Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 50009615
TargetIntegrin alpha-IIb/beta-3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50082933([6-(4-Carbamimidoyl-benzoylamino)-chroman-2-yl]-ac...)
Affinity DataIC50: 2nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50082930([6-(4-Carbamimidoyl-benzoylamino)-1-oxo-1,2,3,4-te...)
Affinity DataIC50: 2nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50085605([6-(4-Carbamimidoyl-2-fluoro-benzoylamino)-1-oxo-1...)
Affinity DataIC50: 3nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50085612([6-(4-Carbamimidoyl-2,6-difluoro-benzoylamino)-1-o...)
Affinity DataIC50: 5nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50085611({6-[(6-Carbamimidoyl-pyridine-3-carbonyl)-amino]-1...)
Affinity DataIC50: 9nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50085614([6-(4-Carbamimidoyl-2-chloro-benzoylamino)-1-oxo-1...)
Affinity DataIC50: 11nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50085607([1-Oxo-6-((E)-3-piperidin-4-yl-acryloylamino)-1,2,...)
Affinity DataIC50: 26nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50085610([1-Oxo-6-(3-piperidin-4-yl-propionylamino)-1,2,3,4...)
Affinity DataIC50: 71nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50085606([6-(4-Carbamimidoyl-2-trifluoromethyl-benzoylamino...)
Affinity DataIC50: 72nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50085609({6-[(5-Carbamimidoyl-thiophene-2-carbonyl)-amino]-...)
Affinity DataIC50: 210nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50085608([1-Oxo-6-(piperidin-4-ylmethoxycarbonylamino)-1,2,...)
Affinity DataIC50: 330nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50085604([1-Oxo-6-(3-piperidin-4-yl-propylamino)-1,2,3,4-te...)
Affinity DataIC50: 610nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrin alpha-IIb/beta-3(Human)
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50085613({1-Oxo-6-[2-(piperidin-4-yloxy)-acetylamino]-1,2,3...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of fibrinogen binding to purified human GPIIb-IIIa in ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed