Compile Data Set for Download or QSAR
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 3629
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36783(2-(1 R-isopropyl-2-hydroxyethylamino)-9-isopropylp...)
Affinity DataIC50: 20nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36784(2-(1 R-isopropyl-2-hydroxyethylamino)-9-isopropylp...)
Affinity DataIC50: 30nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36782(2-(1 R-isopropyl-2-hydroxyethylamino)-9-isopropylp...)
Affinity DataIC50: 33nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36764(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 35nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36788(2-(1 R-isopropyl-2-hydroxyethylamino)-9-isopropylp...)
Affinity DataIC50: 40nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36787(2-(1 R-isopropyl-2-hydroxyethylamino)-9-isopropylp...)
Affinity DataIC50: 52nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36789(2-(1 R-isopropyl-2-hydroxyethylamino)-9-isopropylp...)
Affinity DataIC50: 80nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36786(2-(1 R-isopropyl-2-hydroxyethylamino)-9-isopropylp...)
Affinity DataIC50: 100nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36755(6-(4-methoxybenzylamino) core C2-substituent, 36)
Affinity DataIC50: 100nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36797(2-(2-hydroxyethylpiperidyl)-9-isopropylpurine core...)
Affinity DataIC50: 130nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36754(6-(4-methoxybenzylamino) core C2-substituent, 33)
Affinity DataIC50: 130nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36791(2-(2-hydroxyethylpiperidyl)-9-isopropylpurine core...)
Affinity DataIC50: 160nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36790(2-(1 R-isopropyl-2-hydroxyethylamino)-9-isopropylp...)
Affinity DataIC50: 170nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36757(6-(4-methoxybenzylamino) core C2-substituent, 10)
Affinity DataIC50: 210nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36731(2-(2-hydroxyethylamino)-9-isopropylpurine core C6-...)
Affinity DataIC50: 220nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36759(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 220nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36761(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 230nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36752(6-(4-methoxybenzylamino) core C2-substituent, 75)
Affinity DataIC50: 230nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36781(2-(1 R-isopropyl-2-hydroxyethylamino)-9-isopropylp...)
Affinity DataIC50: 240nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36748(6-(4-methoxybenzylamino) core C2-substituent, 16)
Affinity DataIC50: 240nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36749(6-(4-methoxybenzylamino) core C2-substituent, 211)
Affinity DataIC50: 250nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36733(2-(2-hydroxyethylamino)-9-isopropylpurine core C6-...)
Affinity DataIC50: 270nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36734(2-(2-hydroxyethylamino)-9-isopropylpurine core C6-...)
Affinity DataIC50: 290nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36766(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 300nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36777(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 300nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36747(6-(4-methoxybenzylamino) core C2-substituent, 26)
Affinity DataIC50: 330nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36760(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 350nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36785(2-(1 R-isopropyl-2-hydroxyethylamino)-9-isopropylp...)
Affinity DataIC50: 360nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36732(2-(2-hydroxyethylamino)-9-isopropylpurine core C6-...)
Affinity DataIC50: 400nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36771(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 400nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36730(2-(2-hydroxyethylamino)-9-isopropylpurine core C6-...)
Affinity DataIC50: 420nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36728(2-(2-hydroxyethylamino)-9-isopropylpurine core C6-...)
Affinity DataIC50: 430nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36756(6-(4-methoxybenzylamino) core C2-substituent, 314)
Affinity DataIC50: 450nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36774(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 500nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36776(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 500nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36729(2-(2-hydroxyethylamino)-9-isopropylpurine core C6-...)
Affinity DataIC50: 500nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36768(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 500nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36765(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 500nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36767(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 530nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36741(6-(4-methoxybenzylamino) core C2-substituent, 28)
Affinity DataIC50: 560nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36753(6-(4-methoxybenzylamino) core C2-substituent, 76)
Affinity DataIC50: 600nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36779(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 620nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36735(6-(4-methoxybenzylamino) core C2-substituent, 118)
Affinity DataIC50: 700nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36798(2-(2-hydroxyethylpiperidyl)-9-isopropylpurine core...)
Affinity DataIC50: 790nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36772(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 800nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36758(6-(3-chloroanilino)-9-isopropylpurine core C2-subs...)
Affinity DataIC50: 900nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36740(6-(4-methoxybenzylamino) core C2-substituent, 37)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36736(6-(4-methoxybenzylamino) core C2-substituent, 13)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36796(2-(2-hydroxyethylpiperidyl)-9-isopropylpurine core...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
University of California Berkeley

LigandPNGBDBM36746(6-(4-methoxybenzylamino) core C2-substituent, 209)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition assay using CDK1/cyclin B.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
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