Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50009241
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50081533(CP-199331 | N-{3-[(3R,4R)-6-(5,6-Difluoro-benzothi...)
Affinity DataKi:  0.400nMAssay Description:In vitro binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50081532(CP-199330 | N-{3-[(3R,4R)-6-(7-Chloro-quinolin-2-y...)
Affinity DataKi:  0.600nMAssay Description:In vitro binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50023198(CHEMBL21333 | N-(4-oxo-2-(1H-tetrazol-5-yl)-4H-chr...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding of Cysteinyl leukotriene receptor 1 to guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCysteinyl leukotriene receptor 1(Guinea pig)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50009073(cyclopentyl 3-(2-methoxy-4-((o-tolylsulfonyl)carba...)
Affinity DataKi:  2nMAssay Description:In vitro binding of cysLT1 receptor to guinea pig lung membranes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)