Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

LigandChemical structure of BindingDB Monomer ID 645392BDBM645392(US20240016810, Compound TABLE 16.5 | US20240208964...)
Affinity DataIC50: 14nMAssay Description:The biochemical PIKFyve inhibition assays were run by Carna Biosciences according to proprietary methodology based on the Promega ADP-Glo Kinase assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 645392BDBM645392(US20240016810, Compound TABLE 16.5 | US20240208964...)
Affinity DataIC50: 14nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Kineta

US Patent
LigandChemical structure of BindingDB Monomer ID 645392BDBM645392(US20240016810, Compound TABLE 16.5 | US20240208964...)
Affinity DataIC50: 14nMAssay Description:The biochemical PIKfyve inhibition assays were run by Carna Biosciences according to proprietary methodology based on the Promega ADP-Glo™ Kinase ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2025
Entry Details
US Patent

Target1-phosphatidylinositol 3-phosphate 5-kinase(Human)
Kineta

US Patent
LigandChemical structure of BindingDB Monomer ID 645392BDBM645392(US20240016810, Compound TABLE 16.5 | US20240208964...)
Affinity DataIC50: 14nMAssay Description:The biochemical PIKFyve inhibition assays were run by Carna Biosciences according to proprietary methodology based on the Promega ADP-Glo Kinase assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 645392BDBM645392(US20240016810, Compound TABLE 16.5 | US20240208964...)
Affinity DataIC50: 230nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2025
Entry Details
US Patent