Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50008900
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054245(CHEMBL45281 | cid_176157 | 5-Chloro-N-cyclopropylm...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054252(5-Bromo-N-cyclopropylmethyl-2-methyl-N-propyl-N'-(...)
Affinity DataKi:  2nMAssay Description:Ability to inhibit [125I]CRH binding to human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054250(N-Cyclopropylmethyl-2,5-dimethyl-N-propyl-N'-(2,4,...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054248(2,5-Dimethyl-N,N-dipropyl-N'-(2,4,6-trichloro-phen...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054253(N-Cyclopropylmethyl-5-ethyl-2-methyl-N-propyl-N'-(...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054225(N-Cyclopropylmethyl-6-methyl-N-propyl-N'-(2,4,6-tr...)
Affinity DataKi:  57nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054226(N,N-Diallyl-6-methyl-N'-(2,4,6-trimethyl-phenyl)-[...)
Affinity DataKi:  115nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054230(6-Methyl-N,N-dipropyl-N'-(2,4,6-trimethyl-phenyl)-...)
Affinity DataKi:  130nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054246(N-Cyclopropylmethyl-2-methyl-N-propyl-N'-(2,4,6-tr...)
Affinity DataKi:  253nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054246(N-Cyclopropylmethyl-2-methyl-N-propyl-N'-(2,4,6-tr...)
Affinity DataKi:  253nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054216(N-Benzyl-6-methyl-N-propyl-N'-(2,4,6-trimethyl-phe...)
Affinity DataKi:  490nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054221(N,N-Dibutyl-6-methyl-N'-(2,4,6-trimethyl-phenyl)-[...)
Affinity DataKi:  490nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054239([4-(3,6-Dihydro-2H-pyridin-1-yl)-6-methyl-[1,3,5]t...)
Affinity DataKi:  1.05E+3nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054219(N-Benzyl-N-butyl-6-methyl-N'-(2,4,6-trimethyl-phen...)
Affinity DataKi:  1.05E+3nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054255(N-Cyclopropylmethyl-2-methyl-N-propyl-N'-(2,4,6-tr...)
Affinity DataKi:  1.39E+3nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054223(N-Benzyl-N-ethyl-6-methyl-N'-(2,4,6-trimethyl-phen...)
Affinity DataKi:  1.47E+3nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054241(6-Methyl-N-(4-trifluoromethyl-benzyl)-N'-(2,4,6-tr...)
Affinity DataKi:  1.69E+3nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054234(6,N-Dimethyl-N-phenethyl-N'-(2,4,6-trimethyl-pheny...)
Affinity DataKi:  2.10E+3nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50078345(N-Cyclopropylmethyl-6-methyl-N-propyl-N'-(2,4,6-tr...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
The University of Wollongong

Curated by ChEMBL
LigandPNGBDBM50054235(N-Cyclopropylmethyl-6-ethyl-N-propyl-N'-(2,4,6-tri...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of [125I]CRH binding to human Corticotropin releasing factor receptor 1.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed