Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 50003543
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472534(CHEMBL12661)
Affinity DataEC50: >1.00E+3nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472540(CHEMBL12815)
Affinity DataEC50: <0.0100nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataEC50:  10nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472541(CHEMBL273888)
Affinity DataEC50: <0.0100nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataEC50:  23nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472539(CHEMBL12545)
Affinity DataEC50: >1.00E+3nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472535(CHEMBL12296)
Affinity DataEC50: >1.00E+3nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472538(CHEMBL12418)
Affinity DataEC50: <0.0100nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472537(CHEMBL12664)
Affinity DataEC50: <0.0100nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470868(CHEMBL12795)
Affinity DataEC50: >1.00E+3nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472536(CHEMBL276607)
Affinity DataEC50: >1.00E+3nMAssay Description:The functional activity on melatonin receptor was evaluated by its potency to lighten the skin of Xenopus laevis tadpolesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470869(CHEMBL12477)
Affinity DataEC50: >1.00E+3nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470187(CHEMBL428882)
Affinity DataEC50:  0.0370nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470187(CHEMBL428882)
Affinity DataKi:  0.100nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataKi:  0.540nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.700nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472536(CHEMBL276607)
Affinity DataKi:  1.70nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472540(CHEMBL12815)
Affinity DataKi:  3.20nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472541(CHEMBL273888)
Affinity DataKi:  7.60nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470869(CHEMBL12477)
Affinity DataKi:  8.60nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472537(CHEMBL12664)
Affinity DataKi:  9nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472538(CHEMBL12418)
Affinity DataKi:  10nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472534(CHEMBL12661)
Affinity DataKi:  29nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470868(CHEMBL12795)
Affinity DataKi:  37nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472539(CHEMBL12545)
Affinity DataKi:  38nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472535(CHEMBL12296)
Affinity DataKi:  787nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed