Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50008675
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)
Affinity DataIC50: 17nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063745(2-(2-Iodo-phenylamino)-7-trifluoromethyl-benzo[d][...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibitory activity against purified human C1r protease proteaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075982(4-Methoxy-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin...)
Affinity DataIC50: 700nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075980(4-Chloro-N-ethyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2...)
Affinity DataIC50: 930nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075979(4-Chloro-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-...)
Affinity DataIC50: 1.30E+3nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075992(4-Guanidino-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxaz...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075986(N-Ethyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2-yl)-benz...)
Affinity DataIC50: 1.50E+3nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075981(4-Amino-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2...)
Affinity DataIC50: 2.20E+3nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075978(2-Bromo-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2...)
Affinity DataIC50: 2.80E+3nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075992(4-Guanidino-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxaz...)
Affinity DataIC50: 3.00E+3nMAssay Description:Evaluated in vitro for inhibitory activity against purified human C1r protease incubated in buffer for 60 minutesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075986(N-Ethyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2-yl)-benz...)
Affinity DataIC50: 3.20E+3nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063745(2-(2-Iodo-phenylamino)-7-trifluoromethyl-benzo[d][...)
Affinity DataIC50: 4.00E+3nMAssay Description:Evaluated in vitro for inhibitory activity against purified human C1r protease incubated in buffer for 60 minutesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075993(N-Methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2-yl)-ben...)
Affinity DataIC50: 4.00E+3nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075991(3-Chloro-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-...)
Affinity DataIC50: 4.20E+3nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075989(Naphthalene-1-sulfonic acid methyl-(4-oxo-4H-benzo...)
Affinity DataIC50: 4.30E+3nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075987(4,N-Dimethyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2-yl)...)
Affinity DataIC50: 4.50E+3nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075990(4-tert-Butyl-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxa...)
Affinity DataIC50: 5.83E+3nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075982(4-Methoxy-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin...)
Affinity DataIC50: 6.00E+3nMAssay Description:Evaluated in vitro for inhibitory activity against purified human C1r protease incubated in buffer for 60 minutesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075989(Naphthalene-1-sulfonic acid methyl-(4-oxo-4H-benzo...)
Affinity DataIC50: 6.00E+3nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075993(N-Methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2-yl)-ben...)
Affinity DataIC50: 6.00E+3nMAssay Description:Evaluated in vitro for inhibitory activity against purified human C1r protease incubated in buffer for 60 minutesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075981(4-Amino-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2...)
Affinity DataIC50: 7.00E+3nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075981(4-Amino-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2...)
Affinity DataIC50: 7.00E+3nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075984(2,6-Dichloro-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxa...)
Affinity DataIC50: 7.50E+3nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075987(4,N-Dimethyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2-yl)...)
Affinity DataIC50: 7.80E+3nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075985(3,4-Dichloro-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxa...)
Affinity DataIC50: 8.30E+3nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075986(N-Ethyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2-yl)-benz...)
Affinity DataIC50: 8.30E+3nMAssay Description:Evaluated in vitro for inhibitory activity against purified human C1r protease incubated in buffer for 60 minutesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075989(Naphthalene-1-sulfonic acid methyl-(4-oxo-4H-benzo...)
Affinity DataIC50: 1.00E+4nMAssay Description:Evaluated in vitro for inhibitory activity against purified human C1r protease incubated in buffer for 60 minutesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075984(2,6-Dichloro-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxa...)
Affinity DataIC50: 1.01E+4nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)
Affinity DataIC50: 1.20E+4nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063698(4-Guanidino-benzoic acid 6-carbamimidoyl-naphthale...)
Affinity DataIC50: 1.20E+4nMAssay Description:Evaluated in vitro for inhibitory activity against purified human C1r protease incubated in buffer for 60 minutesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075977(4-Cyano-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075991(3-Chloro-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-...)
Affinity DataIC50: 2.40E+4nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075978(2-Bromo-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2...)
Affinity DataIC50: 2.50E+4nMAssay Description:Evaluated in vitro for inhibitory activity against purified human C1r protease incubated in buffer for 60 minutesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075980(4-Chloro-N-ethyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2...)
Affinity DataIC50: 3.00E+4nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075976(N-Methyl-4-nitro-N-(4-oxo-4H-benzo[d][1,3]oxazin-2...)
Affinity DataIC50: 3.10E+4nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075991(3-Chloro-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-...)
Affinity DataIC50: 5.80E+4nMAssay Description:Evaluated in vitro for inhibitory activity against purified human C1r protease incubated in buffer for 60 minutesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075990(4-tert-Butyl-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxa...)
Affinity DataIC50: 6.00E+4nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075990(4-tert-Butyl-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxa...)
Affinity DataIC50: 6.00E+4nMAssay Description:Evaluated in vitro for inhibitory activity against purified human C1r protease incubated in buffer for 60 minutesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075979(4-Chloro-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-...)
Affinity DataIC50: 6.20E+4nMAssay Description:Evaluated in vitro for inhibitory activity against purified human C1r protease incubated in buffer for 60 minutesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075980(4-Chloro-N-ethyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2...)
Affinity DataIC50: 6.20E+4nMAssay Description:Evaluated in vitro for inhibitory activity against purified human C1r protease incubated in buffer for 60 minutesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075984(2,6-Dichloro-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxa...)
Affinity DataIC50: 6.20E+4nMAssay Description:Evaluated in vitro for inhibitory activity against purified human C1r protease incubated in buffer for 60 minutesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075988(4-Methoxy-N-methyl-N-(4-oxo-4H-benzo[d][1,3]thiazi...)
Affinity DataIC50: 6.25E+4nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075985(3,4-Dichloro-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxa...)
Affinity DataIC50: 6.25E+4nMAssay Description:Evaluated in vitro for inhibitory activity against purified human C1r protease incubated in buffer for 60 minutesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetComplement C1r subcomponent(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075983(N-Methyl-N-(4-oxo-4H-benzo[d][1,3]thiazin-2-yl)-be...)
Affinity DataIC50: 6.25E+4nMAssay Description:In vitro inhibition of purified human C1r protease.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075976(N-Methyl-4-nitro-N-(4-oxo-4H-benzo[d][1,3]oxazin-2...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075982(4-Methoxy-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50063745(2-(2-Iodo-phenylamino)-7-trifluoromethyl-benzo[d][...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075977(4-Cyano-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075978(2-Bromo-N-methyl-N-(4-oxo-4H-benzo[d][1,3]oxazin-2...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSerine protease 1(Human)
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50075988(4-Methoxy-N-methyl-N-(4-oxo-4H-benzo[d][1,3]thiazi...)
Affinity DataIC50: 2.00E+5nMAssay Description:In vitro for inhibition of purified bovine trypsin.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed