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- 7K6H: crystal structure of the first bromodomain (bd1) of human brd4 bound to xmd8-92 (10.1021/ACS.JMEDCHEM.1C01096 )
- 5LRQ: brd4 in complex with erk5 inhibitor xmd8-92 (10.1016/J.EJMECH.2019.05.057 )
- 5BYY: erk5 in complex with small molecule (10.1107/S2059798316004502 )