Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 3628
TargetVitamin D-binding protein(Rat)
Ligand Pharmaceuticals

LigandPNGBDBM36717(1,25(OH)2D3)
Affinity DataIC50: 40nMpH: 7.4 T: 2°CAssay Description:DBP competition binding assay were done using human serum (Scantibodies) or rat serum (Gibco-BRL).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetVitamin D-binding protein(Human)
Ligand Pharmaceuticals

LigandPNGBDBM36717(1,25(OH)2D3)
Affinity DataIC50: 200nMpH: 7.4 T: 2°CAssay Description:DBP competition binding assay were done using human serum (Scantibodies) or rat serum (Gibco-BRL).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetVitamin D-binding protein(Human)
Ligand Pharmaceuticals

LigandPNGBDBM36718(LG190090)
Affinity DataIC50: 1.00E+3nMpH: 7.4 T: 2°CAssay Description:DBP competition binding assay were done using human serum (Scantibodies) or rat serum (Gibco-BRL).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetVitamin D-binding protein(Human)
Ligand Pharmaceuticals

LigandPNGBDBM36719(LG190119)
Affinity DataIC50: 1.00E+3nMpH: 7.4 T: 2°CAssay Description:DBP competition binding assay were done using human serum (Scantibodies) or rat serum (Gibco-BRL).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetVitamin D-binding protein(Human)
Ligand Pharmaceuticals

LigandPNGBDBM36720(LG190155)
Affinity DataIC50: 1.00E+3nMpH: 7.4 T: 2°CAssay Description:DBP competition binding assay were done using human serum (Scantibodies) or rat serum (Gibco-BRL).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetVitamin D-binding protein(Human)
Ligand Pharmaceuticals

LigandPNGBDBM36721(LG190176)
Affinity DataIC50: 1.00E+3nMpH: 7.4 T: 2°CAssay Description:DBP competition binding assay were done using human serum (Scantibodies) or rat serum (Gibco-BRL).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetVitamin D-binding protein(Human)
Ligand Pharmaceuticals

LigandPNGBDBM36722(LG190178)
Affinity DataIC50: 1.00E+3nMpH: 7.4 T: 2°CAssay Description:DBP competition binding assay were done using human serum (Scantibodies) or rat serum (Gibco-BRL).More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Ligand Pharmaceuticals

LigandPNGBDBM36717(1,25(OH)2D3)
Affinity DataKi:  0.5nM ΔG°:  -49.3kJ/molepH: 7.5 T: 2°CAssay Description:VDR in vitro ligand-binding assay using human VDR constructed into a yeast expression plasmid.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Ligand Pharmaceuticals

LigandPNGBDBM36722(LG190178)
Affinity DataKi:  150nM ΔG°:  -36.2kJ/molepH: 7.5 T: 2°CAssay Description:VDR in vitro ligand-binding assay using human VDR constructed into a yeast expression plasmid.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Ligand Pharmaceuticals

LigandPNGBDBM36718(LG190090)
Affinity DataKi: >1.00E+3nM ΔG°: >-31.8kJ/molepH: 7.5 T: 2°CAssay Description:VDR in vitro ligand-binding assay using human VDR constructed into a yeast expression plasmid.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Ligand Pharmaceuticals

LigandPNGBDBM36719(LG190119)
Affinity DataKi: >1.00E+3nM ΔG°: >-31.8kJ/molepH: 7.5 T: 2°CAssay Description:VDR in vitro ligand-binding assay using human VDR constructed into a yeast expression plasmid.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Ligand Pharmaceuticals

LigandPNGBDBM36720(LG190155)
Affinity DataKi: >1.00E+3nM ΔG°: >-31.8kJ/molepH: 7.5 T: 2°CAssay Description:VDR in vitro ligand-binding assay using human VDR constructed into a yeast expression plasmid.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed
TargetVitamin D3 receptor(Human)
Ligand Pharmaceuticals

LigandPNGBDBM36721(LG190176)
Affinity DataKi: >1.00E+3nM ΔG°: >-31.8kJ/molepH: 7.5 T: 2°CAssay Description:VDR in vitro ligand-binding assay using human VDR constructed into a yeast expression plasmid.More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2011
Entry Details Article
PubMed