Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50003544
TargetHistamine H3 receptor(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50127605(VUF-5297 | (1S,2S)-2-(1H-Imidazol-4-yl)-cyclopropy...)
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity was measured against Histamine H3 receptor on rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50121205(CHEBI:18295 | Histamine)
Affinity DataKi:  6.30nMAssay Description:In vitro binding affinity was measured against Histamine H3 receptor on rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetHistamine H3 receptor(Rat)
Vrije Universiteit

Curated by ChEMBL
LigandPNGBDBM50127607(VUF-5296 | 2-(1H-Imidazol-4-yl)-cyclopropylamine |...)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity was measured against Histamine H3 receptor on rat cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed