Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50036745
TargetBifunctional purine biosynthesis protein ATIC(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50369444(CHEMBL608337)
Affinity DataKd:  20nMAssay Description:Binding affinity towards AICAR formyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetBifunctional purine biosynthesis protein ATIC(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50369444(CHEMBL608337)
Affinity DataIC50: 125nMAssay Description:Inhibitory activity against AICAR formyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetBifunctional purine biosynthesis protein ATIC(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50080319(10-Formyl-8-deazafolic acid | CHEMBL114215)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibitory activity against AICAR formyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetBifunctional purine biosynthesis protein ATIC(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM22579(Aminoimidazole-4-carboxamide ribonucleotide | CHEM...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against AICAR formyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetBifunctional purine biosynthesis protein ATIC(Human)
The Pennsylvania State University

Curated by ChEMBL
LigandPNGBDBM50080320((2R)-2-{[4-(N-{[(6R)-2-amino-4-oxo-1,4,4a,5,6,7,8,...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against AICAR formyltransferaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed