Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50008829
TargetProtein kinase C alpha type(Human)
Institute of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50057511(CHEMBL27266 | 13-Hydroxymethyl-10-isopropyl-9-meth...)
Affinity DataKi:  11nMAssay Description:Displacement of phorbol 12,13-dibutyrate (PDBU) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Institute of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50057509(8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1-methyl-...)
Affinity DataKi:  15nMAssay Description:Displacement of phorbol 12,13-dibutyrate (PDBU) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Institute of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50057513(benzolactam-V8 | (2S,5S)-5-Hydroxymethyl-2-isoprop...)
Affinity DataKi:  334nMAssay Description:Displacement of phorbol 12,13-dibutyrate (PDBU) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Institute of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50077648((2S,5S)-7-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...)
Affinity DataKi:  2.10E+4nMAssay Description:Displacement of phorbol 12,13-dibutyrate (PDBU) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Institute of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50077649((2S,5S)-5-Hydroxymethyl-2-isopropyl-1-methyl-1,2,4...)
Affinity DataKi:  1.27E+5nMAssay Description:Displacement of phorbol 12,13-dibutyrate (PDBU) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed