Report error Found 88 Enz. Inhib. hit(s) with all data for entry = 50009460
Affinity DataIC50: 2.30nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.80nMAssay Description:Inhibition of Vitronectin receptor (alpha V beta 3) bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30nMAssay Description:Inhibition of Vitronectin receptor (alpha V beta 3) bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 8.5nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of Vitronectin receptor (alpha V beta 3) bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alphaV-beta3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of adhesion of integrin beta-3-transfected HEK293 cells to fibrinogenMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair
Affinity DataIC50: 44nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibition of Vitronectin receptor (alpha V beta 3) bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of Vitronectin receptor (alpha V beta 3) bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair
Affinity DataIC50: 66nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of adhesion of integrin beta-3-transfected HEK293 cells to fibrinogenMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair
Affinity DataIC50: 83nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Inhibition of Vitronectin receptor (alpha V beta 3) bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair
Affinity DataIC50: 290nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 360nMAssay Description:Inhibitory activity against beta-3-transfected 293 cells using alpha-V beta-3 antagonism assayMore data for this Ligand-Target Pair
Affinity DataIC50: 400nMAssay Description:Inhibition of aggregation of human gel-purified platelets (GPIIbIIIa GPP)More data for this Ligand-Target Pair


































