Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50009167
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080832([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-1-methyl-2-...)
Affinity DataKd:  3nMAssay Description:The compound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Men...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080832([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-1-methyl-2-...)
Affinity DataIC50: 11nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080831([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-cyclohexylc...)
Affinity DataKd:  30nMAssay Description:The compound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Men...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080836(4-[2-[2-(3-Amino-benzyloxycarbonylamino)-3-(4-phos...)
Affinity DataKd:  45nMAssay Description:The compound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Men...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080830([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-2-(4-phosph...)
Affinity DataKd:  60nMAssay Description:The compound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Men...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080834({4-[2-[2-(3-Amino-benzyloxycarbonylamino)-3-(4-pho...)
Affinity DataKd:  60nMAssay Description:The compound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Men...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080831([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-cyclohexylc...)
Affinity DataIC50: 120nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080836(4-[2-[2-(3-Amino-benzyloxycarbonylamino)-3-(4-phos...)
Affinity DataIC50: 153nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080833([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-2-(4-hydrox...)
Affinity DataKd:  155nMAssay Description:The compound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Men...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080834({4-[2-[2-(3-Amino-benzyloxycarbonylamino)-3-(4-pho...)
Affinity DataIC50: 198nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080830([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-2-(4-phosph...)
Affinity DataIC50: 235nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080835([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-2-(4-hydrox...)
Affinity DataKd:  250nMAssay Description:The compound was tested on a LS250B Perkin-Elmer fluorimeter for Growth factor receptor bound protein 2 equilibrium constant(Kd) by the Michaelis-Men...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080833([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-2-(4-hydrox...)
Affinity DataIC50: 497nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGrowth factor receptor-bound protein 2(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50080835([1-[1-(1,2-Dicarbamoyl-ethylcarbamoyl)-2-(4-hydrox...)
Affinity DataIC50: 1.10E+3nMAssay Description:The compound was evaluated for its potency to inhibit the interaction between Growth factor receptor bound protein 2 and phosphotyrosine-containing p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed