Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50036789
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074439BDBM50074439(1-(2-Bromo-4,6-dimethoxy-phenyl)-4,6-dimethyl-1H-p...)
Affinity DataKi:  1nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074411BDBM50074411((2-Bromo-4,6-dimethoxy-phenyl)-(4,6-dimethyl-pyrim...)
Affinity DataKi:  5nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074372BDBM50074372((2-Bromo-4-isopropyl-phenyl)-ethyl-(4-methyl-6-mor...)
Affinity DataKi:  22nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074435BDBM50074435(1-(2-Bromo-4-isopropyl-phenyl)-6-methyl-4-morpholi...)
Affinity DataKi:  28nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074420BDBM50074420(1-(2-Bromo-4,6-dimethoxy-phenyl)-4,6-dimethyl-1H-p...)
Affinity DataKi:  29nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074425BDBM50074425(1-(2-Bromo-4-isopropyl-phenyl)-6-methyl-4-phenyl-1...)
Affinity DataKi:  34nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074429BDBM50074429(1-(2-Bromo-4-isopropyl-phenyl)-6-methyl-4-phenyl-1...)
Affinity DataKi:  36nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074351BDBM50074351((4,6-Dimethyl-pyrimidin-2-yl)-ethyl-(2-iodo-4-isop...)
Affinity DataKi:  38nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074353BDBM50074353(CHEMBL424204 | CHEMBL43216 | (2-Bromo-4,6-dimethox...)
Affinity DataKi:  43nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074350BDBM50074350((2-Bromo-4-isopropyl-phenyl)-(4,6-dimethyl-pyrimid...)
Affinity DataKi:  46nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074437BDBM50074437(1-(2-Bromo-4-isopropyl-phenyl)-4,6-dimethyl-1H-pyr...)
Affinity DataKi:  47nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074432BDBM50074432((4,6-Dimethyl-pyrimidin-2-yl)-(2-iodo-4-isopropyl-...)
Affinity DataKi:  48nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074430BDBM50074430(1-(2-Bromo-4-isopropyl-phenyl)-4-chloro-6-methyl-1...)
Affinity DataKi:  67nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074419BDBM50074419(1-(2-Bromo-4-isopropyl-phenyl)-6-chloro-4-methyl-1...)
Affinity DataKi:  79nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074408BDBM50074408((2-Bromo-4-isopropyl-phenyl)-(4,6-dimethyl-pyrimid...)
Affinity DataKi:  96nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074423BDBM50074423(1-(2-Bromo-4-isopropyl-phenyl)-6-methyl-4-morpholi...)
Affinity DataKi:  112nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074442BDBM50074442(1-(2-Bromo-4-isopropyl-phenyl)-6-methyl-1H-pyrrolo...)
Affinity DataKi:  222nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074427BDBM50074427(1-(2-Bromo-4-isopropyl-phenyl)-4,6-dimethyl-1H-pyr...)
Affinity DataKi:  363nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074417BDBM50074417(1-(2-Bromo-4-isopropyl-phenyl)-6-chloro-4-methyl-1...)
Affinity DataKi:  446nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074440BDBM50074440(1-(2-Bromo-4-isopropyl-phenyl)-4-chloro-6-methyl-1...)
Affinity DataKi:  722nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074418BDBM50074418((2-Bromo-4-isopropyl-phenyl)-(2,6-dimethyl-pyrimid...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074424BDBM50074424(1-(2-Bromo-4-isopropyl-phenyl)-6-methyl-1H-pyrrolo...)
Affinity DataKi:  1.28E+3nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074433BDBM50074433(1-(4-Isopropyl-phenyl)-4,6-dimethyl-1H-pyrrolo[2,3...)
Affinity DataKi:  2.46E+3nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074441BDBM50074441(1-(2-Bromo-4-isopropyl-phenyl)-4,6-dimethyl-1H-pyr...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074426BDBM50074426(1-(2-Bromo-4-isopropyl-phenyl)-4-methyl-1H-pyrrolo...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074438BDBM50074438(1-(2-Bromo-4-isopropyl-phenyl)-4-methyl-1H-pyrrolo...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074421BDBM50074421(1-(2-Bromo-4-isopropyl-phenyl)-4,6-dimethyl-1H-pyr...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074436BDBM50074436((2-Bromo-4-isopropyl-phenyl)-(4,6-dimethyl-pyrimid...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074431BDBM50074431(1-(2-Bromo-4-isopropyl-phenyl)-6-methyl-7-oxy-1H-p...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074416BDBM50074416(1-(2-Bromo-4-isopropyl-phenyl)-6-hydroxy-4-methyl-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074422BDBM50074422(1-(2-Bromo-4-isopropyl-phenyl)-4-methyl-6-phenyl-1...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50074415BDBM50074415(1-(2-Bromo-4-isopropyl-phenyl)-4-methyl-6-phenyl-1...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity was determined against corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2012
Entry Details Article
PubMed