ac-D Nal, D Cpa, D Trp, Asp, Glu, D N...)
Affinity DataKi:  1nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085728(DiCyclo (4-10/5-8) [Ac-D Nal, D Cpa, D Trp, Asp, G...)
Affinity DataKi:  1.20nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085727(Cyclo (5-8) [Ac-D Nal, D Cpa, D Pal, Asp, Asp, D P...)
Affinity DataKi:  1.30nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085723(DiCyclo (4-10/5-8) [Ac-D Nal, D Cpa, D Pal, Asp, G...)
Affinity DataKi:  1.30nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085738(Cyclo (4-10) [Ac-D Nal, D Fpa, D Trp, Glu, Glu, D ...)
Affinity DataKi:  1.30nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085717(Cyclo (4-10) [Ac-D Nal, D Fpa, D Trp, Asp, Glu, D ...)
Affinity DataKi:  1.30nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085713(Cyclo (5,5'-8) [Ac-D Nal, Cpa, D Pal, Asp, Glu(bet...)
Affinity DataKi:  1.80nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085713(Cyclo (5,5'-8) [Ac-D Nal, Cpa, D Pal, Asp, Glu(bet...)
Affinity DataKi:  1.80nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085712(Cyclo (5-8) [Ac-D Nal, D Cpa, D Trp, Asp, Glu, D A...)
Affinity DataKi:  2.30nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085733(Cyclo (5-8) [Ac-D Nal, D Cpa, D Pal, Asp, Cys, D A...)
Affinity DataKi:  2.40nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085714(Cyclo (5-8) [Ac-D Nal, D Cpa, D Pal, Asp, Glu, D P...)
Affinity DataKi:  3.30nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085739(Cyclo (5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp, Asp(G...)
Affinity DataKi:  3.60nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085736(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  4.20nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085708(Cyclo (5-8) [Ac-D Nal, Cpa, D Pal, Asp, D Glu, D A...)
Affinity DataKi:  8.5nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085726(Cyclo (4-10) [Ac-D Nal, D Fpa, D Trp, Asp, Glu, D ...)
Affinity DataKi:  10nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085731(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  12nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085740(Cyclo (5-8) [Ac-D Nal, D Cpa, D Trp, Asp, Glu, D A...)
Affinity DataKi:  20nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085712(Cyclo (5-8) [Ac-D Nal, D Cpa, D Trp, Asp, Glu, D A...)
Affinity DataKi:  21nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085703(Cyclo (5-8) [Ac-D Nal, Cpa, D Pal, Asp, D Glu, D A...)
Affinity DataKi:  120nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085721(DiCyclo (4-10/5,5'-8) [Ac-D Nal, D Cpa, D Pal, Asp...)
Affinity DataKi:  120nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085706(Cyclo (5-8) [Ac-D Nal, Cpa, D Pal, Asp, Asp, D Arg...)
Affinity DataKi:  130nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085724(Cyclo (5-8) [Ac-D Nal, D Cpa, D Trp, Asp, Dcys, D ...)
Affinity DataKi:  450nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085716(Cyclo (5-8) [Ac-D Nal, Cpa, D Trp, Asp, Asp, D Glu...)
Affinity DataKi:  720nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGonadotropin-releasing hormone receptor(Rat)
Salk Institute

Curated by ChEMBL
LigandPNGBDBM50085716(Cyclo (5-8) [Ac-D Nal, Cpa, D Trp, Asp, Asp, D Glu...)
Affinity DataKi:  720nMAssay Description:Competitive radioligand binding assay, in human HEK293 cells stably transfected with the rat Gonadotropin-releasing hormone receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed