Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50008713
TargetMetabotropic glutamate receptor 2(Human)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076389((1S,2S)-2-[(R)-Amino-carboxy-(9-methyl-9H-xanthen-...)
Affinity DataIC50: 34nMAssay Description:Inhibitory activity against human Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50049748(2-Amino-4-(4,4-diphenyl-butyl)-pentanedioic acid |...)
Affinity DataIC50: 400nMAssay Description:Inhibitory activity against human Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50069111((2S,4S)-2-Amino-4-(2,2-diphenyl-ethyl)-pentanedioi...)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibitory activity against human Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076393((1S,2S,3R)-2-((S)-Amino-carboxy-methyl)-3-phenyl-c...)
Affinity DataIC50: 9.90E+3nMAssay Description:Inhibitory activity against Metabotropic glutamate receptor 2 in the rat HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50052256(3-[amino(carboxy)methyl]bicyclo[1.1.1]pentane-1-ca...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50053585((S)-4-(amino(carboxy)methyl)-2-hydroxybenzoic acid...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory activity against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076392((1S,2S)-2-((S)-1-Amino-1-carboxy-ethyl)-cyclopropa...)
Affinity DataIC50: 7.70E+4nMAssay Description:Inhibitory activity against Metabotropic glutamate receptor 2 in the rat HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076395((1R,2S,4R)-4-Amino-cyclopentane-1,2,4-tricarboxyli...)
Affinity DataIC50: 8.80E+4nMAssay Description:Inhibitory activity against Metabotropic glutamate receptor 2 in the rat HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076390(GAMMA-CARBOXY-GLUTAMIC ACID | (S)-2-Amino-4-carbox...)
Affinity DataIC50: 1.02E+5nMAssay Description:Inhibitory activity against Metabotropic glutamate receptor 2 in the rat HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076395((1R,2S,4R)-4-Amino-cyclopentane-1,2,4-tricarboxyli...)
Affinity DataIC50: 1.15E+5nMAssay Description:Inhibitory activity against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50052256(3-[amino(carboxy)methyl]bicyclo[1.1.1]pentane-1-ca...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibitory activity against Metabotropic glutamate receptor 2 in the rat HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076394(ABHD-I | CHEMBL39215 | 2-Amino-bicyclo[2.2.1]hepta...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibitory activity against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50034503(DCG-IV | (2S,2'R,3'R)-2-(2',3')-dicarboxycycloprop...)
Affinity DataIC50: 3.89E+5nMAssay Description:Inhibitory activity against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50056272((2S,6S)-2-Amino-bicyclo[3.1.0]hexane-2,6-dicarboxy...)
Affinity DataIC50: 4.58E+5nMAssay Description:Inhibitory activity against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 1(Rat)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076391(7-Amino-bicyclo[2.2.1]heptane-2,7-dicarboxylic aci...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against Metabotropic glutamate receptor 1 in the rat LLC-PK1/HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMetabotropic glutamate receptor 2(Human)
Parc Club Orsay Université

Curated by ChEMBL
LigandPNGBDBM50076391(7-Amino-bicyclo[2.2.1]heptane-2,7-dicarboxylic aci...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against Metabotropic glutamate receptor 2 in the rat HEK 293 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed