Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50003545
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50222968BDBM50222968(Cipralisant | GT-2331)
Affinity DataKi:  0.126nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472544BDBM50472544(Iodoproxyfan)
Affinity DataKi:  0.126nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472544BDBM50472544(Iodoproxyfan)
Affinity DataKi:  0.126nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472543BDBM50472543(CHEMBL278276)
Affinity DataKi:  0.398nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50214615BDBM50214615(CHEBI:64177 | Clobenpropit)
Affinity DataKi:  1nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50214615BDBM50214615(CHEBI:64177 | Clobenpropit)
Affinity DataKi:  1nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50050180BDBM50050180(4-[3-(4-Bromo-benzyloxy)-propyl]-1H-imidazole | CH...)
Affinity DataKi:  1.26nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50050180BDBM50050180(4-[3-(4-Bromo-benzyloxy)-propyl]-1H-imidazole | CH...)
Affinity DataKi:  1.26nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50215536BDBM50215536(CHEBI:73337 | (R)-Alpha-Methylhistamine | CHEMBL26...)
Affinity DataKi:  2.51nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472551BDBM50472551(proxifan | proxyfan)
Affinity DataKi:  3.16nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50127607BDBM50127607(VUF-5296 | 2-(1H-Imidazol-4-yl)-cyclopropylamine |...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472551BDBM50472551(proxifan | proxyfan)
Affinity DataKi:  5nMAssay Description:PKi was measured by Histamine H3 receptor binding assay (N-alpha-MeHA) on rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472556BDBM50472556(CHEMBL428343)
Affinity DataKi:  12.6nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472542BDBM50472542(CHEMBL18554)
Affinity DataKi:  20nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50127605BDBM50127605(VUF-5297 | (1S,2S)-2-(1H-Imidazol-4-yl)-cyclopropy...)
Affinity DataKi:  25nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472547BDBM50472547(CHEMBL19413)
Affinity DataKi:  50.1nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472545BDBM50472545(CHEMBL418736)
Affinity DataKi:  79.4nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472546BDBM50472546(CHEMBL19469)
Affinity DataKi:  100nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472552BDBM50472552(CHEMBL18696)
Affinity DataKi:  100nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472559BDBM50472559(CHEMBL11919 | (S)-Alpha-Methylhistamine)
Affinity DataKi:  158nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472560BDBM50472560(CHEMBL276987)
Affinity DataKi:  158nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472550BDBM50472550(CHEMBL19329)
Affinity DataKi:  199nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472558BDBM50472558(CHEMBL18685)
Affinity DataKi:  199nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472557BDBM50472557(CHEMBL416365)
Affinity DataKi:  251nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472549BDBM50472549(HISTIDINOL | CHEBI:16255)
Affinity DataKi:  251nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472554BDBM50472554(CHEMBL280034)
Affinity DataKi:  316nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472553BDBM50472553(CHEMBL19588)
Affinity DataKi:  1.25E+3nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472548BDBM50472548(CHEMBL418734)
Affinity DataKi:  1.25E+3nMAssay Description:Affinity for histamine H3 receptor in rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
University of Kuopio

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50472555BDBM50472555(CHEMBL18884)
Affinity DataKi: <1.00E+4nMAssay Description:Binding affinity of compound against Histamine H3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed