Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 25 hits for monomerid = 50381091,50381092,50381093,50381094,50381096,50381097,50381091,50381092,50381093,50381094,50381096,50381097   

TargetTyrosine-protein kinase ITK/TSK(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381096(CHEMBL2017556)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Itk (357-620) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381092(CHEMBL2017552)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Itk (357-620) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381094(CHEMBL2017553)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Itk (357-620) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50381092(CHEMBL2017552)
Affinity DataIC50: 4nMAssay Description:Inhibition of SYK (unknown origin) using FAM-labeled peptide as substrate preincubated for 10 mins followed by substrate addition measured after 25 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2019
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50381092(CHEMBL2017552)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Syk (343 to 635) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381091(CHEMBL2017555)
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Itk (357-620) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381097(CHEMBL2017557)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Itk (357-620) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase ITK/TSK(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381093(CHEMBL2017554)
Affinity DataIC50: 10.9nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Itk (357-620) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation coun...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381096(CHEMBL2017556)
Affinity DataIC50: 39.2nMAssay Description:Inhibition of Lck autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase TXK(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381093(CHEMBL2017554)
Affinity DataIC50: 55.7nMAssay Description:Inhibition of Txk autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381092(CHEMBL2017552)
Affinity DataIC50: 63.9nMAssay Description:Inhibition of Lck autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase TXK(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381094(CHEMBL2017553)
Affinity DataIC50: 66.5nMAssay Description:Inhibition of Txk autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase TXK(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381092(CHEMBL2017552)
Affinity DataIC50: 73.8nMAssay Description:Inhibition of Txk autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase TXK(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381096(CHEMBL2017556)
Affinity DataIC50: 77.5nMAssay Description:Inhibition of Txk autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381093(CHEMBL2017554)
Affinity DataIC50: 162nMAssay Description:Inhibition of Lck autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50381094(CHEMBL2017553)
Affinity DataIC50: 186nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Syk (343 to 635) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381097(CHEMBL2017557)
Affinity DataIC50: 203nMAssay Description:Inhibition of Lck autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase TXK(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381091(CHEMBL2017555)
Affinity DataIC50: 241nMAssay Description:Inhibition of Txk autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50381093(CHEMBL2017554)
Affinity DataIC50: 287nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Syk (343 to 635) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50381096(CHEMBL2017556)
Affinity DataIC50: 358nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Syk (343 to 635) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase TXK(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381097(CHEMBL2017557)
Affinity DataIC50: 441nMAssay Description:Inhibition of Txk autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50381091(CHEMBL2017555)
Affinity DataIC50: 939nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Syk (343 to 635) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381094(CHEMBL2017553)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Lck autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase SYK(Human)
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50381097(CHEMBL2017557)
Affinity DataIC50: 2.47E+3nMAssay Description:Inhibition of recombinant N-terminus His6 tagged Syk (343 to 635) autophosphorylation expressed in insect Sf9 cells using [33P]ATP by scintillation c...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetTyrosine-protein kinase Lck(Human)
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50381091(CHEMBL2017555)
Affinity DataIC50: 3.18E+3nMAssay Description:Inhibition of Lck autophosphorylation using [33P]ATP by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed