Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 8048
TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231517BDBM231517(US9346818, I-2)
Affinity DataIC50: 80nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231516BDBM231516(US9346818, I-1)
Affinity DataIC50: 86nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 8960BDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 94nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231533BDBM231533(US9346818, I-18)
Affinity DataIC50: 154nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231551BDBM231551(US9346818, I-36)
Affinity DataIC50: 161nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231519BDBM231519(US9346818, I-4)
Affinity DataIC50: 167nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231532BDBM231532(US9346818, I-34 | US9346818, I-17)
Affinity DataIC50: 197nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231532BDBM231532(US9346818, I-34 | US9346818, I-17)
Affinity DataIC50: 202nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231525BDBM231525(US9346818, I-10)
Affinity DataIC50: 239nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231540BDBM231540(US9346818, I-25)
Affinity DataIC50: 249nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231518BDBM231518(US9346818, I-3)
Affinity DataIC50: 269nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231534BDBM231534(US9346818, I-19)
Affinity DataIC50: 376nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231521BDBM231521(US9346818, I-6)
Affinity DataIC50: 483nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231522BDBM231522(US9346818, I-7)
Affinity DataIC50: 486nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231520BDBM231520(US9346818, I-5)
Affinity DataIC50: 502nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231524BDBM231524(US9346818, I-9)
Affinity DataIC50: 601nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231544BDBM231544(US9346818, I-35 | US9346818, I-33 | US9346818, I-2...)
Affinity DataIC50: 601nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231536BDBM231536(US9346818, I-21)
Affinity DataIC50: 653nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231523BDBM231523(US9346818, I-8)
Affinity DataIC50: 658nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231535BDBM231535(US9346818, I-20)
Affinity DataIC50: 706nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231526BDBM231526(US9346818, I-11)
Affinity DataIC50: 889nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231544BDBM231544(US9346818, I-35 | US9346818, I-33 | US9346818, I-2...)
Affinity DataIC50: 903nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231552BDBM231552(US9346818, I-37)
Affinity DataIC50: 905nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231544BDBM231544(US9346818, I-35 | US9346818, I-33 | US9346818, I-2...)
Affinity DataIC50: 950nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231538BDBM231538(US9346818, I-23)
Affinity DataIC50: 959nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231556BDBM231556(US9346818, I-41)
Affinity DataIC50: 990nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231554BDBM231554(US9346818, I-39)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231555BDBM231555(US9346818, I-40)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231553BDBM231553(US9346818, I-38)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231530BDBM231530(US9346818, I-15)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231531BDBM231531(US9346818, I-16)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231528BDBM231528(US9346818, I-13)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231529BDBM231529(US9346818, I-14)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231527BDBM231527(US9346818, I-12)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231541BDBM231541(US9346818, I-26)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231539BDBM231539(US9346818, I-24)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231537BDBM231537(US9346818, I-22)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231546BDBM231546(US9346818, I-31)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231547BDBM231547(US9346818, I-32)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231545BDBM231545(US9346818, I-30)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231542BDBM231542(US9346818, I-27)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

TargetAcetylcholinesterase(Mouse)
Zhejiang Hisun Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 231543BDBM231543(US9346818, I-28)
Affinity DataIC50: 2.00E+3nMAssay Description:Modified Ellman method (Alvin V. et al. JWS-USC-75-IX Improves Information Processing and Cognitive Function in Animal Models[J]. Journal of Pharmaco...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent