1811 SMILES Strings for fMet-Leu-Phe receptor

Compound Name
SMILES String
CCN1C(=O)\C(=C2/SC(=S)N(CCCOC)C2=O)c2ccccc12
CCc1nnc(NC(=O)CSc2nnc(-c3cc4ccccc4cc3O)n2CC)s1
CCc1ccccc1NC(=O)C(Cc1cccnc1)C#N
O=C(C1C(N(CC2CCCO2)C(=O)C1=O)c1cccnc1)c1ccco1
O=C(C1C(N(CCc2ccccc2)C(=O)C1=O)c1cccnc1)c1ccco1
COc1cc(ccc1O)C1C(C(=O)c2ccco2)C(=O)C(=O)N1CCc1ccccc1
COc1ccccc1NC(=O)CSc1nnc(Cn2nnc(n2)-c2ccccc2)n1-c1ccccc1
CCOc1cc(ccc1O)C1C(C(=O)c2ccc(C)o2)C(=O)C(=O)N1CCc1ccccc1
C=CCOc1cccc(c1)C1C(C(=O)c2ccco2)C(=O)C(=O)N1CCN1CCOCC1
Clc1ccc(cc1)-c1c[nH]n2c1nc1CCCCc1c2=O
COc1ccccc1C1C(C(=O)c2ccccc2)C(=O)C(=O)N1CC(C)C
Cc1ccc(C)c(c1)C(=O)C1C(N(CCCn2ccnc2)C(=O)C1=O)c1ccncc1
CCc1c(C)nc2c(C#N)c(C)[nH]n2c1=O
COc1cc(ccc1O)C1C(C(=O)c2ccc(C)o2)C(=O)C(=O)N1Cc1cccnc1
COc1ccc(cc1OC)C1C(C(=O)c2ccco2)C(=O)C(=O)N1CCc1ccccc1
CN(C)CCOC(=O)C(O)(C1CCCCC1)c1ccccc1
Cc1cc(SCC(N)=O)nc(SCC(=O)c2ccccc2)n1
CCOc1cccc(c1)C(=O)C1C(N(CCOC)C(=O)C1=O)c1ccc(C)o1
CC(O)CN1C(C(C(=O)c2ccc(C)cc2)C(=O)C1=O)c1ccc(cc1)N(C)C
Cc1[nH]n2c(nc3CCCc3c2=O)c1-c1ccc(Cl)cc1
CC1Oc2ccccc2N(Cc2ccccc2Cl)C1=O
CCOc1cc(ccc1O)C1C(C(=O)c2ccco2)C(=O)C(=O)N1CCc1ccccc1
CCOC(=O)Cc1cc(=O)n2[nH]c(C)c(-c3ccccc3)c2n1
CCOc1cccc(c1)C(=O)C1C(N(Cc2ccco2)C(=O)C1=O)c1ccncc1
COc1cc(ccc1O)C1C(C(=O)c2ccc(C)o2)C(=O)C(=O)N1CCc1ccccc1
O=C(C1C(N(Cc2ccccc2)C(=O)C1=O)c1cccnc1)c1ccco1
O=C(C1C(N(Cc2ccccc2)C(=O)C1=O)c1ccncc1)c1ccco1
COCCCN1C(C(C(=O)c2ccccc2)C(=O)C1=O)c1ccc2OCOc2c1
COc1ccc(CCN2C(C(C(=O)c3ccco3)C(=O)C2=O)c2cccs2)cc1OC
CN(C)c1nc(nc(n1)N(C)C)N(C)C
COc1cccc2C(=O)c3c(O)c4C[C@](O)(C[C@H](O[C@H]5C[C@H](N)[C@H](O)[C@H](C)O5)c4c(O)c3C(=O)c12)C(C)=O
CC1(C)S[C@@H]2[C@H](NC(=O)Cc3ccccc3)C(=O)N2[C@H]1C([O-])=O
N[C@@H](Cc1ccc(O)c(I)c1)C(O)=O
CC1(C)S[C@@H]2[C@H](NC(=O)C(C([O-])=O)c3ccccc3)C(=O)N2[C@H]1C([O-])=O
[H][C@]12CC(C[C@]([H])([C@H]3O[C@@H]13)[N+]2(C)C)OC(=O)[C@H](CO)c1ccccc1
CCCCc1c(O)n(-c2ccccc2)n(-c2ccccc2)c1=O
Oc1c(CCS(=O)c2ccccc2)c(=O)n(-c2ccccc2)n1-c1ccccc1
CCN(CCCc1ccccc1)CCCc1ccccc1
CCOC(=O)c1c(C)[nH]c(C=Nc2ccccc2)c1O |w:11.11|
CCC(=O)Nc1c(C#N)c2nc3ccccc3nc2n1-c1ccccc1C |(15.5,-3.4,;14.73,-2.07,;13.19,-2.07,;12.42,-3.4,;12.42,-.73,;10.88,-.73,;9.98,-1.97,;10.46,-3.44,;10.93,-4.9,;8.52,-1.5,;7.19,-2.27,;5.85,-1.5,;4.48,-2.33,;3.08,-1.53,;3.08,.07,;4.48,.86,;5.85,.04,;7.19,.81,;8.52,.04,;9.98,.51,;10.46,1.97,;9.43,3.12,;9.91,4.58,;11.41,4.9,;12.44,3.75,;11.96,2.29,;12.99,1.14,)|
CCCCn1c(NC(=O)CC)c(C#N)c2nc3ccccc3nc12
CCCCn1c(NC(C)=O)c(C#N)c2nc3ccccc3nc12
CCC(NC(=O)Nc1cc(OC)c(OC)c(OC)c1)(C(F)(F)F)C(F)(F)F
Clc1cccc(c1)C1C(C(=O)c2ccco2)C(=O)C(=O)N1c1ncccn1
OC(=O)C1CC=CCC1C(=O)N1CCN(CC1)c1nc(-c2ccccc2)c2ccccc2n1 |c:5|
COc1ccc(OC)c(c1)C1C(C(=O)c2ccccc2)C(=O)C(=O)N1Cc1ccco1
COc1ccc(OC)c(c1)C1C(C(=O)c2ccco2)C(=O)C(=O)N1CCCN1CCOCC1
COC(=O)c1ccc(cc1)C1C(C(=O)c2ccc(OC)cc2)C(=O)C(=O)N1Cc1ccco1
Cc1ccc(o1)C1C(C(=O)c2cnn(c2C)-c2ccccc2)C(=O)C(=O)N1CCN1CCOCC1
Cc1nc(C)c(s1)C(=O)C1C(N(CCCn2ccnc2)C(=O)C1=O)c1ccc(Cl)cc1
CC(C)OC(=O)C1=C(C)OC(=N)C(C#N)[C@@]11C(=O)N(CC(N)=O)c2ccccc12 |c:6|
COCCCN1C(C(C(=O)c2ccco2)C(=O)C1=O)c1ccc(Br)cc1
COc1ccc(OC)c(c1)C1C(C(=O)c2cc3ccccc3o2)C(=O)C(=O)N1c1cc(C)on1
Cc1cc(no1)N1C(C(C(=O)c2ccc(F)cc2)C(=O)C1=O)c1cccc(Br)c1
O=C(C1C(N(CCCN2CCOCC2)C(=O)C1=O)c1ccccn1)c1cc2ccccc2o1
COc1cccc(C2C(C(=O)c3cc4ccccc4o3)C(=O)C(=O)N2c2cc(C)on2)c1OC
COc1cccc(c1)C1C(C(=O)c2ccc(OC)c(OC)c2)C(=O)C(=O)N1c1cc(C)on1
Cc1cc(no1)N1C(C(C(=O)c2ccc(C)cc2)C(=O)C1=O)c1cccc(Br)c1
CCCOc1ccc(cc1)C1C(C(=O)c2ccco2)C(=O)C(=O)N1CCCn1ccnc1
Cc1c(C)c(=O)oc2c(CN3CCCCC3)c(O)c(Cl)cc12
COCc1cc(ccc1O)C1C(C(=O)c2ccco2)C(=O)C(=O)N1CCOCCO
COc1ccc(cc1)C(=O)C1C(N(C(=O)C1=O)c1nc(C)c(C)s1)c1ccco1
CCOc1ccc(cc1)C(=O)C1C(N(C(=O)C1=O)c1nc(C)c(C)s1)c1ccco1
COc1ccc(CN(C2CCS(=O)(=O)C2)C(=O)c2ccccc2OC)cc1
OCCOCCN1C(C(C(=O)c2cccs2)C(=O)C1=O)c1cccs1
COC(=O)c1[nH]c(C)c(C(=O)C2C(N(CCN3CCOCC3)C(=O)C2=O)c2cccnc2)c1C
COCCCN1C(=O)C(=O)C(C(=O)c2ccc3OCCOc3c2)C11C(=O)N(CC=C)c2ccccc12
CC(C)Oc1ccc(cc1)C1C(C(=O)c2ccc(C)o2)C(=O)C(=O)N1CCCn1ccnc1
Cc1ccc(o1)C1C(C(=O)c2sc(C)nc2C)C(=O)C(=O)N1CCN1CCOCC1
COC(=O)c1[nH]c(C)c(C(=O)C2C(N(CCN3CCOCC3)C(=O)C2=O)c2cccs2)c1C
COc1ccc(cc1OC)-c1c(C)oc2c(CN3CCN(CCO)CC3)c(O)ccc2c1=O
CC1Cc2cc(ccc2O1)C(=O)C1C(N(CCN2CCOCC2)C(=O)C1=O)c1ccccc1F
COc1cc(ccc1O)C1C(C(=O)c2ccc3OC(C)Cc3c2)C(=O)C(=O)N1CCCn1ccnc1
COc1cc(cc(Br)c1O)C1C(C(=O)c2ccco2)C(=O)C(=O)N1c1cc(C)on1
Cc1cc(no1)N1C(C(C(=O)c2ccco2)C(=O)C1=O)c1cccnc1
CCCc1cc(=O)n2[nH]c(C)c(-c3ccccc3)c2n1
COCCCN1C(C(C(=O)c2ccc(OC)cc2C)C(=O)C1=O)c1cccnc1
Cc1[nH]n2c(nc(-c3ccccc3)c(C#N)c2=O)c1-c1ccccc1
Clc1ccc(Cc2nn3c(nnc3s2)-c2ccncc2)cc1
COc1ccc(OC)c(c1)C(=O)c1nc2CCCCCc2n1O
O=S(=O)(Nc1cccc2ncccc12)c1cccs1
Cc1oc2cc(O)cc(O)c2c(=O)c1-c1ccc2OCCCOc2c1
C=CCn1c(NC(=O)c2ccccc2)c(C#N)c2nc3ccccc3nc12
O=C(Cn1c2ccccc2oc1=O)N1CCN(CC1)c1ccccc1
Cc1nn(c(C)c1Oc1ccccc1O)-c1nc2ccccc2s1
CCOC(=O)Nc1ccc(OC)cc1S(=O)(=O)N1CCCCC1
CC1=NC(C)=C(C#N)C(C1C#N)c1ccc2ncccc2c1 |t:1,4|
COCCCN1C(C(C(=O)c2ccco2)C(=O)C1=O)c1ccccc1
FC(F)(F)C1(NC(=O)NCCN2CCOCC2)Oc2ccc(Cl)cc2O1
COc1ccc(C2C(C(=O)c3ccccc3)C(=O)C(=O)N2CC(C)O)c(OC)c1
COc1ccc(cc1OC)-c1cc(nc(n1)N1CCN(Cc2ccccc2)CC1)C(F)(F)F
COc1ccc(cc1NC(=O)C1CCCC1)-c1cn2cccnc2n1
COc1ccc(cc1)-c1nnc(Nc2nc3c(OC)cccc3s2)o1
CC(C)OC(=O)c1nnn(c1CN1CCc2ccccc2C1)-c1nonc1N
Nc1nc(CSc2nc(cc(c2C#N)C(F)(F)F)-c2ccccc2)nc(n1)N1CCOCC1
COc1ccc(cc1NC(=O)C1CC1)-c1cn2cccnc2n1
COC(=O)C1O[N+]([O-])=C(C1c1c[nH]c2ccccc12)C(=O)OC |c:7|
Nc1ccc(Nc2ccccc2N)cc1
Fc1ccc(cc1)-n1ncc2c1ncn(CC(=O)OCc1ccccc1)c2=O
COc1ccc(-c2nnc(Nc3nc4c(OC)cccc4s3)o2)c(OC)c1
CCCS(=O)(=O)N1CCCC(C1)C(=O)N1CCC(Cc2ccccc2)CC1
CN1CCN(CCCNC(=O)Nc2cccc3ccccc23)CC1
CCC(Sc1nc2CCCc2c(=O)[nH]1)C(=O)Nc1cccc(OC)c1
CCC(CCC(=O)Nc1cccc(c1)C(O)=O)C(O)=O
O=C(NC1CCCC1)c1sc(=S)n2c1[nH]c(=O)c1ccccc21
Fc1ccc(Cn2c(=O)cc([nH]c2=O)N2CCc3ccccc23)cc1
COc1ccc(cc1OC)-c1cc(nc(n1)N1CCN(CC1)c1ccccc1)C(F)(F)F
Fc1ccc(cc1)N1CCN(CCCNC(=O)c2cccc(c2)N2CCCC2=O)CC1
COc1ccc(cc1)-c1nc([nH]c(=O)c1C#N)N1CCCC1
O=S(=O)(N1CCc2ccccc12)c1c[nH]cn1
COc1ccccc1C1C(C(=O)c2ccccc2)C(=O)C(=O)N1CCO
CCOC(=O)N1CCC(CC1)NC(=O)c1cc(ccc1CO)C(=O)Nc1ccc(OC)c(OC)c1
CCN(CC)c1ccc(C=NC(C#N)C(=N)C#N)cc1 |w:10.10|
O=C1CCCC(=O)C1C(C#Cc1ccccc1)C1C(=O)CCCC1=O
O=C(NC1CCCCC1)c1sc(=S)n2c1[nH]c(=O)c1ccccc21
CC1CCN(CC1)c1nc(-c2ccccc2)c(C#N)c(=O)[nH]1
CCSc1nnc(NC(=O)CSc2nnc(Cc3cccn3C)n2CCc2ccccc2)s1
COc1ccccc1C1C(C(=O)c2ccccc2)C(=O)C(=O)N1CC(C)O
CN(C)c1ccc(cc1)\N=C1/C(C)=C(C#N)C(=O)N(CCCO)C1=O |t:13|
COc1ccc(cc1OC)-c1cc(nc(n1)N1CCCCC1)C(F)(F)F
OC(=O)CCCNc1cc(N2CCC3(CC2)OCCO3)c2noc3-c4ccccc4C(=O)c1c23
Cc1ccc(cc1)C1C2C(=O)CC(C)(C)CC2=Nc2[nH]c(=S)[nH]c(=O)c12 |c:18|
Cc1ccc(C)c(c1)-n1c(CNC(=O)c2ccco2)nnc1SCC(=O)N1CCc2ccccc12 |(7.19,4.55,;8.73,4.54,;9.5,5.88,;11.04,5.87,;11.81,4.54,;13.35,4.54,;11.04,3.21,;9.5,3.21,;11.8,1.87,;13.34,1.71,;14.37,2.85,;15.87,2.53,;16.91,3.67,;16.43,5.14,;18.41,3.35,;19.04,1.94,;20.57,2.1,;20.89,3.6,;19.56,4.38,;13.65,.2,;12.32,-.57,;11.18,.47,;9.67,.15,;9.19,-1.32,;7.68,-1.63,;6.65,-.49,;7.2,-3.1,;8.1,-4.34,;7.2,-5.58,;5.75,-5.11,;4.41,-5.88,;3.08,-5.11,;3.08,-3.57,;4.41,-2.8,;5.75,-3.57,)|
CCOC(=O)c1ccc(NC(=O)Nc2ccc3N(CC)C(=O)c4cccc2c34)cc1
[H]C12CC(C)(NC(=O)C1C(=O)Nc1ccc(OC)cc1)Oc1ccccc21 |THB:9:8:2:20.26.21,25:26:2:5.8.6|
CSCCC1C(C#N)C(=N)Oc2[nH]nc(-c3cccs3)c12
CCCCNC(=O)c1sc(=S)n2c1[nH]c(=O)c1ccccc21
COc1ccc(NC(=O)C(N(C)C(=O)c2cnccn2)c2ccc(C)cc2)cc1
CCOc1cc(cc(OCC)c1OCC)C(=O)NCc1nnc(SCC(=O)OC)n1C
CCOC(=O)c1sc(=S)n2c1[nH]c(=O)c1ccc(cc21)C(=O)OC
CCOC(=O)CCn1nc(cc1N)-c1ccc(Cl)cc1
CNc1nn(nc1N)-c1cccc(Cl)c1
Cc1csc(NC(=O)CCn2c3ccccc3oc2=O)n1
O=C(NCc1cccnc1)C1N(C2CCCCCC2)C(=O)c2ccccc12
CN(C)c1ccc(cc1)\N=C1/C(C)=C(C#N)C(=O)N(C)C1=O |t:13|
COc1ccc(Cl)cc1-n1c2nc(SCC(=O)NCC3CCCO3)[nH]c(=O)c2sc1=S |(22.17,.5,;20.66,.18,;19.63,1.33,;20.11,2.79,;19.08,3.94,;17.57,3.62,;16.54,4.77,;17.09,2.16,;18.12,1.01,;17.64,-.45,;16.19,-.92,;14.85,-.15,;13.52,-.92,;12.19,-.15,;10.85,-.92,;9.52,-.15,;9.52,1.39,;8.18,-.92,;6.85,-.15,;5.52,-.92,;5.36,-2.45,;3.85,-2.77,;3.08,-1.44,;4.11,-.29,;13.52,-2.46,;14.85,-3.23,;14.85,-4.77,;16.19,-2.46,;17.64,-2.93,;18.54,-1.69,;20.08,-1.69,)|
COc1ccc2nc(Nc3nc(C)c(s3)C(C)=O)sc2c1
COCCN1Cc2cccc(C(=O)NCc3ccc4OCOc4c3)c2C1=O
CCOc1ccccc1NC(=O)CSc1nccn1-c1ccccc1
[H]C12CCC([H])(O1)C(C2C(O)=O)C(=O)Nc1cc(cc(c1)C(=O)OC(C)C)C(=O)OC(C)C |TLB:12:7:6:3.2,THB:9:8:6:3.2|
O=C(NCc1cccnc1)C1N(C2CCCCCCC2)C(=O)c2ccccc12
COc1ccc(cc1OC)-c1nc(no1)-c1ccc(NC(=O)c2ccc(Br)o2)cc1
COC(=O)Cc1n[nH]c2OC(=N)C(C#N)C(C3CCCC=C3)c12 |c:20|
[H]C12CC(C)(Oc3ccccc13)N(CCO)C(=O)C2C(=O)Nc1ccc(C)cc1 |TLB:13:12:2:5.11.6,THB:10:11:2:12.18.16,19:18:2:5.11.6|
COc1cccc(OC)c1C(=O)C(C#N)c1nc2ccccc2[nH]1
COC(=O)[C@H](C(C)C)n1c(C)c(C(C)=O)c(C(C)=O)c1C
Clc1ccccc1-c1nnc(NC(=O)c2ccc(cc2)S(=O)(=O)N2CCCCCC2)o1
COc1ccccc1-n1c(CNC(=O)c2ccco2)nnc1SCC(=O)Nc1ccc(F)cc1 |(7.82,-2.09,;9.15,-1.32,;10.49,-2.09,;10.49,-3.63,;11.82,-4.4,;13.15,-3.63,;13.15,-2.09,;11.82,-1.32,;11.82,.22,;10.57,1.13,;9.11,.65,;7.97,1.68,;6.5,1.21,;6.18,-.3,;5.36,2.24,;5.52,3.77,;4.11,4.4,;3.08,3.25,;3.85,1.92,;11.05,2.59,;12.59,2.59,;13.07,1.13,;14.53,.65,;15.68,1.68,;17.14,1.21,;17.46,-.3,;18.28,2.24,;19.75,1.76,;20.07,.26,;21.53,-.22,;22.68,.81,;24.14,.33,;22.36,2.32,;20.89,2.79,)|
Oc1nc(sc1C(=C)c1ccc(Br)cc1)N1CCCC1
Cc1c(oc2ccc(cc12)S(=O)(=O)N1CCOCC1)C(=O)NC1CCCc2ccccc12
CCC(CC)C(=O)Nc1n(-c2ccccc2)c(=O)nc2n(ncc12)-c1ccccc1
Cc1ccccc1Nc1cc2ccccc2c(=O)[nH]1
CCc1nn2c(nc(CSc3nc4sc5CCCCc5c4c(=O)n3C)cc2=O)s1
CCC(C)(N(CC1CCCO1)C(=O)c1ccc2OCOc2c1)C(=O)NC1CCCC1
CCn1cc(C(=O)NC2CCC(C)CC2)c(=O)c2cc(ccc12)S(=O)(=O)N1CCCCC1 |(11.08,4.26,;12.42,3.49,;12.42,1.95,;11.08,1.18,;11.08,-.36,;9.75,-1.13,;9.75,-2.67,;8.41,-.36,;7.08,-1.13,;7.08,-2.67,;5.75,-3.44,;4.41,-2.67,;3.08,-3.44,;4.41,-1.13,;5.75,-.36,;12.42,-1.13,;12.42,-2.67,;13.75,-.36,;15.13,-1.18,;16.52,-.39,;16.52,1.21,;15.13,2,;13.75,1.18,;17.85,-1.17,;18.63,.16,;17.08,-2.5,;19.18,-1.94,;19.18,-3.48,;20.51,-4.26,;21.84,-3.49,;21.85,-1.95,;20.52,-1.18,)|
COC(=O)C1(CC1)S(=O)(=O)c1cccc2nsnc12
Cc1c(CNCc2cccs2)c(C(O)=O)c(C)n1Cc1ccccc1
CCN(C(=O)Cc1c([nH]c2ccccc12)C(O)=O)c1cc(OC)ccc1OC
CCOC(=O)CSc1nnc(CNC(=O)c2cc(OCC)c(OCC)c(OCC)c2)n1C
COc1ccc(cc1NC(=O)CC(C)C)-c1cn2cccnc2n1
CCC(SC1=Nc2ccccc2C2=NC(CC(C)C)C(=O)N12)C(=O)Nc1ccc2OCOc2c1 |t:4,13|
COc1ccc(cc1OC)-c1cc(nc(NC2CCCC2)n1)C(F)(F)F
Cc1c(oc2ccc(cc12)S(=O)(=O)N1CCOCC1)C(=O)Nc1ccc(C)c(C)c1
CCCC(=O)Nc1c2CS(=O)Cc2nn1-c1ccc(OC)cc1
Cc1cccc(c1C)-n1nc2CSCc2c1NC(=O)c1ccco1
CCCCCNC(=O)c1ccc2c(c1)n1c([nH]c2=O)c(sc1=S)C(=O)NCC1CCCO1
CCOC(=O)N1CCN(CC1)c1cc(NCCC(O)=O)c2C(=O)c3ccccc3-c3onc1c23
CC(=O)SCC(=O)N=c1sc2cc(F)ccc2n1C |w:7.6|
CCCC(=O)Nc1cc(ccc1OC)-c1cn2cccnc2n1
O=C(C1C(N(CCN2CCOCC2)C(=O)C1=O)c1ccccc1)c1cccs1
CCOC(=O)C1CCN(Cc2ccc(cc2)C(=O)OC)CC1
Cc1nnc(SCc2cnc(o2)-c2ccccc2)[nH]c1=O
COc1ccccc1Oc1c(C)oc2cc(OC(=O)c3ccco3)ccc2c1=O
COc1ccccc1-c1c(C)oc2cc(OC(=O)c3ccco3)ccc2c1=O |(3.08,1.74,;4.41,.97,;4.41,-.57,;3.08,-1.34,;3.08,-2.88,;4.41,-3.65,;5.75,-2.88,;5.75,-1.34,;7.08,-.57,;7.08,.97,;5.75,1.74,;8.41,1.74,;9.75,.97,;11.13,1.8,;12.52,1,;13.85,1.78,;15.19,1.01,;15.19,-.53,;16.52,1.79,;16.67,3.32,;18.18,3.65,;18.95,2.32,;17.93,1.17,;12.52,-.6,;11.13,-1.39,;9.75,-.57,;8.41,-1.34,;8.41,-2.88,)|
CCCOc1ccc(cc1)C1C(C(=O)c2ccc(C)o2)C(=O)C(=O)N1CCCn1ccnc1
OCc1nc2ccccc2n1CC(O)Cn1ccc2ccccc12
C=CCOc1ccc(cc1)C1C(C(=O)c2ccco2)C(=O)C(=O)N1Cc1cccnc1
Cc1c(oc2cc(C)c(C)cc12)C(=O)NC1CCS(=O)(=O)C1
Clc1ccc(cc1)C(=O)N(Cc1cccs1)C1CCS(=O)(=O)C1
O=C(NC1CCCC1)C1CC1c1ccccc1
COc1ccc(C)cc1NC(=O)C1CCCCC1C(O)=O
COc1cc(c(Cl)c(Br)c1O)-n1nc(C)c2C(C(C#N)C(=N)Oc12)c1ccccc1
COc1ccc(OC)c(c1)C1C(C(=O)c2cccs2)C(=O)C(=O)N1c1cc(C)on1
O=c1cc(nc([nH]1)N1CCN(Cc2ccccc2)CC1)-c1ccccc1
Cc1cccc(OCC(=O)Nc2cc(C)ccc2O)c1
CCCOc1ccc(cc1)C1C(C(=O)c2ccc(C)o2)C(=O)C(=O)N1Cc1cccnc1
CCOc1ccc(cc1)C1C(C(=O)c2ccco2)C(=O)C(=O)N1Cc1cccnc1
CC(C)CN(CC(C)C)C(=O)CS(=O)(=O)Cc1ccccc1
COc1ccc(CC(=O)Nc2ccc(cc2)-c2nnc(o2)-c2ccc(C)cc2)cc1
OC(=O)C1CCCCC1C(=O)Nc1ccc(cc1)C(=O)NCC1CCCO1
COc1cc2\C(C(=O)N3c2c(c1)C(C)=CC3(C)C)=C1\SC(NC(C)=O)=NC1=O |c:15,27|
CCCc1nc2ccccc2c3n1nc(n3)N
[H]C12CCC([H])(C1)C(C2C(O)=O)C(=O)Nc1ccc(OC)c(OC)c1 |TLB:12:7:6:3.2,THB:9:8:6:3.2|
CSc1ccccc1NS(=O)(=O)c1ccccc1
CCOC(=O)Cc1cc(=O)n2[nH]c(C)c(-c3ccc(OC)cc3)c2n1
COc1ccc(cc1)S(=O)(=O)NC(C)C(=O)Nc1cccc(c1)C(C)=O
COCCCN1C(C(C(=O)c2ccc3OC(C)Cc3c2)C(=O)C1=O)c1cccnc1
CCOc1ccc(cc1)C1C(C(=O)c2ccco2)C(=O)C(=O)N1CCCn1ccnc1
COc1ccc2cnn(-c3ccccc3)c(=O)c2c1OC
Cc1[nH]n2c(nc3CCCc3c2=O)c1-c1ccccc1
COc1cccc2cc(oc12)C(=O)C1C(N(Cc2ccco2)C(=O)C1=O)c1cccnc1
Cc1ccc(o1)C(=O)C1C(N(Cc2ccccc2)C(=O)C1=O)c1cccnc1
COC(=O)c1[nH]c(C)c(C(=O)C2C(N(CCCN3CCOCC3)C(=O)C2=O)c2ccccn2)c1C
COc1cccc(c1)-c1nc(CS(=O)(=O)CC(=O)NCCC(C)C)c(C)o1
CCCCSc1nc(O)cc(=O)n1CC=C
OC(=O)CC1Oc2ccc(Cl)cc2NC1=O
CCOC(=O)c1c(NC(=O)c2cc(on2)C2CC2)sc2CCCCc12
CCCNC(=O)CS(=O)(=O)Cc1nc(oc1C)-c1cccc(OC)c1
Cc1ccsc1C1C2C(=O)CC(C)(C)CC2=Nc2ncnn12 |c:17|
COc1ccc2ccccc2c1C1CC(=O)N2CN(CSC2=C1C#N)C1CCCCC1 |c:24|
CC1CCN(CC1)S(=O)(=O)c1ccc2n(CC(=O)NCc3ccc4OCOc4c3)c(=O)oc2c1
COc1ccc(cc1)-n1c(Cc2cccn2C)nnc1SCC(=O)Nc1ccc(Cl)cc1
CN1CCN(CC1)c1cc(NCCOC(C)=O)c2C(=O)c3ccccc3-c3onc1c23
CC(CCc1ccco1)NC(=O)CCc1c(C)nc2c(c(C)nn2c1C)-c1ccc(F)cc1
Cc1ccc(NC(=O)C2CCCN2S(=O)(=O)c2cccc3cccnc23)cc1F
Cc1cccc(c1)C1CC(Nc2nc(N)nn12)c1ccc(Cl)cc1
Cc1ccc(Nc2nc(cs2)C2CC2)cc1
COc1ccc(cc1OC)-c1nc(no1)-c1ccc(Br)o1
Clc1ccc(cc1Cl)C1CC(c2cccs2)n2ncnc2N1
Fc1ccc(cc1)-c1nnc2ccc(nn12)N1CCCC1
Cc1cc(NC(=O)CSc2nnc(Cn3c4ccccc4sc3=O)n2-c2ccccc2C)no1 |(21.13,4.72,;19.62,4.4,;18.99,2.99,;17.46,3.16,;16.43,2.01,;14.92,2.34,;14.45,3.8,;13.89,1.19,;12.38,1.52,;11.35,.37,;11.67,-1.13,;10.33,-1.9,;9.19,-.87,;7.68,-1.19,;7.2,-2.65,;5.75,-3.12,;4.41,-2.35,;3.08,-3.12,;3.08,-4.66,;4.41,-5.43,;5.75,-4.66,;7.2,-5.13,;8.1,-3.89,;9.64,-3.89,;9.82,.54,;9.05,1.87,;7.51,1.87,;6.74,3.21,;7.52,4.54,;9.06,4.54,;9.82,3.2,;11.36,3.2,;17.14,4.66,;18.48,5.43,)|
Brc1ccc(o1)C(=O)Nc1ccc(Nc2ccccc2)cc1
[H]C12[#6]-[#6]C([H])([#6](-[#6]1-[#6](-[#8])=O)-[#6](=O)-[#7]-c1cc(-[#8]-[#6])ccc1-[#8]-[#6])\[#6]2=[#6](\[#6])-[#6] |TLB:11:6:24:3.2,THB:8:7:24:3.2|
COC(=O)COc1ccc2c(c1)oc(C)c(Oc1ccccc1)c2=O
COCCCN1C(C(C(=O)c2ccco2)C(=O)C1=O)c1cccc(Br)c1
CCOc1ccc(cc1)C(=O)C1C(N(CC2CCCO2)C(=O)C1=O)c1ccc(C)o1
Cc1ccc(cc1)C(=O)C1C(N(CCN2CCOCC2)C(=O)C1=O)c1cccnc1
Cc1ccc(o1)C1C(C(=O)c2ccc(Cl)cc2)C(=O)C(=O)N1CC1CCCO1
COc1ccc2c(c1)oc(C)c(N1C(=O)c3ccccc3C1=O)c2=O
Cc1ccc(F)c(NC(=O)C2CCCCC2C(O)=O)c1
Clc1ccc(cc1Cl)C1C(C(=O)c2ccco2)C(=O)C(=O)N1c1ncccn1
COc1ccc(cc1OC)C1C(C(=O)c2cccs2)C(=O)C(=O)N1c1nnc(C)s1
CCOC(=O)c1oc2cc(O)ccc2c(=O)c1-c1ccccc1OC |(4.41,5.39,;4.41,3.85,;5.75,3.08,;5.75,1.54,;4.41,.77,;7.08,.77,;8.41,1.54,;9.75,.77,;11.13,1.59,;12.52,.8,;13.85,1.58,;12.52,-.8,;11.13,-1.59,;9.75,-.77,;8.41,-1.54,;8.41,-3.08,;7.08,-.77,;5.75,-1.54,;4.41,-.77,;3.08,-1.54,;3.08,-3.08,;4.41,-3.85,;5.75,-3.08,;7.08,-3.85,;7.08,-5.39,)|
CN1C(=O)\C(=C2/SC(=S)N(C(CCC(O)=O)C(O)=O)C2=O)c2ccccc12
COc1cc(cc(OC)c1OC)C1C(C(=O)c2cccs2)C(=O)C(=O)N1Cc1ccco1
COc1ccc(cc1OC)C1C(C(=O)c2ccco2)C(=O)C(=O)N1Cc1cccnc1
COc1ccc(cc1)C(=O)C1C(N(CCN2CCOCC2)C(=O)C1=O)c1ccc(C)cc1
O=C1Nc2ccccc2\C1=C1\SC(=S)N(CC2CCCO2)C1=O
COCCN1C(C(C(=O)c2ccco2)C(=O)C1=O)c1cccc(Oc2ccccc2)c1
Cc1ccc(o1)C1C(C(=O)c2ccc(Br)cc2)C(=O)C(=O)N1Cc1ccco1
Cc1nnc(s1)N1C(C(C(=O)c2cccs2)C(=O)C1=O)c1ccc(OCC=C)cc1
CCOc1cccc(c1)C(=O)C1C(N(Cc2cccnc2)C(=O)C1=O)c1ccco1
Cc1nc2c(c[nH]n2c(=O)c1Cc1ccccc1)C#N
Cc1[nH]n2c(nc(C)c(Cc3ccccc3)c2=O)c1C#N
CCOC(=O)Cc1cc(=O)n2[nH]c(C)c(-c3ccc(Cl)cc3)c2n1
COc1cccc(c1)C(=O)C1C(N(Cc2cccnc2)C(=O)C1=O)c1ccco1
[H]C12CC3([H])CC([H])(C1)CC(C2)(C3)c1c(O)n(-c2ccccc2)n(-c2ccccc2)c1=O |TLB:8:1:12:6.9.5,8:6:12:1.11.2,THB:2:1:9:3.12.5,2:3:9:1.11.8|
O=C(C1C(N(Cc2ccccc2)C(=O)C1=O)c1ccco1)c1ccco1
CCOc1ccc(cc1)C(=O)C1C(N(CC2CCCO2)C(=O)C1=O)c1ccco1
Cc1[nH]n2c(nc(cc2=O)-c2ccc(cc2)[N+]([O-])=O)c1-c1ccccc1
Clc1ccc(cc1)C1C(C(=O)c2ccco2)C(=O)C(=O)N1c1ncccn1
[H]C12CCC([H])(O1)C(C2C(O)=O)C(=O)Nc1cc(cc(c1)C(=O)OCC)C(=O)OCC |TLB:12:7:6:3.2,THB:9:8:6:3.2|
COc1ccc2c(c1)oc(C)c(-c1cnn(c1)-c1ccccc1)c2=O
OC(=O)C1CCCCC1C(=O)Nc1ccccc1Cl
CCCNC(=S)Nc1ccc(Nc2ccccc2)cc1
c1ccc(cc1)Nc2ccc(cc2)N
CCCOc1ccc2c(c1)oc(C)c(N1C(=O)c3ccccc3C1=O)c2=O
Cc1ccc(Nc2ccc(cc2N)C(O)=O)cc1
Cc1[nH]n2c(nc3CCCc3c2=O)c1-c1cccc2ccccc12 |(8.07,-3.45,;8.84,-2.12,;10.36,-1.96,;10.68,-.47,;9.35,.3,;9.35,1.84,;10.68,2.61,;11,4.11,;12.53,4.27,;13.15,2.87,;12.01,1.84,;12.01,.3,;13.35,-.47,;8.21,-.72,;6.71,-.4,;6.23,1.06,;4.72,1.38,;3.69,.23,;4.17,-1.23,;3.08,-2.41,;3.57,-3.94,;5.14,-4.27,;6.2,-3.07,;5.68,-1.55,)|
CC(C)(C)CC(=O)Nc1ccc(Nc2ccccc2)cc1
O=C(C1C(N(Cc2ccco2)C(=O)C1=O)c1ccccc1)c1cccs1
CCc1cc2c(cc1OC(=O)C(C)(C)C)oc(COCC(O)=O)c(-c1nc3ccccc3n1C)c2=O |(15.91,-4.32,;15.92,-2.78,;14.59,-2,;13.19,-2.79,;11.82,-1.97,;11.82,-.43,;13.19,.4,;14.59,-.4,;15.92,.38,;15.91,1.92,;14.58,2.68,;17.24,2.69,;18.57,3.47,;16.47,4.02,;18.02,1.36,;10.48,.34,;9.15,-.43,;7.82,.34,;7.82,1.88,;6.48,2.65,;6.48,4.19,;5.15,4.96,;7.82,4.96,;9.15,-1.97,;7.82,-2.74,;6.42,-2.11,;5.39,-3.25,;3.85,-3.25,;3.08,-4.58,;3.85,-5.92,;5.39,-5.92,;6.16,-4.58,;7.66,-4.26,;8.8,-5.29,;10.48,-2.74,;10.48,-4.28,)|
Cc1nc2c(C)cccn2c1C(=O)C1C(N(CCN2CCOCC2)C(=O)C1=O)c1cccs1
COCCN1C(C(C(=O)c2cccs2)C(=O)C1=O)c1ccccc1
COc1ccccc1Oc1c(C)oc2c(CN(C)C)c(O)ccc2c1=O
COc1ccc(cc1)C(=O)C1C(N(Cc2ccco2)C(=O)C1=O)c1ccc(OC)cc1OC
CCOc1ccccc1Oc1c(C)oc2cc(OC(=O)c3ccco3)ccc2c1=O
Cc1cccc(Nc2ccccc2C(=O)NCc2ccco2)c1C
CCOc1ccc(cc1)C1C(C(=O)c2cccs2)C(=O)C(=O)N1CCCn1ccnc1
Cc1sc(NC(=O)C2CCCCC2C(O)=O)c(C(N)=O)c1-c1ccc(cc1)C(C)(C)C
[H]C12CCC([H])(O1)C(C2C(O)=O)C(=O)Nc1sc(C)c(c1C(=O)OCC)-c1ccc(C)cc1 |TLB:12:7:6:3.2,THB:9:8:6:3.2|
[H]C12CCC([H])(O1)C(C2C(O)=O)C(=O)Nc1scc(c1C(=O)OCC)-c1ccc(cc1)-c1ccccc1 |TLB:12:7:6:3.2,THB:9:8:6:3.2|
CCCCCCN1C(C(C(=O)c2ccccc2)C(=O)C1=O)c1ccc(O)c(OC)c1
COc1ccccc1-c1c(oc2cc(OC(=O)c3ccco3)ccc2c1=O)C(F)(F)F |(7.08,-4.42,;7.08,-2.88,;5.75,-2.11,;4.41,-2.88,;3.08,-2.11,;3.08,-.57,;4.41,.2,;5.75,-.57,;7.08,.2,;7.08,1.74,;8.41,2.51,;9.75,1.74,;11.13,2.57,;12.52,1.77,;13.85,2.55,;15.19,1.78,;15.19,.24,;16.52,2.56,;16.67,4.09,;18.18,4.42,;18.95,3.09,;17.93,1.94,;12.52,.17,;11.13,-.62,;9.75,.2,;8.41,-.57,;8.41,-2.11,;5.75,2.51,;4.41,3.28,;6.52,3.85,;4.98,1.18,)|
OC(=O)C1CCCCC1C(=O)Nc1ccc(Br)cc1
CCc1cc2c(cc1OC(C)=O)oc(C)c(-c1nc3ccccc3n1C)c2=O |(15.91,-2.7,;15.92,-1.16,;14.59,-.39,;13.19,-1.18,;11.82,-.36,;11.82,1.18,;13.19,2.01,;14.59,1.22,;15.92,1.99,;15.91,3.53,;17.24,4.31,;14.58,4.3,;10.48,1.95,;9.15,1.18,;7.82,1.95,;9.15,-.36,;7.82,-1.13,;6.42,-.5,;5.39,-1.64,;3.85,-1.64,;3.08,-2.97,;3.85,-4.31,;5.39,-4.31,;6.16,-2.97,;7.66,-2.65,;8.8,-3.68,;10.48,-1.13,;10.48,-2.67,)|
COCCN1C(C(C(=O)c2ccccc2)C(=O)C1=O)c1ccccc1OC
COCCN1C(C(C(=O)c2ccccc2)C(=O)C1=O)c1cc(OC)ccc1OC
COCCN1C(C(C(=O)c2ccccc2)C(=O)C1=O)c1ccc(cc1)C(C)C
COc1ccc(C2C(C(=O)c3ccccc3)C(=O)C(=O)N2c2cccc(Cl)c2)c(OC)c1
COc1ccc(OC)c(c1)C1C(C(=O)c2ccccc2)C(=O)C(=O)N1c1ccc(C)c(Cl)c1
CC(C)c1ccc(cc1)C1C(C(=O)c2ccccc2)C(=O)C(=O)N1Cc1cccnc1
COc1ccc(OC)c(c1)C1C(C(=O)c2ccccc2)C(=O)C(=O)N1c1cccnc1
COc1ccc(cc1OC)-c1c(oc2cc(OC(=O)c3cccnc3)ccc2c1=O)C(F)(F)F
COc1ccc(cc1OC)-c1c(oc2cc(OC(=O)c3ccco3)ccc2c1=O)C(F)(F)F
COc1ccc(cc1OC)-c1c(oc2c(CN3CCOCC3)c(O)ccc2c1=O)C(F)(F)F
FC(F)(F)c1oc2cc(OC(=O)c3ccco3)ccc2c(=O)c1-c1ccccc1Cl |(4.41,2.51,;5.75,1.74,;6.52,3.08,;4.98,.41,;7.08,.97,;8.41,1.74,;9.75,.97,;11.13,1.8,;12.52,1,;13.85,1.78,;15.19,1.01,;15.19,-.53,;16.52,1.79,;17.93,1.17,;18.95,2.32,;18.18,3.65,;16.67,3.32,;12.52,-.6,;11.13,-1.39,;9.75,-.57,;8.41,-1.34,;8.41,-2.88,;7.08,-.57,;5.75,-1.34,;4.41,-.57,;3.08,-1.34,;3.08,-2.88,;4.41,-3.65,;5.75,-2.88,;7.08,-3.65,)|
FC(F)(F)c1oc2cc(OC(=O)c3cccs3)ccc2c(=O)c1-c1ccccc1Cl |(4.41,2.51,;5.75,1.74,;6.52,3.08,;4.98,.41,;7.08,.97,;8.41,1.74,;9.75,.97,;11.13,1.8,;12.52,1,;13.85,1.78,;15.19,1.01,;15.19,-.53,;16.52,1.79,;17.93,1.17,;18.95,2.32,;18.18,3.65,;16.67,3.32,;12.52,-.6,;11.13,-1.39,;9.75,-.57,;8.41,-1.34,;8.41,-2.88,;7.08,-.57,;5.75,-1.34,;4.41,-.57,;3.08,-1.34,;3.08,-2.88,;4.41,-3.65,;5.75,-2.88,;7.08,-3.65,)|
FC(F)(F)c1oc2cc(OC(=O)c3cccs3)ccc2c(=O)c1Oc1ccccc1Br
COc1ccc(C2C(C(=O)c3cccs3)C(=O)C(=O)N2CCN2CCOCC2)c(OC)c1
COc1ccc(C2C(C(=O)c3ccco3)C(=O)C(=O)N2CCN2CCOCC2)c(OC)c1
COc1ccc(C2C(C(=O)c3ccccc3)C(=O)C(=O)N2CCCn2ccnc2)c(OC)c1
COc1ccc(cc1)C1C(C(=O)c2cccs2)C(=O)C(=O)N1CCCn1ccnc1
O=C(C1C(N(CCCn2ccnc2)C(=O)C1=O)c1cccnc1)c1ccco1
COc1ccc(cc1OC)C1C(C(=O)c2ccco2)C(=O)C(=O)N1CCCN1CCOCC1
CC(C)c1ccc(cc1)C1C(C(=O)c2ccc(C)cc2)C(=O)C(=O)N1c1nnc(C)s1
COCCCN1C(C(C(=O)c2ccccc2)C(=O)C1=O)c1ccc(cc1)C(C)C
COCCCN1C(C(C(=O)c2ccccc2)C(=O)C1=O)c1ccc(O)c(OC)c1
COc1ccc(OC)c(c1)C1C(C(=O)c2ccc(C)cc2)C(=O)C(=O)N1CCC(O)=O
COc1ccc(cc1OC)C1C(C(=O)c2cc3ccccc3o2)C(=O)C(=O)N1CCN(C)C
COc1cc(ccc1O)C1C(C(=O)c2cc3ccccc3o2)C(=O)C(=O)N1CCN(C)C
O=C(C1C(N(CCCN2CCOCC2)C(=O)C1=O)c1cccnc1)c1cc2ccccc2o1
O=C(C1C(N(CCCn2ccnc2)C(=O)C1=O)c1cccnc1)c1cc2ccccc2o1
COc1cccc(\C=C2\C(=O)NN(C2=O)c2ccc(C)cc2)c1
Clc1ccc(cc1)C(=O)C1C(NC(=O)C1=O)c1ccc(Br)cc1
COc1ccc(cc1)C(=O)C1C(NC(=O)C1=O)c1ccc(OC)cc1OC
Fc1ccc(cc1)N1C(C(C(=O)c2ccccc2)C(=O)C1=O)c1ccc(Br)cc1
Cc1ccc(cc1)C(=O)C1C(N(Cc2cccnc2)C(=O)C1=O)c1ccc(Br)cc1
COc1ccc(C2C(C(=O)c3ccc(C)cc3)C(=O)C(=O)N2Cc2cccnc2)c(OC)c1
OC(=O)CCCN1C(\C=C\c2ccccc2)C(C(=O)c2ccccc2)C(=O)C1=O
COc1cc(ccc1O)C1C(C(C)=O)C(=O)C(=O)N1c1ccc(Br)cc1
Brc1ccc(cc1)C1C(C(=O)c2ccccc2)C(=O)C(=O)N1CN1CCOCC1
Clc1ccc(cc1)C1C(C(=O)c2cccs2)C(=O)C(=O)N1CCc1ccccc1
OC(=O)C(CC(=O)c1ccccc1)=Nc1sc2CCCc2c1C#N |w:13.14|
Cc1ccc(cc1Br)N1C(C(C(=O)c2ccccc2)C(=O)C1=O)c1cccc(F)c1
CCCCCCOc1cccc(c1)N1C(C(C(=O)c2ccccc2)C(=O)C1=O)c1cccc(F)c1
CC(=O)C1C(N(CCc2c(C)[nH]c3ccccc23)C(=O)C1=O)c1cccc(F)c1
COc1ccc(cc1)C(=O)C1C(N(CCc2c[nH]c3ccccc23)C(=O)C1=O)c1ccc(cc1)C(C)C
CC(C)C(=O)N(Cc1ccco1)S(=O)(=O)c1cccc2cccnc12
CCCC(=O)N(Cc1ccco1)S(=O)(=O)c1cccc2cccnc12
COc1ccc(cc1)-c1c(C)[nH]n2c1nc1CCCCc1c2=O
COc1cccc(c1)-c1ccnc2[nH]n(-c3ccccc3)c(=O)c12
Cc1cccc(C)c1NC(=O)C(NC(=O)Cc1cccs1)c1ccccc1
CCC(C)(N(Cc1cccs1)C(C)=O)C(=O)NC1CCCCC1
COc1ccc(cc1)C1C(C(=O)N2CCCC(C)C2)c2ccccc2C(=O)N1C
COc1ccc(OC)c(CNC(=O)Cn2c3ccccc3sc2=O)c1
Cc1sc2n(Cc3ccccc3F)c(=O)n(Cc3ccccc3)c(=O)c2c1C
Cc1cccc(c1)C1CC(=O)NC2=C1C(=O)CC(C2)c1cccs1 |c:13|
FC(F)(F)c1ccccc1C1CC(=O)NC2=C1C(=O)CC(C2)c1cccs1 |c:16|
Cc1nc2c(c([nH]n2c(=O)c1Cc1ccccc1)C(F)(F)F)-c1ccc(Cl)cc1
COc1ccccc1N1CCN(CC1)c1nc(cc(n1)C(F)(F)F)-c1ccccc1
FC(F)(F)C(=O)N1CCN(CC1)c1nc(-c2ccccc2)c2ccccc2n1
COc1ccc(cc1OC)-c1cc(nc(n1)N1CCN(CC1)C(c1ccccc1)c1ccccc1)C(F)(F)F
CCOC(=O)N1CCN(CC1)c1nc(cc(n1)C(F)(F)F)-c1ccc(OC)c(OC)c1
CCC(=O)Nc1cc(ccc1OC)-c1cn2cccnc2n1
COc1ccc(cc1NC(=O)C(C)C)-c1cn2cccnc2n1
COc1ccc(cc1NC(=O)CC1CCCCC1)-c1cn2cccnc2n1
COc1ccc(cc1NC(=O)c1c(F)cccc1F)-c1cn2cccnc2n1
COc1ccc(cc1NC(=O)c1c(F)cccc1Cl)-c1cn2cccnc2n1
COc1ccc(CC(=O)Nc2cc(ccc2OC)-c2cn3cccnc3n2)cc1
COc1ccc(cc1NC(=O)Cc1ccc(Cl)cc1)-c1cn2cccnc2n1
CSCC[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](CC(O)=O)NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)C(C)C)C(N)=O
CSCC[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](CCC(O)=O)NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)C(C)C)C(N)=O
CSCC[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](Cc1cnc[nH]1)NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)C(C)C)C(N)=O
CSCC[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](CC(O)=O)NC(=O)[C@@H](CCCCN)NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)C(C)C)C(N)=O
CSCC[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](CCC(O)=O)NC(=O)[C@@H](CCCCN)NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)C(C)C)C(N)=O
CSCC[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CCCCN)NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)C(C)C)C(N)=O
CSCC[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1cnc[nH]1)NC(=O)[C@@H](CCCCN)NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)C(C)C)C(N)=O
CSCC[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](CCCCN)NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)C(C)C)C(N)=O
CSCC[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](CCCCN)NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)C(N)=O
CSCC[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](CCCCN)NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)C(C)C)C(N)=O
CSCC[C@@H](NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](CCCCN)NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)C(N)=O
CSCC[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)[C@@H](CCCN=C(N)N)NC(=O)[C@@H](N)Cc1c[nH]c2ccccc12)C(C)C)C(N)=O |wU:32.40,12.16,wD:43.44,20.29,8.8,4.4,(5.12,.93,;6.45,1.7,;6.45,3.24,;7.79,4.01,;7.79,5.55,;9.13,6.26,;10.45,5.52,;10.45,3.98,;11.76,6.17,;13.15,5.32,;14.49,5.99,;14.49,7.53,;15.92,5.25,;15.92,3.67,;14.54,2.87,;14.63,1.34,;13.2,.65,;17.24,5.99,;18.49,5.32,;18.49,3.77,;19.9,6.1,;19.9,7.63,;18.6,8.44,;18.6,9.98,;17.27,10.75,;15.94,9.98,;14.6,10.75,;15.94,8.44,;17.27,7.67,;21.12,5.25,;22.39,6.1,;22.39,7.72,;23.71,5.32,;25.19,6.17,;25.19,7.71,;26.52,8.48,;26.52,10.02,;27.86,10.79,;27.86,12.33,;29.19,10.02,;23.71,3.79,;24.91,3.07,;26.09,3.79,;24.91,1.53,;23.76,.65,;26.25,.76,;27.58,1.53,;27.74,3.06,;29.25,3.38,;30.02,2.04,;31.52,1.72,;32.05,.25,;30.97,-.89,;29.46,-.57,;28.99,.9,;11.83,7.72,;10.58,8.51,;13.17,8.49,;6.52,6.38,;5.25,5.55,;6.52,7.93,)|
CSCC[C@@H](NC(=O)[C@@H](NC(=O)[C@H](CCSC)NC(=O)[C@@H](N)Cc1ccc(O)cc1)C(C)C)C(N)=O
COc1ccc(cc1)[C@H]1CC(=O)NC[C@@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
COc1ccc(cc1)[C@H]1CCN(C[C@@H]1NC(=O)Nc1ccc(Cl)cc1)C(C)=O |r|
COc1ccc(cc1)[C@H]1CC(=O)NC[C@@H]1NC(=O)Nc1ccc(Br)cc1 |r|
COc1ccc(cc1)[C@H]1CCNC[C@@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
COc1cc(F)c([C@H]2CCN(C[C@@H]2NC(=O)Nc2ccc(Cl)cc2)C(C)=O)c(F)c1 |r|
COc1ccc(cc1)[C@H]1CCNC[C@@H]1NC(=O)Nc1ccc(Br)cc1 |r|
COc1ccc(cc1)[C@H]1CC(=O)N(C)C[C@@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
COc1cc(F)c([C@H]2CCNC[C@@H]2NC(=O)Nc2ccc(Br)cc2)c(F)c1 |r|
COc1cc(F)c([C@H]2CCNC[C@@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1 |r|
COc1ccc(cc1)[C@H]1CC(=O)N(C)C[C@@H]1NC(=O)Nc1ccc(Cl)cc1
COc1ccc(cc1)[C@@H]1CC(=O)N(C)C[C@H]1NC(=O)Nc1ccc(Cl)cc1
COc1ccc(cc1)[C@H]1CCN(C[C@@H]1NC(=O)Nc1ccc(Cl)cc1)C(=O)C1CC1 |r|
COc1ccc(cc1)[C@H]1CCN(C[C@@H]1NC(=O)Nc1ccc(Cl)cc1)C(=O)CO |r|
COc1ccc(cc1)[C@H]1CCN(C[C@@H]1NC(=O)Nc1ccc(Cl)cc1)C(=O)C(C)(F)F |r|
COCCC(=O)N1CC[C@@H]([C@H](C1)NC(=O)Nc1ccc(Cl)cc1)c1ccc(OC)cc1 |r|
COc1ccc(cc1)[C@H]1CCN(C[C@@H]1NC(=O)Nc1ccc(Cl)cc1)C(=O)C1CCOCC1 |r|
COc1ccc(cc1)[C@H]1CCN(C[C@@H]1NC(=O)Nc1ccc(Cl)cc1)C(=O)C(C)C |r|
COc1ccc(cc1)[C@H]1CCN(C[C@@H]1NC(=O)Nc1ccc(Cl)cc1)C(=O)CC(C)C |r|
COc1ccc(cc1)[C@H]1CCN(C[C@@H]1NC(=O)Nc1ccc(Cl)nc1)C(C)=O |r|
COc1ccc(cc1)[C@H]1CC(=O)N(CC(N)=O)C[C@@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
COC(=O)CN1C[C@H](NC(=O)Nc2ccc(Cl)cc2)[C@H](CC1=O)c1ccc(OC)cc1
COc1cc(F)c([C@H]2CC(=O)NC[C@@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1 |r|
COc1ccc(cc1)[C@H]1CC(=O)N(CC2CC2)C[C@@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
COc1ccc(cc1)[C@H]1CCN(C[C@@H]1NC(=O)Nc1cncnc1)C(C)=O |r|
COc1ccc(cc1)[C@H]1CCN(C[C@@H]1NC(=O)Nc1ccc(C)nc1)C(C)=O |r|
COc1ccc(cc1)[C@H]1CCN(C[C@@H]1NC(=O)Nc1ccc(nc1)C(F)(F)F)C(C)=O |r|
COc1cc(F)c([C@H]2CC(=O)N(CC3CC3)C[C@@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1 |r|
COc1ccc(cc1)[C@H]1CCN(C[C@@H]1NC(=O)Nc1ccc(Cl)cc1)C(=O)CCO |r|
COc1cc(F)c([C@H]2CC(=O)N(CCO)C[C@@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1 |r|
COc1ccc(cc1)[C@H]1CC(=O)N(CCO)C[C@@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
COc1cc(F)c([C@H]2CCNC[C@@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1
COc1cc(F)c([C@@H]2CCNC[C@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1
COc1cc(F)c([C@H]2CCN(C[C@@H]2NC(=O)Nc2ccc(Cl)cc2)C(=O)C2CC2)c(F)c1
COc1cc(F)c([C@@H]2CCN(C[C@H]2NC(=O)Nc2ccc(Cl)cc2)C(=O)C2CC2)c(F)c1
COc1ccc([C@H]2CC(=O)NC[C@@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1
COc1ccc([C@@H]2CC(=O)NC[C@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1
COc1ccc([C@H]2CCNC[C@@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1 |r|
COc1ccc([C@@H]2CCNC[C@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1 |r|
COc1cc(F)c([C@H]2CC(=O)NC[C@@H]2NC(=O)Nc2ccncc2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CC(=O)NC[C@H]2NC(=O)Nc2ccncc2)c(F)c1 |r|
COc1cc(F)c([C@H]2CC(=O)NC[C@@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1
COc1cc(F)c([C@@H]2CC(=O)NC[C@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1
COc1cc(F)c([C@H]2CC(=O)NC[C@@H]2NC(=O)Nc2ccc(Cl)s2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CC(=O)NC[C@H]2NC(=O)Nc2csc(Cl)c2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CC(=O)NC[C@H]2NC(=O)Nc2cc3ccccc3s2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CC(=O)NC[C@H]2NC(=O)Nc2ccc(Oc3ccccc3)cc2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CC(=O)NC[C@H]2NC(=O)Nc2cc(C)ns2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CC(=O)NC[C@H]2NC(=O)Nc2ncc(Cl)s2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CC(=O)NC[C@H]2NC(=O)Nc2ccc(Cl)c(O)c2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CC(=O)NC[C@H]2NC(=O)Nc2ccc(Cl)c(F)c2)c(F)c1 |r|
COCCN1CC(NC(=O)Nc2ccc(Cl)cc2)C(CC1=O)c1ccc(OC)cc1F |w:22.23,6.6|
COc1ccc(C2CC(=O)N(CC(F)F)CC2NC(=O)Nc2ccc(Cl)cc2)c(F)c1 |w:5.5,16.17|
COCCN1CC(NC(=O)Nc2ccc(Cl)cc2)C(CC1=O)c1ccc(F)cc1F |w:22.23,6.6|
FC(F)CN1CC(NC(=O)Nc2ccc(Cl)cc2)C(CC1=O)c1ccc(F)cc1F |w:22.23,6.6|
Fc1ccc(C2CC(=O)NCC2NC(=O)Nc2ccc(Cl)cc2)c(F)c1 |w:4.4,11.12|
CCc1cc(F)c([C@H]2CC(=O)NC[C@@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1 |r|
FC(F)Oc1cc(F)c([C@H]2CC(=O)NC[C@@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1 |r|
CSc1ccc(cc1)[C@H]1CC(=O)NC[C@@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
CCc1ccc(cc1)[C@H]1CC(=O)NC[C@@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
FC(F)Oc1ccc(cc1)[C@H]1CC(=O)NC[C@@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
CS(=O)(=O)c1ccc(cc1)[C@H]1CC(=O)NC[C@@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
COc1ccc(cc1)[C@H]1CC(=O)NC[C@@H]1NC(=O)Nc1ccc(Cl)cc1
COc1ccc(cc1)[C@@H]1CC(=O)NC[C@H]1NC(=O)Nc1ccc(Cl)cc1
Clc1ccc(NC(=O)N[C@H]2CNCC[C@@H]2c2ccccc2)cc1
Clc1ccc(NC(=O)N[C@@H]2CNCC[C@H]2c2ccccc2)cc1
Clc1ccc(NC(=O)N[C@H]2CN(CC[C@@H]2c2ccccc2)C(=O)C2CC2)cc1
Clc1ccc(NC(=O)N[C@@H]2CN(CC[C@H]2c2ccccc2)C(=O)C2CC2)cc1
COc1ccc([C@H]2CCN(C[C@@H]2NC(=O)Nc2ccc(Cl)cc2)C(=O)C2CC2)c(F)c1
COc1cc(F)c(C2C(CCCN2C)NC(=O)Nc2ccc(Cl)cc2)c(F)c1
COc1ccc(cc1)C1C(CCCN1C)NC(=O)Nc1ccc(Cl)cc1
Clc1ccc(NC(=O)NC2CNC(=O)CC2c2ccc(Cl)cc2)cc1 |w:16.16,9.8|
CS(=O)(=O)Nc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3)C2=O)c(F)c1F |r|
OCc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
OCc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3)C2=O)c(F)c1F |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3c(F)cc(Cl)cc3F)C2=O)c(F)c1F |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3)C(F)(F)F)C2=O)c(F)c1F |r|
CS(=O)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
Fc1c(F)c(ccc1N1CC[C@@H](NC(=O)Nc2ccc(Cl)cc2)C1=O)-c1ccccc1C#N |r|
Fc1cc(Cl)ccc1NC(=O)N[C@@H]1CCN(C1=O)c1ccc(c(F)c1F)-c1ccccc1C#N |r|
CS(=O)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3)C2=O)c(F)c1F |r|
CS(=O)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3)C(F)(F)F)C2=O)c(F)c1F |r|
CC(N)c1cccc(c1)-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3)C2=O)c(F)c1F |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ncc(Cl)cc3F)C2=O)c(F)c1F |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(cc1)N1CC[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3cnc(Cl)cn3)C2=O)c(F)c1F |r|
Fc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3)C2=O)c(F)c1F |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cn3)C2=O)c(F)c1F |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3cnc(cn3)C(F)(F)F)C2=O)c(F)c1F |r|
Fc1ncccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3)C2=O)c(F)c1F |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(cc1)N1CC[C@@H](NC(=O)Nc2ccc(nc2)C(F)(F)F)C1=O |r|
Fc1cc(Cl)ccc1NC(=O)N[C@@H]1CCN(C1=O)c1ccc(c(F)c1F)-c1ccccc1F |r|
CS(=O)(=O)Nc1ncccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CS(=O)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cn3)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(c1)C1CC1 |r|
CC(C)c1cc(ccc1N1CC[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C1=O)-c1ccccc1NS(C)(=O)=O |r|
Cn1ccc(n1)-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CS(=O)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
COC[C@@H]1C[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C(=O)N1c1ccc(c(F)c1F)-c1ccccc1P(C)(C)=O |r|
OCc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1 |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
COc1c(F)c(ccc1-c1ccccc1NS(C)(=O)=O)N1CC[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C1=O |r|
COc1c(F)c(ccc1-c1ccccc1CO)N1CC[C@@H](NC(=O)Nc2ccc(cc2F)C(F)(F)F)C1=O |r|
COc1c(F)c(ccc1N1CC[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C1=O)-c1ccccc1NS(C)(=O)=O |r|
CC(C)c1cc(ccc1N1CC[C@@H](NC(=O)Nc2ccc(cc2F)C(F)(F)F)C1=O)-c1ccccc1NS(C)(=O)=O |r|
CC(C)c1cc(ccc1N1CC[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C1=O)-c1ccccc1CO |r|
CS(=O)(=O)c1ccccc1-c1ccc(N2[C@H](CO)C[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CC(C)c1cc(ccc1N1CC[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C1=O)-c1ccccc1S(C)(=O)=O |r|
OCc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3)C(F)(F)F)C2=O)c(F)c1F |r|
CS(=O)(=O)c1ccccc1-c1ccc(N2[C@H](CO)C[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(c1)C1CC1 |r|
CC(NC(C)=O)c1cccc(c1)-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CC(C)c1cc(ccc1N1CC[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C1=O)-c1ccccc1P(C)(C)=O |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(c1)C1CC1 |r|
CC(C)c1cc(ccc1N1CC[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C1=O)-c1cccnc1NS(C)(=O)=O |r|
CS(=O)(=O)Nc1ncccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(c1)C1CC1 |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cn3)C2=O)c(F)c1F |r|
CC(N)c1cccc(c1)-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(OC(F)(F)F)cc3)C2=O)c(F)c1F |r|
CS(=O)(=O)c1ccccc1-c1cc(F)c(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1 |r|
CP(C)(=O)c1ccccc1-c1cc(F)c(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1 |r|
COc1ccc(NC(=O)N[C@@H]2CCN(C2=O)c2ccc(c(F)c2F)-c2ccccc2S(C)(=O)=O)cc1 |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ncc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ncc(Cl)cc3F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CS(=N)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CC(C)c1cc(ccc1N1CC[C@@H](NC(=O)Nc2ccc(cc2F)C(F)(F)F)C1=O)-c1ccccc1P(C)(C)=O |r|
CC(C)c1cc(ccc1N1CC[C@@H](NC(=O)Nc2ncc(Cl)cc2F)C1=O)-c1ccccc1P(C)(C)=O |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3cnc(Cl)cn3)C2=O)c(c1)C1CC1 |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3cnc(Cl)cn3)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cn3)C(F)(F)F)C2=O)c(F)c1F |r|
COc1ccc(NC(=O)N[C@@H]2CCN(C2=O)c2ccc(c(F)c2F)-c2ccccc2P(C)(C)=O)cc1 |r|
CS(=N)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CCP(=O)(CC)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ncc(Cl)cc3F)C2=O)c(F)c1F |r|
CCP(=O)(CC)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(OC(F)(F)F)cc3F)C2=O)c(F)c1F |r|
CP(C)(=O)c1c(F)cccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
COc1ccc(NC(=O)N[C@@H]2CCN(C2=O)c2ccc(c(F)c2F)-c2ccccc2P(C)(C)=O)c(F)c1 |r|
CP(C)(=O)c1c(F)cccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ncccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ncccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CCP(=O)(CC)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1cc(F)c(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1 |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1Cl |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(Cl)c1Cl |r|
FC(F)n1cc(cn1)-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(Cl)c1Cl |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1Cl |r|
OC[C@@H]1C[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C(=O)N1c1ccc(c(F)c1F)-c1ccccc1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1C(F)(F)F |r|
CP(C)(=O)c1ncncc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CP(C)(=O)c1c(F)cccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1Cl |r|
CP(C)(=O)c1c(F)cccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1Cl |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1OC(F)(F)F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1OC(F)(F)F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1C1CC1 |r|
COC[C@@H]1C[C@@H](NC(=O)Nc2ccc(cc2F)C(F)(F)F)C(=O)N1c1ccc(c(F)c1F)-c1ccccc1P(C)(C)=O |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(c1F)C(F)(F)F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(c1F)C(F)(F)F |r|
CP(C)(=O)c1ncncc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1C(F)(F)F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1C(F)F |r|
Cc1c(F)c(ccc1N1CC[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C1=O)-c1ccccc1P(C)(C)=O |r|
Fc1cc(ccc1NC(=O)N[C@@H]1CCN(C1=O)c1ccc(c(F)c1F)-c1cccc2CNS(=O)(=O)c12)C(F)(F)F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(Cl)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(Cl)c1F |r|
CCP(=O)(CC)c1ncccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CCOP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CC1(C)CN(C(=O)[C@@H]1NC(=O)Nc1ccc(cc1F)C(F)(F)F)c1ccc(c(F)c1F)-c1ccccc1P(C)(C)=O |r|
CC1(C)CN(C(=O)[C@@H]1NC(=O)Nc1ccc(Cl)cc1F)c1ccc(c(F)c1F)-c1ccccc1P(C)(C)=O |r|
CCOP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c2OC(F)(F)Oc12 |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(C(F)F)c1F |r|
COP(=O)(OC)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CC1C[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C(=O)N1c1ccc(c(F)c1F)-c1ccccc1P(C)(C)=O |r|
CC1(C)CN(C(=O)[C@@H]1NC(=O)Nc1ccc(cc1F)C(F)(F)F)c1ccc(c(F)c1F)-c1cccnc1P(C)(C)=O |r|
CP(C)(=O)c1ccccc1-c1ccc(N2[C@H](CO)C[C@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2[C@H](CO)C[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CC1(C)CN(C(=O)[C@@H]1NC(=O)Nc1ccc(Cl)cc1F)c1ccc(c(F)c1F)-c1cccnc1P(C)(C)=O |r|
CP(C)(=O)c1ccccc1-c1ccc(N2[C@H](CO)C[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CC1C[C@@H](NC(=O)Nc2ccc(cc2F)C(F)(F)F)C(=O)N1c1ccc(c(F)c1F)-c1ccccc1P(C)(C)=O |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(C2CC2)c1F |r|
COc1ncccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
Fc1cc(Cl)ccc1NC(=O)N[C@@H]1CCN(C1=O)c1ccc(c(F)c1F)-c1ccccc1N1CCOC1=O |r|
CC1C[C@@H](NC(=O)Nc2ccc(cc2F)C(F)(F)F)C(=O)N1c1ccc(c(F)c1F)-c1cccnc1P(C)(C)=O |r|
CC1C[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C(=O)N1c1ccc(c(F)c1F)-c1cccnc1P(C)(C)=O |r|
CP(C)(=O)c1ncccc1-c1ccc(N2[C@H](CO)C[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC(CO)[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC(CO)[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CC1C[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C(=O)N1c1ccc(c(F)c1F)-c1ccccc1S(C)(=O)=O |r|
CC1(C)CN(C(=O)[C@@H]1NC(=O)Nc1cnc(Cl)cn1)c1ccc(c(F)c1F)-c1ccccc1P(C)(C)=O |r|
CP(C)(=O)c1ccccc1-c1ccc(N2[C@H](CN3CCOCC3)C[C@@H](NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC3(CC3)[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3csc(Cl)c3)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3cccc(Cl)c3)C2=O)c(F)c1F |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)s3)C2=O)c(F)c1F |r|
Cc1ccc(NC(=O)NC2CCCN(C2=O)c2ccc(cc2)-c2cccnc2)cc1
Clc1ccc(NC(=O)NC2CCCN(C2=O)c2ccc(cc2)-c2cccnc2)cc1
COc1ccc(NC(=O)NC2CCCN(C2=O)c2ccc(cc2F)-c2ccccc2S(C)(=O)=O)cc1
Cc1cnc(NC(=O)NC2CCCN(C2=O)c2ccc(cc2F)-c2ccccc2S(C)(=O)=O)s1
CS(=O)(=O)c1ccccc1-c1ccc(N2CCCC(NC(=O)Nc3ccc(Cl)nn3)C2=O)c(F)c1
CS(=O)(=O)c1ccccc1-c1ccc(N2CCCC(NC(=O)Nc3ccc(F)cc3)C2=O)c(F)c1
FC(F)(F)c1ccc(NC(=O)NC2CCCN(C2=O)c2ccc(cc2)-c2ccccc2)cc1
Cc1ccncc1-c1ccc(cc1)N1CCCC(NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O
NC(=O)c1ccc(cc1)-c1ccc(cc1)N1CCCC(NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O
Cc1ccc(cc1)-c1ccc(cc1)N1CCCC(NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O
OCc1ccccc1-c1ccc(cc1)N1CCC[C@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O |r|
Clc1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)-c2ccccc2C#N)cc1 |r|
OCc1ccccc1-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(Cl)cc2)C1=O |r|
NC(=O)c1ccccc1-c1ccc(N2CCC[C@@H](NC(=O)Nc3ccc(Cl)cc3)C2=O)c(F)c1 |r|
Clc1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)-c2c(Cl)cccc2Cl)cc1 |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(Cl)cc2)C1=O |r|
Fc1cccc(c1F)-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O |r|
CCOc1ncccc1-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O |r|
NC(=O)c1ccccc1-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O |r|
CN(c1ncccc1-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O)S(C)(=O)=O |r|
FC(F)(F)c1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)-c2cncc(c2)N2CCOCC2)cc1 |r|
NC(=O)c1ccccc1-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(F)cc2)C1=O |r|
Cc1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)-c2ccccc2C(N)=O)c(C)c1 |r|
COc1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)-c2ccccc2C(N)=O)cc1Cl |r|
NC(=O)c1ccccc1-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(F)c(F)c2)C1=O |r|
CC(C)(C)NS(=O)(=O)c1ccccc1-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(Cl)cc2)C1=O |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(cn2)C(F)(F)F)C1=O |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C1=O |r|
COc1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)-c2ccccc2NS(C)(=O)=O)c(F)c1 |r|
COc1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)-c2ccccc2NS(C)(=O)=O)cc1 |r|
FC(F)(F)c1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)N2CCCCC2=O)cc1 |r|
FC(F)(F)c1ccc(NC(=O)N[C@H]2CCCN(C2=O)c2ccc(cc2)N2CC3(COC3)C2)cc1 |r|
FC(F)(F)c1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)N2CC3(COC3)C2)nc1 |r|
COCC1CCCCN1c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O |r|
COCC1CCCCN1c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(nc2)C(F)(F)F)C1=O |r|
COC[C@@H]1CCCN1c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(Cl)cn2)C1=O |r|
COC[C@@H]1CCCN1c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(Cl)cc2)C1=O |r|
CS(=O)(=O)N1CCN(CC1)c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O |r|
FC(F)(F)c1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)N2CCCCC2)cc1 |r|
Fc1cc(ccc1N1CCC[C@@H](NC(=O)Nc2ccc(nc2)C(F)(F)F)C1=O)N1CCCCC1=O |r|
FC(F)(F)c1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(nc2)N2CCOCC2)cc1 |r|
OCC1CCCN(C1)c1ccc(cn1)N1CCC[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O |r|
CC(=O)N[C@@H]1CCN(C1)c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O |r|
FC(F)(F)c1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)N2CCCC(F)(F)C2)cc1 |r|
CN(C)C1CCCN(C1)c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O |r|
CN(C)C1CCN(C1)c1ccc(N2CCC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(F)c1 |r|
CN(C)C1CCN(C1)c1ccc(cc1F)N1CCC[C@@H](NC(=O)Nc2ccc(Cl)cc2)C1=O |r|
Clc1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)N2C[C@@H]3COC[C@@H]3C2)cc1 |r|
Clc1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)N2CCC3(CCCO3)CC2)cc1 |r|
FC(F)(F)c1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(nc2)N2C[C@@H]3CC[C@H](C2)O3)cc1 |r|
Fc1cc(ccc1N1CCC[C@@H](NC(=O)Nc2ccc(Cl)cc2)C1=O)N1C[C@@H]2CC[C@H](C1)O2 |r|
CS(=O)(=O)NCC1(CCC1)c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2cnc(Cl)cn2)C1=O |r|
CS(=O)(=O)NCC1(CC1)c1ccc(cc1F)N1CCC[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O |r|
CS(=O)(=O)NCC1(CC1)c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2cnc(Cl)cn2)C1=O |r|
CS(=O)(=O)NCC1(CC1)c1ccc(cc1)N1CCC[C@H](NC(=O)Nc2ncc(Cl)cc2F)C1=O |r|
CS(=O)(=O)NCC1(CC1)c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O |r|
FC(F)(F)c1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)C2(CN3CCOCC3)CCC2)cn1 |r|
Clc1ccc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2)C2(CN3CCOCC3)CC2)nc1 |r|
FC(F)(F)c1ccc(NC(=O)N[C@H]2CCCN(C2=O)c2ccc(cc2)C2(CN3CCCC3)CCC2)cn1 |r|
FC(F)(F)c1ccc(NC(=O)N[C@H]2CCCN(C2=O)c2ccc(cc2)C2(CN3CCCC3)CCCC2)cn1 |r|
FC(F)(F)c1ccc(NC(=O)N[C@H]2CCCN(C2=O)c2ccc(cc2)C2(CN3CCOCC3)CCC2)cn1 |r|
CS(=O)(=O)NCC1(CC1)c1ccc(cc1)N1C[C@@H](O)C[C@H](NC(=O)Nc2ncc(cc2F)C(F)(F)F)C1=O |r|
CS(=O)(=O)NCC1(CC1)c1ccc(cc1)N1C[C@@H](O)C[C@@H](NC(=O)Nc2ncc(Cl)cc2F)C1=O |r|
CC(NC(C)=O)C1(CC1)c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(nc2)C(F)(F)F)C1=O |r|
OC1CCC(C1)c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C1=O |r|
COc1c(F)c(ccc1-c1ccccc1CO)N1CC[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C1=O |r|
CS(=N)(=O)c1ccccc1-c1ccc(N2CCC(NC(=O)Nc3ccc(cc3F)C(F)(F)F)C2=O)c(F)c1F
CS(=O)(=O)Nc1ccccc1-c1ccc(cc1)N1C[C@H](O)C[C@@H](NC(=O)Nc2ccc(Cl)cc2)C1=O |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(cc2F)C(F)(F)F)C1=O |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(cc1)N1C[C@H](O)C[C@@H](NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(cc1)N1C[C@H](O)C[C@H](NC(=O)Nc2ncc(Cl)cc2F)C1=O |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(cc1)N1C[C@H](O)C[C@@H](NC(=O)Nc2ccc(Cl)cn2)C1=O |r|
COc1cc(ccc1N1CCC[C@@H](NC(=O)Nc2ncc(cc2F)C(F)(F)F)C1=O)-c1ccccc1NS(C)(=O)=O |r|
COc1cc(ccc1N1CCC[C@@H](NC(=O)Nc2ccc(cn2)C(F)(F)F)C1=O)-c1ccccc1NS(C)(=O)=O |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(OC(F)F)nc2)C1=O |r|
Cc1cnc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(cc2F)-c2ccccc2NS(C)(=O)=O)cn1 |r|
COc1cnc(NC(=O)N[C@@H]2CCCN(C2=O)c2ccc(c(F)c2)-c2ccccc2NS(C)(=O)=O)c(F)c1 |r|
CS(=O)(=O)Nc1ccccc1-c1cc(F)c(N2CCC[C@@H](NC(=O)Nc3ccc(Cl)cc3)C2=O)c(F)c1 |r|
NCc1cccc(c1F)-c1ccc(cc1)N1CCC[C@@H](NC(=O)Nc2ccc(Cl)cc2)C1=O |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(cc1)N1C[C@H](O)C[C@@H](NC(=O)Nc2ccc(Cl)cc2F)C1=O |r|
CS(=O)(=O)Nc1ccccc1-c1ccc(N2CCC[C@@H](NC(=O)Nc3ccc(Cl)cc3F)C2=O)c(Cl)c1 |r|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccccc1 |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.35,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.91,;-3.43,3.82,;-4.84,3.19,;-5,1.66,;-3.75,.76,)|
COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccccc1
COc1cccc(c1)-c1cn(c(NC(=O)c2ccc(OC(F)F)cc2)n1)-c1c(F)cc(OC)cc1F |(-7.65,1.94,;-6.41,1.04,;-5,1.66,;-4.84,3.19,;-3.43,3.82,;-2.19,2.91,;-2.35,1.38,;-3.75,.76,;-1.1,.48,;-1.1,-1.06,;.36,-1.54,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;.36,.95,;.84,-3,;-.19,-4.15,;-1.7,-3.83,;.28,-5.61,;1.79,-5.93,;2.27,-7.4,;1.24,-8.54,;2.82,-4.79,;2.35,-3.32,;3.38,-2.18,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccc(F)cc1 |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.92,;-3.43,3.82,;-4.84,3.19,;-6.09,4.1,;-5,1.66,;-3.75,.76,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccc(Cl)c(C)c1 |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.92,;-3.43,3.82,;-4.84,3.19,;-6.09,4.1,;-5,1.66,;-6.41,1.04,;-3.75,.76,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccc(cc1)C(F)(F)F |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.92,;-3.43,3.82,;-4.84,3.19,;-5,1.66,;-3.75,.76,;-6.09,4.1,;-7.49,3.47,;-5.92,5.63,;-6.25,2.57,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccc(OC(F)F)cc1 |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.92,;-3.43,3.82,;-4.84,3.19,;-6.09,4.1,;-5.92,5.63,;-7.17,6.54,;-4.52,6.26,;-5,1.66,;-3.75,.76,)|
COc1cc(F)c(c(F)c1)-n1c(C)c(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccccc1 |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-2.35,-1.97,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.92,;-3.43,3.82,;-4.84,3.19,;-5,1.66,;-3.75,.76,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccc2ccccc2c1 |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-3.75,.76,;-5,1.66,;-4.84,3.19,;-6.09,4.1,;-5.92,5.63,;-4.52,6.26,;-3.27,5.35,;-3.43,3.82,;-2.19,2.92,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1cccc(F)c1 |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.92,;-3.43,3.82,;-4.84,3.19,;-5,1.66,;-6.41,1.04,;-3.75,.76,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccc(Cl)cc1 |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.92,;-3.43,3.82,;-4.84,3.19,;-6.09,4.1,;-5,1.66,;-3.75,.76,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1cccc(Cl)c1 |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-3.75,.76,;-5,1.66,;-4.84,3.19,;-3.43,3.82,;-3.27,5.35,;-2.19,2.92,)|
COc1cc(F)c(c(F)c1)-n1c(C)c(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccc(Cl)cc1 |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-2.35,-1.97,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.92,;-3.43,3.82,;-4.84,3.19,;-6.09,4.1,;-5,1.66,;-3.75,.76,)|
COc1ccc(cc1)-c1cn(c(NC(=O)c2ccc(OC(F)F)cc2)n1)-c1c(F)cc(OC)cc1F |(-7.49,3.47,;-6.09,4.1,;-4.84,3.19,;-3.43,3.82,;-2.19,2.92,;-2.35,1.38,;-3.75,.76,;-5,1.66,;-1.1,.48,;-1.1,-1.06,;.36,-1.54,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;.36,.95,;.84,-3,;-.19,-4.15,;-1.7,-3.83,;.28,-5.61,;1.79,-5.93,;2.27,-7.4,;1.24,-8.54,;2.82,-4.79,;2.34,-3.32,;3.38,-2.18,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccc(C)cc1 |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.92,;-3.43,3.82,;-4.84,3.19,;-6.09,4.1,;-5,1.66,;-3.75,.76,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccc(cc1)C#N |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.92,;-3.43,3.82,;-4.84,3.19,;-5,1.66,;-3.75,.76,;-6.09,4.1,;-7.33,5,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1cccc(c1)C#N |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.92,;-3.43,3.82,;-4.84,3.19,;-5,1.66,;-3.75,.76,;-6.41,1.04,;-7.81,.41,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccc(Cl)c(Cl)c1 |(1.24,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.38,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.92,;-3.43,3.82,;-4.84,3.19,;-6.09,4.1,;-5,1.66,;-6.41,1.04,;-3.75,.76,)|
COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccc2OCCc2c1
COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccnc(Cl)c1
COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccc(F)cc1F
COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccc2sccc2c1
COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1nc2ccccc2s1
COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1nccs1
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccccc1F |(1.23,-8.54,;2.27,-7.4,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.95,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-3.76,.76,;-5,1.66,;-4.84,3.19,;-3.43,3.82,;-2.19,2.92,;-.78,3.54,)|
COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1nc2cc(Cl)ccc2o1
COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C1CCCCC1
COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccccn1
CCOC(=O)c1cc(on1)-c1cn(c(NC(=O)c2ccc(OC(F)F)cc2)n1)-c1ccc(OC)cc1
CCOC(=O)c1cn(c(NC(=O)c2ccc(OC(F)F)cc2)n1)-c1ccc(OC)cc1
COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C12CC3CC(CC(C3)C1)C2 |TLB:33:32:35:29.28.27,33:28:35:34.32.31,29:30:34:33.28.27,THB:29:28:34:35.30.31|
COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(C)(C)C
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccccc1F |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-3.76,.76,;-5,1.66,;-4.84,3.19,;-3.43,3.82,;-2.19,2.92,;-.78,3.54,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccnc(Cl)c1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.83,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-3.76,.76,;-5,1.66,;-4.84,3.19,;-3.43,3.82,;-3.27,5.35,;-2.19,2.92,)|
COc1cc(F)c(c(F)c1)-n1cc(CC(C)C)nc1NC(=O)c1ccc(OC(F)F)cc1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;-2.35,1.38,;-3.76,.76,;-5,1.66,;-3.92,-.77,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccc(F)c(F)c1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-3.76,.76,;-5,1.66,;-4.84,3.2,;-6.09,4.1,;-3.44,3.82,;-3.27,5.35,;-2.19,2.92,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C1CC1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.14,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-3.89,1.38,;-3.12,2.72,)|
CCOC(=O)c1cn(c(NC(=O)c2ccc(OC(F)F)cc2)n1)-c1c(F)cc(OC)cc1F |(-4.84,3.19,;-3.44,3.82,;-2.19,2.92,;-2.35,1.38,;-3.76,.76,;-1.1,.48,;-1.1,-1.06,;.36,-1.54,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;.36,.96,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;1.79,-5.93,;2.26,-7.39,;1.23,-8.54,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,)|
CCc1cn(c(NC(=O)c2ccc(OC(F)F)cc2)n1)-c1c(F)cc(OC)cc1F |(-3.76,.76,;-2.35,1.38,;-1.1,.48,;-1.1,-1.06,;.36,-1.54,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;.36,.96,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;1.79,-5.93,;2.26,-7.39,;1.23,-8.54,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1nccs1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.14,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-3.81,.91,;-4.72,2.15,;-3.81,3.4,;-2.35,2.92,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C1CCOCC1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.14,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.92,;-3.43,3.82,;-4.84,3.19,;-5,1.66,;-3.76,.76,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(F)(F)C(F)(F)F |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.14,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-3.76,.76,;-2.51,-.15,;-2.19,2.92,;-3.43,3.82,;-.78,3.54,;-.94,2.01,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(F)(F)F |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.14,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-3.76,.76,;-2.51,-.15,;-2.19,2.92,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)NCc1cc[nH]n1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.15,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.54,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.38,;-2.19,2.92,;-3.76,.76,;-5,1.66,;-6.41,1.04,;-6.73,-.47,;-8.26,-.63,;-8.89,.78,;-7.74,1.81,)|
COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)N1CCNCC1
COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)NCCCO
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)NCc1cccnc1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-5,1.66,;-6.41,1.04,;-7.66,1.94,;-9.06,1.31,;-9.22,-.22,;-7.98,-1.12,;-6.57,-.5,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)NCc1ccncc1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-5,1.66,;-6.41,1.04,;-7.66,1.94,;-9.06,1.31,;-9.22,-.22,;-7.98,-1.12,;-6.57,-.5,)|
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COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)N1CCC[C@H]1CO |r,wD:34.38,(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-5.09,1.53,;-6.24,.5,;-5.61,-.91,;-4.08,-.75,;-3.05,-1.89,;-3.52,-3.36,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)N1CCCC(O)C1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-3.92,-.77,;-5.32,-1.4,;-6.57,-.49,;-6.41,1.04,;-7.66,1.94,;-5,1.66,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)N1CCC(O)CC1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-5,1.66,;-6.41,1.04,;-6.57,-.49,;-7.98,-1.12,;-5.32,-1.4,;-3.92,-.77,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)NCCO |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-5,1.66,;-6.41,1.04,;-7.66,1.94,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)N1CCOCC1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-5,1.66,;-6.41,1.04,;-6.57,-.49,;-5.32,-1.4,;-3.92,-.77,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)N1CCN(C)CC1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-5,1.66,;-6.41,1.04,;-6.57,-.49,;-7.98,-1.12,;-5.32,-1.4,;-3.92,-.77,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)NCc1cnc(C)cn1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-5,1.66,;-6.41,1.04,;-7.66,1.94,;-9.06,1.32,;-9.22,-.22,;-10.63,-.84,;-7.98,-1.12,;-6.57,-.49,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)N1CC[C@H](O)C1 |r,wD:33.36,(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-4.08,-.75,;-5.61,-.91,;-6.23,.5,;-7.74,.82,;-5.09,1.53,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)N1CCNC(=O)C1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-3.92,-.77,;-5.32,-1.4,;-6.57,-.49,;-6.41,1.04,;-7.66,1.94,;-5,1.66,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)N1CCC(CO)C1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-4.08,-.75,;-5.61,-.91,;-6.24,.5,;-7.74,.82,;-8.77,-.33,;-5.09,1.53,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)NCCCO |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.27,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-5,1.66,;-6.41,1.04,;-7.66,1.94,;-9.06,1.32,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)N1CCNCC1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.26,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-5,1.66,;-6.41,1.04,;-6.57,-.49,;-5.33,-1.4,;-3.92,-.77,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)Nc1cn[nH]c1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.26,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-5,1.66,;-6.47,1.19,;-7.37,2.43,;-6.47,3.68,;-5,3.2,)|
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COc1ccc(cc1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C1CCCNC1
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CCNC(=O)N1CCC(CC1)c1cn(c(NC(=O)c2ccc(OC(F)F)cc2)n1)-c1c(F)cc(OC)cc1F |(-10.15,3.75,;-8.74,4.38,;-7.49,3.47,;-6.09,4.1,;-5.93,5.63,;-4.84,3.2,;-3.44,3.82,;-2.19,2.92,;-2.35,1.39,;-3.76,.76,;-5,1.66,;-1.1,.48,;-1.1,-1.06,;.36,-1.53,;1.26,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;.36,.96,;.84,-3,;-.19,-4.14,;-1.7,-3.82,;.28,-5.61,;1.79,-5.93,;2.26,-7.39,;1.23,-8.54,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C1CCN(CC1)C(=O)CCC(N)=O |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.14,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.26,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.44,3.82,;-4.84,3.2,;-5,1.66,;-3.76,.76,;-6.09,4.1,;-5.93,5.63,;-7.49,3.47,;-8.74,4.38,;-10.15,3.75,;-11.39,4.66,;-10.31,2.22,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C1CCN(CC1)C(=O)CCO |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.14,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.26,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.44,3.82,;-4.84,3.2,;-5,1.66,;-3.76,.76,;-6.09,4.1,;-5.93,5.63,;-7.49,3.47,;-8.74,4.38,;-10.15,3.75,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(=O)N1CCC(CO)CC1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.14,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.26,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-2.19,2.92,;-3.76,.76,;-5,1.66,;-6.41,1.04,;-6.57,-.49,;-7.98,-1.12,;-9.22,-.22,;-5.33,-1.4,;-3.92,-.77,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C(C)C |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.14,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.26,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,;-2.35,1.39,;-3.76,.76,;-2.19,2.92,)|
COc1cc(F)c(c(F)c1)-n1cc(Cc2ccccc2)nc1NC(=O)c1ccc(OC(F)F)cc1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.2,-4.14,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;-2.35,1.39,;-3.76,.76,;-5,1.66,;-6.41,1.04,;-6.57,-.49,;-5.33,-1.4,;-3.92,-.77,;.36,.96,;1.26,-.29,;2.8,-.29,;3.57,1.04,;2.8,2.38,;5.12,1.04,;5.88,-.29,;7.42,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.42,2.38,;5.88,2.38,)|
CCOC(=O)Cc1cn(c(NC(=O)c2ccc(OC(F)F)cc2)n1)-c1c(F)cc(OC)cc1F |(-7.66,1.94,;-6.41,1.04,;-5,1.66,;-3.76,.76,;-3.92,-.77,;-2.35,1.39,;-1.1,.48,;-1.1,-1.06,;.36,-1.53,;1.26,-.29,;2.8,-.29,;3.57,1.04,;2.8,2.38,;5.12,1.04,;5.88,-.29,;7.42,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.42,2.38,;5.88,2.38,;.36,.96,;.84,-3,;-.2,-4.14,;-1.7,-3.82,;.28,-5.61,;1.79,-5.93,;2.26,-7.39,;1.23,-8.54,;2.82,-4.79,;2.34,-3.32,;3.37,-2.18,)|
COc1cc(F)c(c(F)c1)-n1cc(Cc2nnc(C)o2)nc1NC(=O)c1ccc(OC(F)F)cc1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.19,-4.14,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;-2.35,1.39,;-3.76,.76,;-4.08,-.75,;-5.61,-.91,;-6.24,.5,;-7.74,.82,;-5.09,1.53,;.36,.96,;1.26,-.29,;2.81,-.29,;3.58,1.04,;2.81,2.38,;5.12,1.04,;5.89,-.29,;7.43,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.43,2.38,;5.89,2.38,)|
COc1cc(F)c(c(F)c1)-n1cc(CC2CC(O)C2)nc1NC(=O)c1ccc(OC(F)F)cc1 |(-8.66,3.08,;-7.13,2.92,;-6.5,1.51,;-4.97,1.35,;-4.34,-.06,;-2.81,-.22,;-5.25,-1.3,;-6.78,-1.14,;-7.69,-2.39,;-7.41,.26,;-4.62,-2.71,;-3.12,-3.03,;-2.96,-4.56,;-1.62,-5.33,;-1.62,-6.87,;-.53,-7.96,;-1.62,-9.05,;-1.62,-10.59,;-2.71,-7.96,;-4.36,-5.19,;-5.39,-4.04,;-6.92,-4.2,;-7.55,-5.61,;-6.65,-6.86,;-9.08,-5.77,;-9.71,-7.18,;-11.24,-7.34,;-12.15,-6.09,;-13.68,-6.26,;-14.3,-7.66,;-13.4,-8.91,;-15.84,-7.82,;-11.52,-4.69,;-9.99,-4.53,)|
COc1cc(F)c(c(F)c1)-n1cc(CC2CC3(CNC3)C2)nc1NC(=O)c1ccc(OC(F)F)cc1 |(-3.75,11.57,;-2.5,10.67,;-2.66,9.14,;-1.42,8.23,;-1.58,6.7,;-.33,5.79,;-2.99,6.07,;-4.23,6.98,;-5.64,6.35,;-4.07,8.51,;-3.15,4.54,;-2,3.51,;-2.63,2.1,;-1.86,.77,;-.32,.77,;.77,1.86,;1.86,.77,;2.95,1.86,;4.04,.77,;2.95,-.32,;.77,-.32,;-4.16,2.26,;-4.48,3.77,;-5.89,4.4,;-7.13,3.49,;-6.97,1.96,;-8.54,4.12,;-9.79,3.21,;-11.19,3.84,;-11.35,5.37,;-12.76,6,;-12.92,7.53,;-14.33,8.16,;-11.68,8.43,;-10.11,6.28,;-8.7,5.65,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C1CCC(O)CC1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.2,-4.14,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.26,-.29,;2.8,-.29,;3.57,1.04,;2.8,2.38,;5.12,1.04,;5.88,-.29,;7.42,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.42,2.38,;5.88,2.38,;-2.35,1.39,;-2.19,2.92,;-3.44,3.82,;-4.84,3.2,;-6.09,4.1,;-5,1.66,;-3.76,.76,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1nc2ncc(N)cc2[nH]1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.2,-4.14,;-1.7,-3.82,;.84,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.79,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;.36,.96,;1.26,-.29,;2.8,-.29,;3.57,1.04,;2.8,2.38,;5.12,1.04,;5.88,-.29,;7.42,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.42,2.38,;5.88,2.38,;-2.35,1.39,;-2.35,2.93,;-3.82,3.4,;-4.44,4.81,;-5.97,4.97,;-6.88,3.72,;-8.41,3.88,;-6.25,2.32,;-4.72,2.16,;-3.82,.91,)|
COc1cc(F)c(c(F)c1)-n1cc(Cc2ccccn2)nc1NC(=O)c1ccc(OC(F)F)cc1 |(1.23,-8.54,;2.26,-7.39,;1.79,-5.93,;.28,-5.61,;-.2,-4.14,;-1.7,-3.82,;.83,-3,;2.34,-3.32,;3.37,-2.18,;2.82,-4.78,;.36,-1.53,;-1.1,-1.06,;-1.1,.48,;-2.35,1.39,;-3.76,.76,;-3.92,-.77,;-5.33,-1.4,;-6.57,-.49,;-6.41,1.04,;-5,1.66,;.36,.96,;1.26,-.29,;2.8,-.29,;3.57,1.04,;2.8,2.38,;5.12,1.04,;5.88,-.29,;7.42,-.29,;8.2,1.04,;9.74,1.04,;10.51,2.38,;9.74,3.71,;12.05,2.38,;7.42,2.38,;5.88,2.38,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C1CNC1 |(-8.66,3.08,;-7.13,2.92,;-6.5,1.51,;-4.97,1.35,;-4.34,-.06,;-2.81,-.22,;-5.25,-1.3,;-6.78,-1.14,;-7.69,-2.39,;-7.41,.27,;-4.62,-2.71,;-3.12,-3.03,;-2.95,-4.56,;-4.36,-5.19,;-5.39,-4.04,;-6.92,-4.2,;-7.55,-5.61,;-6.64,-6.86,;-9.08,-5.77,;-9.71,-7.18,;-11.24,-7.34,;-12.14,-6.09,;-13.68,-6.25,;-14.3,-7.66,;-13.4,-8.91,;-15.83,-7.82,;-11.52,-4.69,;-9.99,-4.53,;-1.62,-5.33,;-.13,-4.93,;.27,-6.42,;-1.22,-6.82,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)-c1ccn[nH]1 |(-8.66,3.08,;-7.13,2.92,;-6.5,1.51,;-4.97,1.35,;-4.34,-.06,;-2.81,-.22,;-5.25,-1.3,;-6.78,-1.14,;-7.69,-2.39,;-7.41,.27,;-4.62,-2.71,;-3.12,-3.03,;-2.95,-4.56,;-4.36,-5.19,;-5.39,-4.04,;-6.92,-4.2,;-7.55,-5.61,;-6.64,-6.86,;-9.08,-5.77,;-9.71,-7.18,;-11.24,-7.34,;-12.15,-6.09,;-13.68,-6.26,;-14.3,-7.66,;-13.4,-8.91,;-15.84,-7.82,;-11.52,-4.69,;-9.99,-4.53,;-1.62,-5.33,;-.21,-4.71,;.82,-5.85,;.05,-7.18,;-1.46,-6.86,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C1CC(N)C1 |(-8.66,3.08,;-7.13,2.92,;-6.5,1.51,;-4.97,1.35,;-4.34,-.06,;-2.81,-.22,;-5.25,-1.3,;-6.78,-1.14,;-7.69,-2.39,;-7.41,.27,;-4.62,-2.71,;-3.11,-3.03,;-2.95,-4.56,;-4.36,-5.19,;-5.39,-4.04,;-6.92,-4.2,;-7.55,-5.61,;-6.64,-6.86,;-9.08,-5.77,;-9.71,-7.18,;-11.24,-7.34,;-12.14,-6.09,;-13.68,-6.26,;-14.3,-7.66,;-13.4,-8.91,;-15.83,-7.82,;-11.52,-4.69,;-9.99,-4.53,;-1.62,-5.33,;-.13,-4.93,;.27,-6.42,;1.6,-7.19,;-1.22,-6.82,)|
COc1cc(F)c(c(F)c1)-n1cc(CC2CC(C2)NCC(F)(F)F)nc1NC(=O)c1ccc(OC(F)F)cc1 |(-8.66,3.08,;-7.13,2.92,;-6.5,1.51,;-4.97,1.35,;-4.34,-.06,;-2.81,-.22,;-5.25,-1.3,;-6.78,-1.14,;-7.69,-2.39,;-7.41,.26,;-4.62,-2.71,;-3.12,-3.03,;-2.96,-4.56,;-1.62,-5.33,;-1.62,-6.87,;-.53,-7.96,;-1.62,-9.05,;-2.71,-7.96,;-1.62,-10.59,;-2.95,-11.36,;-4.29,-10.59,;-5.62,-11.36,;-4.29,-9.05,;-4.29,-12.13,;-4.36,-5.19,;-5.39,-4.04,;-6.92,-4.2,;-7.55,-5.61,;-6.65,-6.86,;-9.08,-5.77,;-9.71,-7.18,;-11.24,-7.34,;-12.15,-6.09,;-13.68,-6.26,;-14.3,-7.66,;-13.4,-8.91,;-15.83,-7.82,;-11.52,-4.69,;-9.99,-4.53,)|
COc1cc(F)c(c(F)c1)-n1cc(nc1NC(=O)c1ccc(OC(F)F)cc1)C1CC(C1)NS(C)(=O)=O |(-8.66,3.08,;-7.13,2.92,;-6.5,1.51,;-4.97,1.35,;-4.34,-.06,;-2.81,-.22,;-5.25,-1.3,;-6.78,-1.14,;-7.69,-2.39,;-7.41,.27,;-4.62,-2.71,;-3.11,-3.03,;-2.95,-4.56,;-4.36,-5.19,;-5.39,-4.04,;-6.92,-4.2,;-7.55,-5.61,;-6.64,-6.86,;-9.08,-5.77,;-9.71,-7.18,;-11.24,-7.34,;-12.14,-6.09,;-13.68,-6.26,;-14.3,-7.66,;-13.4,-8.91,;-15.83,-7.82,;-11.52,-4.69,;-9.99,-4.53,;-1.62,-5.33,;-.13,-4.93,;.27,-6.42,;-1.22,-6.82,;1.6,-7.19,;1.6,-8.73,;1.6,-10.27,;.27,-9.5,;2.93,-9.5,)|
CS(=O)(=O)c1ccc(cc1)-c1ccc(cc1)N1CCCC(NC(=O)Nc2ccc(cc2)C(F)(F)F)C1=O
COc1cc(F)c([C@@H]2CN(C(=O)C2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(N3CCOCC3)c2C(F)(F)F)c(F)c1 |r,wU:7.6,17.17,wD:20.24,(-6.62,7.85,;-7.25,6.44,;-6.34,5.19,;-4.81,5.35,;-3.91,4.11,;-2.38,4.27,;-4.53,2.7,;-3.63,1.45,;-4.1,-.01,;-2.86,-.92,;-1.61,-.01,;-.15,-.49,;-2.09,1.45,;-1.18,2.7,;.35,2.62,;1.05,1.25,;1.19,3.91,;2.73,3.83,;3.58,5.11,;5.12,5.02,;5.8,3.64,;4.95,2.36,;3.42,2.45,;7.34,3.54,;8.19,4.83,;8.03,2.16,;-2.86,-2.46,;-1.53,-3.23,;-1.53,-4.77,;-2.86,-5.54,;-4.19,-4.77,;-5.53,-5.54,;-6.86,-4.77,;-8.19,-5.54,;-8.19,-7.08,;-6.86,-7.85,;-5.53,-7.08,;-4.19,-3.23,;-5.53,-2.46,;-5.53,-.92,;-6.86,-3.22,;-6.86,-1.69,;-6.07,2.54,;-6.69,1.13,;-6.97,3.79,)|
COCC(CO)n1cccc(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)Nc2ccccc2)c2c(OC)ccn(C)c2=O)c(F)c1 |r|
COCCn1cccc(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(Cl)ccc4C3)C2=O)c2ccc(OC)cc2)c1=O |r|
CCn1cccc(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(Cl)ccc4C3)C2=O)c2ccc(OC)cc2)c1=O |r|
COCCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3)C2=O)c2c(F)cc(OC)cc2F)c1=O |r,w:17.17|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)NC2CCc3cc(Cl)ccc3C2)c2c(OC)ccn(C)c2=O)c(F)c1 |r,w:16.17|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)NC2CCc3cc(Cl)ccc3C2)c2ncccc2C(F)(F)F)c(F)c1 |r|
COCCn1cccc(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3)C2=O)c2ccc(OC)cc2)c1=O |r|
CCn1cccc(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3)C2=O)c2ccc(OC)cc2)c1=O |r|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)NC2CCc3cc(Cl)ccc3C2)c2cccn(CCO)c2=O)c(F)c1 |r|
COc1ccc2CC(CCc2c1)NC(=O)N[C@H]1[C@@H]([C@H](C)N(C1=O)c1ncccc1OC)c1c(F)cc(OC)cc1F |r|
COCCn1cccc(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(Cl)ccc4C3)C2=O)c2c(F)cc(OC)cc2F)c1=O |r|
COc1ccc2CC(CCc2c1)NC(=O)N[C@H]1[C@@H](CN(C1=O)c1cccn(CCO)c1=O)c1c(F)cc(OC)cc1F |r|
COCCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(Cl)ccc4C3)C2=O)c2c(F)cc(OC)cc2F)c1=O |r,w:17.17|
COCCC1C=CC=C(N2[C@@H](C)[C@H]([C@H](NC(=O)NC3CCc4cc(Cl)ccc4C3)C2=O)c2c(F)cc(OC)cc2F)C1=O |r,c:5,t:7|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)NC2CCc3ccccc3C2)c2ncccc2C(F)(F)F)c(F)c1 |r|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(N3C[C@H](C)N(C)[C@H](C)C3)c2C(F)(F)F)c(F)c1 |r,wU:7.6,17.17,wD:37.39,33.35,12.13,20.24,(-6,8.62,;-6.63,7.21,;-5.72,5.96,;-6.35,4.56,;-5.44,3.31,;-6.07,1.9,;-3.91,3.47,;-3.01,2.22,;-3.48,.76,;-2.24,-.15,;-.99,.76,;.47,.28,;-1.47,2.22,;-.56,3.47,;.97,3.31,;1.6,1.9,;1.87,4.56,;3.41,4.39,;4.31,5.64,;5.84,5.48,;6.47,4.07,;5.56,2.83,;4.03,2.99,;8,3.91,;8.91,5.16,;8.63,2.5,;-2.24,-1.69,;-.9,-2.46,;-.9,-4,;-2.24,-4.77,;-3.57,-4,;-4.9,-4.77,;-4.9,-6.31,;-6.24,-7.08,;-6.24,-8.62,;-7.57,-6.31,;-8.91,-7.08,;-7.57,-4.77,;-8.91,-4,;-6.24,-4,;-3.62,-2.43,;-4.95,-1.66,;-6.29,-.89,;-5.72,-2.99,;-4.18,-.32,;-3.29,4.88,;-1.75,5.04,;-4.19,6.12,)|
COCCn1cccc(N2[C@@H](C)[C@H]([C@H](NC(=O)NC3CCc4cc(Cl)ccc4C3)C2=O)c2c(F)cc(OC)cc2F)c1=O |r|
COc1ccc2CC(COc2c1)NC(=O)N[C@H]1[C@@H](CN(C1=O)c1ncccc1C(F)(F)F)c1c(F)cc(OC)cc1F |r|
COCCn1cccc(N2[C@@H](C)[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3)C2=O)c2c(F)cc(OC)cc2F)c1=O |r|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(N3CCN(C)CC3)c2C(F)(F)F)c(F)c1 |r,wU:7.6,17.17,wD:12.13,20.24,(-6,7.85,;-6.63,6.44,;-5.72,5.19,;-6.35,3.79,;-5.44,2.54,;-6.07,1.13,;-3.91,2.7,;-3.01,1.45,;-3.48,-.01,;-2.24,-.92,;-.99,-.01,;.47,-.49,;-1.47,1.45,;-.56,2.7,;.97,2.54,;1.6,1.13,;1.87,3.79,;3.41,3.62,;4.31,4.87,;5.84,4.71,;6.47,3.3,;5.56,2.06,;4.03,2.22,;8,3.14,;8.91,4.39,;8.63,1.73,;-2.24,-2.46,;-.9,-3.23,;-.9,-4.77,;-2.24,-5.54,;-3.57,-4.77,;-4.9,-5.54,;-6.24,-4.77,;-7.57,-5.54,;-7.57,-7.08,;-8.91,-7.85,;-6.24,-7.85,;-4.9,-7.08,;-3.62,-3.2,;-4.95,-2.43,;-6.29,-1.66,;-5.72,-3.76,;-4.18,-1.09,;-3.29,4.11,;-1.75,4.27,;-4.19,5.35,)|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)NC2CC[C@@H](CC2)C(F)F)c2ncccc2C(F)(F)F)c(F)c1 |r,wU:7.6,20.24,wD:12.13,(-8.53,5.84,;-7,6,;-6.1,4.75,;-6.73,3.34,;-5.83,2.09,;-6.46,.69,;-4.3,2.25,;-3.4,1,;-3.88,-.47,;-2.64,-1.38,;-1.39,-.48,;.07,-.96,;-1.86,.99,;-.95,2.23,;.58,2.06,;1.2,.65,;1.49,3.3,;3.02,3.13,;3.64,1.72,;5.17,1.56,;6.09,2.8,;5.47,4.21,;3.94,4.38,;7.62,2.63,;8.24,1.22,;8.53,3.87,;-2.65,-2.92,;-1.32,-3.69,;-1.33,-5.23,;-2.66,-6,;-3.99,-5.22,;-3.99,-3.68,;-5.32,-2.9,;-6.65,-2.13,;-6.09,-4.23,;-4.54,-1.57,;-3.67,3.65,;-2.13,3.8,;-4.56,4.9,)|
COCCn1cccc(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3)C2=O)c2c(F)cc(OC)cc2F)c1=O |r|
COc1ccc(cc1)[C@H]1C[C@@H]1NC(=O)N[C@H]1[C@@H](CN(C1=O)c1ncccc1C(F)(F)F)c1c(F)cc(OC)cc1F |r|
COc1ccc2CC(COc2c1)NC(=O)N[C@H]1[C@@H](CN(C1=O)c1cccn(CCO)c1=O)c1c(F)cc(OC)cc1F |r|
CCn1cccc(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3)C2=O)c2c(F)cc(OC)cc2F)c1=O |r|
COCCn1ccc(OC)c(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(Cl)ccc4C3)C2=O)c2c(F)cc(OC)cc2F)c1=O |r,w:18.18|
COc1ccc2c(OCC(NC(=O)N[C@H]3[C@@H](CN(C3=O)c3cccn(CCO)c3=O)c3c(F)cc(OC)cc3F)C2(C)C)c1 |r,w:10.9|
COCCn1cccc(N2[C@@H](C)[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3(C)C)C2=O)c2c(F)cc(OC)cc2F)c1=O |r|
COCCn1cccc(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3)C2=O)c2ccc(Cl)cc2)c1=O |r|
COCCn1cccc(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3(C)C)C2=O)c2c(F)cc(OC)cc2F)c1=O |r|
COc1ccc2CC(CCc2c1)NC(=O)N[C@H]1[C@@H](CN(C1=O)c1ncccc1C(F)(F)F)c1c(F)cc(OC)cc1F |r,w:12.13|
COc1ccc2CC(CCc2c1)NC(=O)N[C@H]1[C@@H](CN(C1=O)c1ncccc1C(F)(F)F)c1c(F)cc(OC)cc1F |r|
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2ncccc2OC)c(F)c1 |r,wU:7.6,21.25,8.8,wD:13.14,18.18,(-8.53,5.83,;-7,5.99,;-6.1,4.74,;-6.72,3.33,;-5.82,2.09,;-6.44,.68,;-4.29,2.25,;-3.38,1,;-3.86,-.46,;-5.32,-.94,;-2.61,-1.37,;-1.36,-.46,;.1,-.94,;-1.84,1,;-.94,2.25,;.6,2.09,;1.22,.68,;1.5,3.33,;3.03,3.17,;3.66,1.77,;5.19,1.61,;6.1,2.85,;5.47,4.26,;3.94,4.42,;7.63,2.69,;8.53,3.94,;8.25,1.28,;-2.61,-2.91,;-3.94,-3.68,;-3.94,-5.22,;-2.61,-5.99,;-1.28,-5.22,;-1.28,-3.68,;.06,-2.91,;1.39,-3.68,;-3.66,3.66,;-2.13,3.82,;-4.56,4.9,)|
COCCn1ccc(OC)c(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3)C2=O)c2c(F)cc(OC)cc2F)c1=O |r,w:18.18|
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2ncccc2OC(C)C)c(F)c1 |r,wU:7.6,21.25,8.8,wD:13.14,18.18,(-8.53,5.83,;-7,5.99,;-6.1,4.74,;-6.72,3.33,;-5.82,2.09,;-6.44,.68,;-4.29,2.25,;-3.38,1,;-3.86,-.46,;-5.32,-.94,;-2.61,-1.37,;-1.36,-.46,;.1,-.94,;-1.84,1,;-.94,2.25,;.6,2.09,;1.22,.68,;1.5,3.33,;3.03,3.17,;3.66,1.77,;5.19,1.61,;6.1,2.85,;5.47,4.26,;3.94,4.42,;7.63,2.69,;8.53,3.94,;8.25,1.28,;-2.61,-2.91,;-3.94,-3.68,;-3.94,-5.22,;-2.61,-5.99,;-1.28,-5.22,;-1.28,-3.68,;.06,-2.91,;1.39,-3.68,;2.72,-2.91,;1.39,-5.22,;-3.66,3.66,;-2.13,3.82,;-4.56,4.9,)|
CCn1cccc(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3(C)C)C2=O)c2c(F)cc(OC)cc2F)c1=O |r|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)NCC2CCCCC2)c2ncccc2C(F)(F)F)c(F)c1 |r|
COc1ccc2CC(CCc2c1)NC(=O)N[C@H]1[C@@H](CN(C1=O)c1c(OC)ccn(C)c1=O)c1c(F)cc(OC)cc1F |r|
COc1ccc2c(CCC(NC(=O)N[C@H]3[C@@H](CN(C3=O)c3ncccc3C(F)(F)F)c3c(F)cc(OC)cc3F)C2(C)C)c1 |r|
COc1ccc2c(CCC(NC(=O)N[C@H]3[C@@H]([C@H](C)N(C3=O)c3ncccc3C(F)(F)F)c3c(F)cc(OC)cc3F)C2(C)C)c1 |r|
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2ncccc2F)c(F)c1 |r,wU:7.6,21.25,8.8,wD:13.14,18.18,(-8.53,5.83,;-7,5.99,;-6.1,4.74,;-6.72,3.33,;-5.82,2.09,;-6.44,.68,;-4.29,2.25,;-3.38,1,;-3.86,-.46,;-5.32,-.94,;-2.61,-1.37,;-1.36,-.46,;.1,-.94,;-1.84,1,;-.94,2.25,;.6,2.09,;1.22,.68,;1.5,3.33,;3.03,3.17,;3.66,1.77,;5.19,1.61,;6.1,2.85,;5.47,4.26,;3.94,4.42,;7.63,2.69,;8.53,3.94,;8.25,1.28,;-2.61,-2.91,;-3.94,-3.68,;-3.94,-5.22,;-2.61,-5.99,;-1.28,-5.22,;-1.28,-3.68,;.06,-2.91,;-3.66,3.66,;-2.13,3.82,;-4.56,4.9,)|
COCC(CO)n1cccc(N2[C@@H](C)[C@H]([C@H](NC(=O)N[C@H]3CC[C@@H](CC3)C(F)F)C2=O)c2c(F)cc(OC)cc2F)c1=O |r,wU:14.32,23.26,12.12,wD:15.15,20.19,(2.72,-6.37,;1.39,-7.14,;.06,-6.37,;.06,-4.83,;1.39,-4.06,;2.72,-4.83,;-1.28,-4.06,;-2.61,-4.83,;-3.94,-4.06,;-3.94,-2.52,;-2.61,-1.75,;-2.61,-.21,;-3.86,.69,;-5.32,.22,;-3.38,2.16,;-1.84,2.16,;-.94,3.4,;.6,3.24,;1.22,1.84,;1.5,4.49,;3.03,4.33,;3.66,2.92,;5.19,2.76,;6.1,4.01,;5.47,5.41,;3.94,5.57,;7.63,3.84,;8.53,5.09,;8.25,2.44,;-1.36,.69,;.1,.22,;-4.29,3.4,;-5.82,3.24,;-6.44,1.84,;-6.72,4.49,;-6.1,5.9,;-7,7.14,;-8.53,6.98,;-4.56,6.06,;-3.66,4.81,;-2.13,4.97,;-1.28,-2.52,;.06,-1.75,)|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2cccn(CCO)c2=O)c(F)c1 |r,wU:7.6,20.24,wD:12.13,17.17,(-6.35,6.76,;-7.03,5.37,;-6.17,4.09,;-6.85,2.71,;-5.99,1.43,;-6.67,.05,;-4.45,1.54,;-3.6,.26,;-4.13,-1.19,;-2.91,-2.14,;-1.64,-1.28,;-.19,-1.81,;-2.06,.2,;-1.11,1.41,;.42,1.19,;.99,-.24,;1.37,2.41,;2.89,2.19,;3.47,.76,;4.99,.54,;5.94,1.75,;5.37,3.18,;3.84,3.4,;7.47,1.53,;8.42,2.74,;8.04,.1,;-2.97,-3.68,;-1.67,-4.5,;-1.73,-6.04,;-3.09,-6.76,;-4.39,-5.94,;-5.75,-6.66,;-7.06,-5.84,;-8.42,-6.56,;-4.33,-4.4,;-5.64,-3.58,;-3.78,2.92,;-2.24,3.02,;-4.63,4.2,)|
COc1cc(F)c([C@@H]2[C@@H](C)N(C(=O)[C@H]2NC(=O)NCC2CCCCC2)c2ncccc2OC)c(F)c1 |r|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)NC2CCC3(CC3)CC2)c2ncccc2C(F)(F)F)c(F)c1 |r|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(NC3CCOCC3)c2C(F)(F)F)c(F)c1 |r,wU:7.6,20.24,wD:12.13,17.17,(-8.53,8.14,;-7,8.3,;-6.1,7.05,;-6.72,5.64,;-5.82,4.4,;-6.44,2.99,;-4.29,4.56,;-3.38,3.31,;-3.86,1.85,;-2.61,.94,;-1.36,1.85,;.1,1.37,;-1.84,3.31,;-.94,4.56,;.6,4.4,;1.22,2.99,;1.5,5.64,;3.03,5.48,;3.66,4.08,;5.19,3.92,;6.1,5.16,;5.47,6.57,;3.94,6.73,;7.63,5,;8.53,6.25,;8.25,3.59,;-2.61,-.6,;-1.28,-1.37,;-1.28,-2.91,;-2.61,-3.68,;-3.94,-2.91,;-5.28,-3.68,;-5.28,-5.22,;-6.61,-5.99,;-6.61,-7.53,;-5.28,-8.3,;-3.94,-7.53,;-3.94,-5.99,;-3.99,-1.34,;-5.33,-.57,;-6.66,.2,;-6.1,-1.9,;-4.56,.76,;-3.66,5.97,;-2.13,6.13,;-4.56,7.21,)|
COCCNc1ccnc(N2C[C@H]([C@H](NC(=O)N[C@H]3CC[C@@H](CC3)C(F)F)C2=O)c2c(F)cc(OC)cc2F)c1C(F)(F)F |r,wU:12.30,21.24,wD:13.13,18.17,(-8.24,-4.8,;-8.28,-6.34,;-6.97,-7.14,;-5.61,-6.41,;-5.57,-4.87,;-4.22,-4.14,;-2.91,-4.94,;-1.55,-4.21,;-1.51,-2.67,;-2.82,-1.87,;-2.78,-.33,;-4,.61,;-3.49,2.06,;-1.95,2.02,;-1.01,3.24,;.52,3.04,;1.11,1.62,;1.46,4.26,;2.99,4.06,;3.57,2.63,;5.1,2.43,;6.04,3.65,;5.45,5.08,;3.92,5.28,;7.57,3.45,;8.5,4.67,;8.15,2.03,;-1.51,.54,;-.06,.03,;-4.36,3.33,;-5.89,3.21,;-6.56,1.83,;-6.76,4.49,;-6.1,5.87,;-6.97,7.14,;-8.5,7.03,;-4.56,5.99,;-3.69,4.72,;-2.16,4.84,;-4.22,-2.57,;-5.54,-1.76,;-6.85,-.96,;-6.34,-3.08,;-4.73,-.45,)|
COCCn1cccc(N2C[C@H]([C@H](NC(=O)N[C@H]3CC[C@@H](CC3)C(F)F)C2=O)c2c(F)cc(OC)cc2F)c1=O |r,wU:11.29,20.23,wD:12.12,17.16,(-9.04,-5.9,;-7.71,-6.67,;-6.37,-5.9,;-5.04,-6.67,;-3.68,-5.93,;-2.37,-6.74,;-1.02,-6.01,;-.98,-4.47,;-2.29,-3.66,;-2.25,-2.12,;-3.47,-1.18,;-2.95,.27,;-1.41,.23,;-.47,1.45,;1.05,1.25,;1.64,-.18,;1.99,2.47,;3.52,2.26,;4.11,.84,;5.63,.64,;6.57,1.86,;5.99,3.28,;4.46,3.48,;8.1,1.65,;9.04,2.88,;8.69,.23,;-.98,-1.25,;.48,-1.77,;-3.82,1.54,;-5.36,1.42,;-6.02,.03,;-6.23,2.69,;-5.56,4.08,;-6.43,5.35,;-5.77,6.74,;-4.03,4.2,;-3.16,2.93,;-1.62,3.05,;-3.64,-4.39,;-4.95,-3.59,)|
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2cccn(CCO)c2=O)c(F)c1 |r,wU:7.6,21.25,8.8,wD:13.14,18.18,(-8.53,5.83,;-7,5.99,;-6.1,4.74,;-6.72,3.33,;-5.82,2.09,;-6.44,.68,;-4.29,2.25,;-3.38,1,;-3.86,-.46,;-5.32,-.94,;-2.61,-1.37,;-1.36,-.46,;.1,-.94,;-1.84,1,;-.94,2.25,;.6,2.09,;1.22,.68,;1.5,3.33,;3.03,3.17,;3.66,1.77,;5.19,1.61,;6.1,2.85,;5.47,4.26,;3.94,4.42,;7.63,2.69,;8.53,3.94,;8.25,1.28,;-2.61,-2.91,;-1.28,-3.68,;-1.28,-5.22,;-2.61,-5.99,;-3.94,-5.22,;-5.28,-5.99,;-6.61,-5.22,;-7.95,-5.99,;-3.94,-3.68,;-5.28,-2.91,;-3.66,3.66,;-2.13,3.82,;-4.56,4.9,)|
CNC(=O)CNc1ccnc(N2C[C@H]([C@H](NC(=O)N[C@H]3CC[C@@H](CC3)C(F)F)C2=O)c2c(F)cc(OC)cc2F)c1C(F)(F)F |r,wU:13.31,22.25,wD:14.14,19.18,(-9.57,-5.22,;-8.24,-4.45,;-6.91,-5.22,;-6.91,-6.76,;-5.57,-4.45,;-4.24,-5.22,;-2.9,-4.45,;-1.57,-5.22,;-.24,-4.45,;-.24,-2.91,;-1.57,-2.14,;-1.57,-.6,;-2.82,.31,;-2.34,1.77,;-.8,1.77,;.1,3.02,;1.64,2.86,;2.26,1.45,;2.54,4.1,;4.07,3.94,;4.7,2.54,;6.23,2.38,;7.14,3.62,;6.51,5.03,;4.98,5.19,;8.67,3.46,;9.57,4.71,;9.29,2.05,;-.32,.31,;1.14,-.17,;-3.25,3.02,;-4.78,2.86,;-5.4,1.45,;-5.68,4.1,;-5.06,5.51,;-5.96,6.76,;-7.49,6.6,;-3.52,5.67,;-2.62,4.43,;-1.09,4.59,;-2.95,-2.88,;-4.29,-2.11,;-5.62,-1.34,;-5.06,-3.44,;-3.52,-.78,)|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(NCC3CCOC3)c2C(F)(F)F)c(F)c1 |r,wU:7.6,20.24,wD:12.13,17.17,(-7.61,6.75,;-6.08,6.91,;-5.17,5.67,;-5.8,4.26,;-4.89,3.01,;-5.52,1.61,;-3.36,3.17,;-2.46,1.93,;-2.93,.46,;-1.69,-.44,;-.44,.46,;1.02,-.01,;-.92,1.93,;-.01,3.17,;1.52,3.01,;2.15,1.61,;2.43,4.26,;3.96,4.1,;4.58,2.69,;6.12,2.53,;7.02,3.78,;6.39,5.18,;4.86,5.34,;8.55,3.62,;9.46,4.86,;9.18,2.21,;-1.69,-1.98,;-.35,-2.75,;-.35,-4.29,;-1.69,-5.06,;-3.02,-4.29,;-4.35,-5.06,;-5.69,-4.29,;-7.02,-5.06,;-7.18,-6.59,;-8.69,-6.91,;-9.46,-5.58,;-8.43,-4.43,;-3.07,-2.72,;-4.4,-1.95,;-5.73,-1.18,;-5.17,-3.29,;-3.63,-.62,;-2.73,4.58,;-1.2,4.74,;-3.64,5.83,)|
CNC(=O)C(C)Nc1ccnc(N2C[C@H]([C@H](NC(=O)N[C@H]3CC[C@@H](CC3)C(F)F)C2=O)c2c(F)cc(OC)cc2F)c1C(F)(F)F |r,wU:14.32,23.26,wD:15.15,20.19,(-8.78,-6.69,;-7.69,-5.6,;-6.36,-6.37,;-6.36,-7.91,;-5.03,-5.6,;-3.69,-6.37,;-5.03,-4.06,;-3.69,-3.29,;-2.36,-4.06,;-1.03,-3.29,;-1.03,-1.75,;-2.36,-.98,;-2.36,.56,;-3.61,1.46,;-3.13,2.93,;-1.59,2.93,;-.68,4.17,;.85,4.01,;1.47,2.61,;1.75,5.26,;3.28,5.1,;3.91,3.69,;5.44,3.53,;6.35,4.78,;5.72,6.18,;4.19,6.34,;7.88,4.61,;8.78,5.86,;8.5,3.21,;-1.11,1.46,;.35,.99,;-4.03,4.17,;-5.57,4.01,;-6.19,2.61,;-6.47,5.26,;-5.85,6.67,;-6.75,7.91,;-8.28,7.75,;-4.31,6.83,;-3.41,5.58,;-1.88,5.74,;-3.74,-1.72,;-5.08,-.95,;-6.41,-.18,;-5.85,-2.29,;-4.3,.38,)|
COc1ccc2CC(CCc2c1)NC(=O)N[C@H]1[C@@H](CN(C1=O)c1cccn(CC(O)C(F)(F)F)c1=O)c1c(F)cc(OC)cc1F |r|
COCC(CO)n1cccc(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3)C2=O)c2c(F)cc(OC)cc2F)c1=O |r|
COc1ccc2CC(CCc2c1)NC(=O)N[C@H]1[C@@H](CN(C1=O)c1c(C)ccn(CCO)c1=O)c1c(F)cc(OC)cc1F |r|
COCCn1nccc(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3)C2=O)c2c(F)cc(OC)cc2F)c1=O |r|
CCn1nccc(N2C[C@H]([C@H](NC(=O)NC3CCc4cc(OC)ccc4C3)C2=O)c2c(F)cc(OC)cc2F)c1=O |r|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(N3CCN(CC3)S(C)(=O)=O)c2C(F)(F)F)c(F)c1 |r,wU:7.6,20.24,wD:12.13,17.17,(-7.49,7.65,;-5.96,7.81,;-5.06,6.56,;-5.68,5.16,;-4.78,3.91,;-5.4,2.5,;-3.25,4.07,;-2.34,2.83,;-2.82,1.36,;-1.57,.46,;-.32,1.36,;1.14,.88,;-.8,2.83,;.1,4.07,;1.64,3.91,;2.26,2.5,;2.54,5.16,;4.07,4.99,;4.7,3.59,;6.23,3.43,;7.14,4.67,;6.51,6.08,;4.98,6.24,;8.67,4.51,;9.57,5.76,;9.29,3.11,;-1.57,-1.08,;-.24,-1.85,;-.24,-3.39,;-1.57,-4.16,;-2.9,-3.39,;-4.24,-4.16,;-5.57,-3.39,;-6.91,-4.16,;-6.91,-5.7,;-5.57,-6.47,;-4.24,-5.7,;-8.24,-6.47,;-9.57,-7.24,;-9.01,-5.14,;-7.47,-7.81,;-2.95,-1.83,;-4.29,-1.06,;-5.62,-.29,;-5.06,-2.39,;-3.52,.28,;-2.62,5.48,;-1.09,5.64,;-3.52,6.72,)|
COc1ccc2CC(CCc2c1)NC(=O)N[C@H]1[C@@H]([C@H](C)N(C1=O)c1cccn(CCO)c1=O)c1c(F)cc(OC)cc1F |r|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(N3CCC(C)(O)C3)c2C(F)(F)F)c(F)c1 |r,wU:7.6,20.24,wD:12.13,17.17,(-8.24,6.75,;-6.71,6.91,;-5.8,5.67,;-6.43,4.26,;-5.52,3.01,;-6.15,1.61,;-3.99,3.17,;-3.09,1.93,;-3.56,.46,;-2.32,-.44,;-1.07,.46,;.39,-.01,;-1.55,1.93,;-.64,3.17,;.89,3.01,;1.52,1.61,;1.8,4.26,;3.33,4.1,;3.95,2.69,;5.49,2.53,;6.39,3.78,;5.76,5.18,;4.23,5.34,;7.92,3.62,;8.83,4.86,;8.55,2.21,;-2.32,-1.98,;-.98,-2.75,;-.98,-4.29,;-2.32,-5.06,;-3.65,-4.29,;-4.98,-5.06,;-5.14,-6.59,;-6.65,-6.91,;-7.42,-5.58,;-8.83,-6.21,;-8.67,-4.67,;-6.39,-4.43,;-3.7,-2.72,;-5.03,-1.95,;-6.37,-1.18,;-5.8,-3.29,;-4.26,-.62,;-3.36,4.58,;-1.83,4.74,;-4.27,5.83,)|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(NCC3CCCO3)c2C(F)(F)F)c(F)c1 |r,wU:7.6,20.24,wD:12.13,17.17,(-8.27,7.91,;-6.74,8.07,;-5.84,6.82,;-6.46,5.41,;-5.56,4.17,;-6.19,2.76,;-4.03,4.33,;-3.12,3.08,;-3.6,1.62,;-2.35,.71,;-1.11,1.62,;.36,1.14,;-1.58,3.08,;-.68,4.33,;.85,4.17,;1.48,2.76,;1.76,5.41,;3.29,5.25,;3.92,3.85,;5.45,3.69,;6.35,4.93,;5.73,6.34,;4.2,6.5,;7.89,4.77,;8.79,6.02,;8.51,3.36,;-2.35,-.83,;-1.02,-1.6,;-1.02,-3.14,;-2.35,-3.91,;-3.69,-3.14,;-5.02,-3.91,;-5.02,-5.45,;-6.35,-6.22,;-6.51,-7.75,;-8.02,-8.07,;-8.79,-6.73,;-7.76,-5.59,;-3.73,-1.57,;-5.07,-.8,;-6.4,-.03,;-5.84,-2.13,;-4.3,.54,;-3.4,5.74,;-1.87,5.9,;-4.31,6.98,)|
COc1ccc2CC(CCc2c1)NC(=O)N[C@H]1[C@@H](CN(C1=O)c1cccn(C(F)F)c1=O)c1c(F)cc(OC)cc1F |r|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(N3C[C@@H]4C[C@H]3CN4C)c2C(F)(F)F)c(F)c1 |r,wU:7.6,20.24,wD:12.13,17.17,35.36,33.35,(-8.16,6.98,;-6.63,7.14,;-5.72,5.9,;-6.35,4.49,;-5.44,3.24,;-6.07,1.84,;-3.91,3.4,;-3.01,2.16,;-3.48,.69,;-2.24,-.21,;-.99,.69,;.47,.22,;-1.47,2.16,;-.56,3.4,;.97,3.24,;1.6,1.84,;1.87,4.49,;3.41,4.33,;4.03,2.92,;5.56,2.76,;6.47,4.01,;5.84,5.41,;4.31,5.57,;8,3.84,;8.91,5.09,;8.63,2.44,;-2.24,-1.75,;-.9,-2.52,;-.9,-4.06,;-2.24,-4.83,;-3.57,-4.06,;-4.9,-4.83,;-4.9,-6.37,;-6.24,-7.14,;-5.84,-5.59,;-6.24,-4.06,;-7.57,-4.83,;-7.57,-6.37,;-8.91,-7.14,;-3.62,-2.49,;-4.95,-1.72,;-6.29,-.95,;-5.72,-3.06,;-4.18,-.39,;-3.29,4.81,;-1.75,4.97,;-4.19,6.06,)|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(NCCS(C)(=O)=O)c2C(F)(F)F)c(F)c1 |r,wU:7.6,20.24,wD:12.13,17.17,(-8.01,7.33,;-6.47,7.49,;-5.57,6.24,;-6.2,4.83,;-5.29,3.59,;-5.92,2.18,;-3.76,3.75,;-2.85,2.5,;-3.33,1.04,;-2.08,.13,;-.84,1.04,;.63,.56,;-1.31,2.5,;-.41,3.75,;1.12,3.59,;1.75,2.18,;2.03,4.83,;3.56,4.67,;4.19,3.27,;5.72,3.11,;6.62,4.35,;6,5.76,;4.47,5.92,;8.15,4.19,;9.06,5.44,;8.78,2.78,;-2.08,-1.41,;-.75,-2.18,;-.75,-3.72,;-2.08,-4.49,;-3.42,-3.72,;-4.75,-4.49,;-4.75,-6.03,;-6.08,-6.8,;-7.57,-6.4,;-8.66,-7.49,;-7.97,-4.91,;-9.06,-6,;-3.47,-2.15,;-4.8,-1.38,;-6.13,-.61,;-5.57,-2.71,;-4.03,-.05,;-3.13,5.16,;-1.6,5.32,;-4.04,6.4,)|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(NC3CCOC3)c2C(F)(F)F)c(F)c1 |r,wU:7.6,20.24,wD:12.13,17.17,(-8.53,7.78,;-7,7.94,;-6.1,6.7,;-6.72,5.29,;-5.82,4.04,;-6.44,2.64,;-4.29,4.2,;-3.38,2.96,;-3.86,1.49,;-2.61,.59,;-1.36,1.49,;.1,1.02,;-1.84,2.96,;-.94,4.2,;.6,4.04,;1.22,2.64,;1.5,5.29,;3.03,5.13,;3.66,3.72,;5.19,3.56,;6.1,4.81,;5.47,6.21,;3.94,6.37,;7.63,4.65,;8.53,5.89,;8.25,3.24,;-2.61,-.95,;-1.28,-1.72,;-1.28,-3.26,;-2.61,-4.03,;-3.94,-3.26,;-5.28,-4.03,;-5.28,-5.57,;-4.03,-6.48,;-4.51,-7.94,;-6.05,-7.94,;-6.52,-6.48,;-3.99,-1.69,;-5.33,-.92,;-6.66,-.15,;-6.1,-2.26,;-4.56,.41,;-3.66,5.61,;-2.13,5.77,;-4.56,6.86,)|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(N3CC(C)(O)C3)c2C(F)(F)F)c(F)c1 |r,wU:7.6,20.24,wD:12.13,17.17,(-8.53,6.76,;-7,6.92,;-6.1,5.67,;-6.72,4.26,;-5.82,3.02,;-6.44,1.61,;-4.29,3.18,;-3.38,1.93,;-3.86,.47,;-2.61,-.44,;-1.36,.47,;.1,-.01,;-1.84,1.93,;-.94,3.18,;.6,3.02,;1.22,1.61,;1.5,4.26,;3.03,4.1,;3.66,2.7,;5.19,2.53,;6.1,3.78,;5.47,5.19,;3.94,5.35,;7.63,3.62,;8.53,4.87,;8.25,2.21,;-2.61,-1.98,;-1.28,-2.75,;-1.28,-4.29,;-2.61,-5.06,;-3.94,-4.29,;-5.28,-5.06,;-6.77,-4.66,;-7.16,-6.15,;-8.5,-6.92,;-8.39,-5.21,;-5.68,-6.54,;-3.99,-2.72,;-5.33,-1.95,;-6.66,-1.18,;-6.1,-3.28,;-4.56,-.62,;-3.66,4.59,;-2.13,4.75,;-4.56,5.83,)|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(N3CCN4CCCC4C3)c2C(F)(F)F)c(F)c1 |r,wU:7.6,20.24,wD:12.13,17.17,(-8.25,7.81,;-6.72,7.98,;-5.82,6.73,;-6.44,5.32,;-5.54,4.08,;-6.17,2.67,;-4.01,4.24,;-3.1,2.99,;-3.58,1.53,;-2.33,.62,;-1.09,1.53,;.38,1.05,;-1.56,2.99,;-.66,4.24,;.87,4.08,;1.5,2.67,;1.78,5.32,;3.31,5.16,;3.94,3.75,;5.47,3.59,;6.37,4.84,;5.75,6.25,;4.22,6.41,;7.91,4.68,;8.81,5.92,;8.53,3.27,;-2.33,-.92,;-1,-1.69,;-1,-3.23,;-2.33,-4,;-3.67,-3.23,;-5,-4,;-6.33,-3.23,;-7.67,-4,;-7.67,-5.54,;-8.81,-6.57,;-8.18,-7.98,;-6.65,-7.81,;-6.33,-6.31,;-5,-5.54,;-3.71,-1.66,;-5.05,-.89,;-6.38,-.12,;-5.82,-2.22,;-4.28,.44,;-3.38,5.64,;-1.85,5.81,;-4.29,6.89,)|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(NCC(C)(C)O)c2C(F)(F)F)c(F)c1 |r,wU:7.6,20.24,wD:12.13,17.17,(-8.5,7.71,;-6.96,7.82,;-6.1,6.55,;-6.77,5.16,;-5.9,3.89,;-6.57,2.5,;-4.37,4,;-3.5,2.73,;-4.02,1.28,;-2.81,.33,;-1.53,1.2,;-.08,.68,;-1.96,2.68,;-1.02,3.89,;.51,3.68,;1.09,2.26,;1.45,4.9,;2.98,4.69,;3.56,3.27,;5.08,3.06,;6.03,4.27,;5.45,5.7,;3.92,5.91,;7.55,4.06,;8.5,5.28,;8.14,2.64,;-2.86,-1.21,;-1.55,-2.02,;-1.6,-3.56,;-2.95,-4.28,;-4.26,-3.47,;-5.62,-4.2,;-5.67,-5.74,;-7.03,-6.47,;-7.84,-7.77,;-6.3,-7.82,;-8.34,-5.65,;-4.26,-1.9,;-5.57,-1.09,;-6.88,-.28,;-6.38,-2.4,;-4.76,.22,;-3.7,5.39,;-2.16,5.5,;-4.56,6.66,)|
COCCn1cccc(N2[C@@H](C)[C@H]([C@H](NC(=O)N[C@H]3CC[C@@H](CC3)C(F)F)C2=O)c2c(F)cc(OC)cc2F)c1=O |r,wU:12.30,21.24,10.10,wD:13.13,18.17,(-7.95,-6.76,;-7.95,-5.22,;-6.61,-4.45,;-5.28,-5.22,;-3.94,-4.45,;-2.61,-5.22,;-1.28,-4.45,;-1.28,-2.91,;-2.61,-2.14,;-2.61,-.6,;-3.86,.31,;-5.32,-.17,;-3.38,1.77,;-1.84,1.77,;-.94,3.02,;.6,2.86,;1.22,1.45,;1.5,4.1,;3.03,3.94,;3.66,2.54,;5.19,2.38,;6.1,3.62,;5.47,5.03,;3.94,5.19,;7.63,3.46,;8.53,4.71,;8.25,2.05,;-1.36,.31,;.1,-.17,;-4.29,3.02,;-5.82,2.86,;-6.44,1.45,;-6.72,4.1,;-6.1,5.51,;-7,6.76,;-8.53,6.6,;-4.56,5.67,;-3.66,4.43,;-2.13,4.59,;-3.94,-2.91,;-5.28,-2.14,)|
COCC(CO)n1ccnc(N2C[C@H]([C@H](NC(=O)N[C@H]3CC[C@@H](CC3)C(F)F)C2=O)c2c(F)cc(OC)cc2F)c1=O |r,wU:13.31,22.25,wD:14.14,19.18,(-4.24,-8.62,;-4.24,-7.08,;-5.57,-6.31,;-5.57,-4.77,;-6.91,-4,;-8.24,-4.77,;-4.24,-4,;-2.9,-4.77,;-1.57,-4,;-1.57,-2.46,;-2.9,-1.69,;-2.9,-.15,;-4.15,.76,;-3.67,2.22,;-2.13,2.22,;-1.23,3.47,;.3,3.31,;.93,1.9,;1.21,4.56,;2.74,4.39,;3.37,2.99,;4.9,2.83,;5.8,4.07,;5.18,5.48,;3.64,5.64,;7.33,3.91,;8.24,5.16,;7.96,2.5,;-1.66,.76,;-.19,.28,;-4.58,3.47,;-6.11,3.31,;-6.74,1.9,;-7.02,4.56,;-6.39,5.96,;-7.3,7.21,;-6.67,8.62,;-4.86,6.12,;-3.95,4.88,;-2.42,5.04,;-4.24,-2.46,;-5.57,-1.69,)|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)N[C@H]2CC[C@@H](CC2)C(F)F)c2nccc(N3CCOCC3)c2C(F)(F)F)c(F)c1 |r,wU:7.6,20.24,wD:12.13,17.17,(-8.5,7.01,;-6.96,7.12,;-6.1,5.85,;-6.77,4.46,;-5.9,3.19,;-6.57,1.8,;-4.37,3.3,;-3.5,2.03,;-4.02,.58,;-2.81,-.37,;-1.53,.5,;-.08,-.02,;-1.96,1.98,;-1.02,3.19,;.51,2.98,;1.09,1.56,;1.45,4.2,;2.98,3.99,;3.56,2.56,;5.08,2.35,;6.03,3.57,;5.45,5,;3.92,5.21,;7.55,3.36,;8.5,4.58,;8.14,1.94,;-2.86,-1.91,;-1.55,-2.72,;-1.6,-4.26,;-2.95,-4.99,;-4.26,-4.17,;-5.62,-4.9,;-6.9,-4.05,;-8.28,-4.73,;-8.38,-6.27,;-7.1,-7.12,;-5.72,-6.44,;-4.26,-2.61,;-5.57,-1.79,;-6.88,-.98,;-6.38,-3.1,;-4.76,-.48,;-3.7,4.69,;-2.16,4.8,;-4.56,5.96,)|
COc1cc(F)c(C2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccnc2C#N)c(F)c1
COc1cc(F)c(C2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccc(=O)n(C)c2)c(F)c1
COc1cc(F)c(C2CN(CC3CC3)C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CC(O)C(F)(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(Cl)ccc2C#N)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ncccc2C(F)(F)F)c(F)c1
COc1ccc(F)c(c1)N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)(F)F)cc2)C1=O)c1c(F)cc(OC)cc1F
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(cc2)C(F)(F)F)c2ncccc2F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(=O)n2C)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccc(=O)n2C)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(Cl)cc(c2)C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cc(ccn2)P(C)(C)=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cc(F)cc(OC(C)C)c2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ncccc2C#N)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(Cl)cc(OC(C)C)c2)c(F)c1
COc1cc(F)c([C@@H]2CN(Cc3ccccc3P(C)(C)=O)C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c(F)c1
COc1cc(F)c([C@@H]2CN(Cc3ccccc3P(C)(C)=O)C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ccccc2P(C)(C)=O)c(F)c1
COc1cc(F)c([C@@H]2CN(CC3CC3)C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccnc2C#N)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ncccc2P(C)(C)=O)c(F)c1
COc1ccnc(c1)N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)(F)F)cc2)C1=O)c1c(F)cc(OC)cc1F
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccc(n2)C(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ncccc2P(C)(C)=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ccc(=O)n(C)c2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ncccc2CO)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ncccc2F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(F)cc(OC(C)C)c2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccnc2P(C)(C)=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccccc2P(C)(C)=O)c(F)c1
COc1ccnc(c1)N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)F)cc2)C1=O)c1c(F)cc(OC)cc1F
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ncccc2F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(C)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)N2CCN(C)CC2)c(F)c1
COCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
CCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2ncccc2OC)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(OC)cc(n2)N2C[C@@H]3C[C@H]2CN3C)c(F)c1 |THB:29:31:37.36:34,38:37:31.32:34|
COCC(CN)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2C[C@H](C)N(C)[C@H](C)C2)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2ncccc2OC(C)C)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CC(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2CCC2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CC(O)C(F)(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)N2C[C@H](C)N(C)[C@H](C)C2)c(F)c1
COc1cc(F)c([C@@H]2[C@@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(OC)cc(n2)N2C[C@@H]3C[C@H]2CN3C)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2C[C@H]3C[C@@H]2CN3C)c(F)c1 |TLB:28:33:38.39:36,40:39:33.34:36|
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)N2C[C@@H]3C[C@H]2CN3C)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(C(F)F)c2=O)c(F)c1
COCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2CCN(C)CC2)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CCC(F)(F)F)c2=O)c(F)c1
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)(F)F)cc1)c1c(C)ccn(CC2CC2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2nc(ccc2F)N2CCOCC2=O)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CC(F)F)c2=O)c(F)c1
COCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(C)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2nc(NC3CCOC3)ccc2F)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CCO)c2=O)c(F)c1
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)(F)F)cc1)c1cccn(CCO)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccnc(N3C[C@@H]4C[C@H]3CN4C)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2C3CCCC3C2=O)c(F)c1
CCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)C2=CC=NC(C2C#N)N2CCN(C)CC2)c(F)c1 |c:30,t:28|
FC(F)Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(OC)cc(n2)N2C[C@@H]3C[C@H]2CN3C)c(F)c1
COc1cc(F)c([C@@H]2[C@@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)N2C[C@@H]3C[C@H]2CN3C)c(F)c1
FC(F)Oc1ccc(cc1)C(=O)N[C@H]1[C@@H](CN(C1=O)c1cccn(CCC(F)(F)F)c1=O)c1ccc(Cl)cc1
FC(F)(F)CCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COCCn1cccc(N2[C@@H](C)[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CCC(F)(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2ncccc2OC)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ncccc2OC)c(F)c1
COCC(CN)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
CCn1cccc(N2[C@@H](C)[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2F)c1=O
CCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2F)c1=O
CCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CCN(C)C)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CC(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2ccc[nH]c2=O)c(F)c1
CCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CC(C)O)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CC(F)F)c2=O)c(F)c1
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)F)cc1)c1cccn(CC(F)F)c1=O
COCC(C(=O)N(C)C)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
CCn1cccc(N2[C@@H](C)[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccn(C(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccc[nH]c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CC3CC(F)(F)C3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CCN(C)C)c2=O)c(F)c1
CCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CCN3CCOCC3)c2=O)c(F)c1
COCCn1cccc(N2[C@@H](C)[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2CC(C)OCC2=O)c(F)c1
OCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COC(C)Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CC(C)O)c2=O)c(F)c1
COCCn1cccc(N2[C@@H](C)[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(OC)cc(NCCO)n2)c(F)c1
COCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)(F)F)cc1)c1c(C)ccn(CCO)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nccc(N3C[C@H](C)N(C)[C@H](C)C3)c2C(F)(F)F)c(F)c1
OCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nc(C)ccc2F)c(F)c1
COCC(CO)n1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2nc(ccc2F)N(C)C(C)=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CCO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(cc2)C(F)(F)F)c2cccn(C3CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2CC(F)(F)C2)c(F)c1
COCC(CO)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)(F)F)cc1)c1cccn(CC(F)F)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)(F)F)cc1)c1c(C)ccn(CC(F)F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(NC3CCOC3)ccc2F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccnc2OC(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2nc(ccc2F)N2CC(C)OCC2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(NC3CCOC3)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ncccc2OC(C)C)c(F)c1
COCCn1cccc(N2[C@H](C)[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
CCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nccc(NCC(C)O)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccn(CCO)c2=O)c(F)c1
COCC(C(=O)N1CCOCC1)n1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O |w:3.2|
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)(F)F)cc1)c1c(C)ccn(C2CCOC2)c1=O |w:33.36|
COCC(CO)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COCC(C(=O)N(C)C)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2CCC(O)C2=O)c(F)c1
COCC(CO)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
COCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccc(CO)[nH]c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2ccc(C)n(C)c2=O)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CCO)c2=O)c(F)c1
COCC(CO)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CC(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(NC(C)=O)ccc2F)c(F)c1
COC(Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O)C(F)(F)F
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CC(F)F)c2=O)c(F)c1
COCC(C(=O)N(C)C)n1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O |w:2.2|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CC3CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccnc(N3C[C@H](C)N(C)[C@H](C)C3)c2C(F)(F)F)c(F)c1
COCC(CO)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccnc2OC2CCOC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2CCCS2(=O)=O)c(F)c1
CCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(cc3)C(F)(F)F)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(N3C[C@@H]4C[C@H]3CN4C)c2C#N)c(F)c1
COC(Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O)C(F)(F)F
COCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(NC3CC3)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CCN3CC4(COC4)C3)c2=O)c(F)c1
CCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(NCC(C)(C)O)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(N3C[C@H](C)N(C)[C@H](C)C3)c2C#N)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(cn(C)c2=O)C(F)(F)F)c(F)c1
CCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ncccc2F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CCO)c2=O)c(F)c1
COCC(CO)n1cccc(N2[C@@H](C)[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CC(C)O)c2=O)c(F)c1 |w:33.35|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N(C)C(C)=O)c(F)c1
COCCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CC(C)(CO)CO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(OC)cc(n2)N2C[C@H](C)N(C)[C@H](C)C2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(N3C[C@H](C)N(C)[C@H](C)C3)c2C(F)(F)F)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CC(F)F)c2=O)c(F)c1
CCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccc(OC(F)F)c2)c(F)c1
COCCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CC(C)(CO)CO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(C(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(Cl)cn(C)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CC(F)(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CC(F)(F)F)c2=O)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CC3CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccn(C)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CC3CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(Cl)ccn(C)c2=O)c(F)c1
CCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CCC(F)(F)F)c2=O)c(F)c1
COCCn1cccc(N2[C@H](C)[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(C3CCOC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccnc2OCCN2CC3(COC3)C2)c(F)c1
COc1cc(F)c([C@@H]2[C@@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2ncccc2OC)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2C)C(F)(F)F)c(F)c1
CCn1cc(F)cc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2nc(NC(C)=O)ccc2F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(cn(C)c2=O)C#N)c(F)c1
COCCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2CC3(COC3)C2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CCN3CC4(COC4)C3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)N2C[C@H]3C[C@@H]2CO3)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nc(ccc2N2CC[C@H](O)C2)C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)N2C[C@H](C)N(C)[C@H](C)C2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)N2C[C@H](C)N(C)[C@H](C)C2)c(F)c1
CCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(C)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COCC(CO)n1cccc(N2[C@@H](C)[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CCO)c2=O)c(F)c1
COCCn1cccc(N2[C@H](C)[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CCF)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2ncccc2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2OC)N2CC3(COC3)C2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(N3CCN(CC3)S(C)(=O)=O)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2OC)N2C[C@H](C)N(C)[C@H](C)C2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ccc(CO)n(C)c2=O)c(F)c1
CCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NCc2ccc(OC(F)F)cc2)c2cccn(CC3CC3)c2=O)c(F)c1
CCn1cc(F)cc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2nccc(N3C[C@@H]4C[C@H]3CN4C)c2C(F)(F)F)c(F)c1
COCCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(OC)cc(n2)N2CCN(C)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccnc2OC2CCOC2)c(F)c1
FC(F)Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nc(CO)ccc2F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(cn(C)c2=O)C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nccc(NCC(C)(C)O)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ccc(CO)[nH]c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CCC(F)(F)F)c2=O)c(F)c1
CCn1cccc(N2[C@H](C)[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccc(CO)n(C)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(C)cn(C)c2=O)c(F)c1
COCC(C(=O)N(C)C)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2nc(ccc2F)N2[C@H](CO)CCC2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(C)ccc2C(F)(F)F)c(F)c1
COCC(C(=O)N(C)C)n1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O |w:3.2|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(N3CCN(C)CC3)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(ccn(C)c2=O)C#N)c(F)c1
COCC(CO)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
COC(C)Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
CCn1cccc(N2[C@H](C)[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2C[C@H]3C[C@@H]2CO3)c(F)c1
COCC(C(=O)N(C)C)n1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O |w:3.2|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CCF)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nc(ccc2OC)N2C[C@@H]3C[C@H]2CN3C)c(F)c1
COCCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
CNc1ccnc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1C(F)(F)F
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CCO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2[C@@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CCO)c2=O)c(F)c1
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)F)cc1)c1c(C)ccn(C2CCOC2)c1=O |w:32.35|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2[C@H](CO)CCC2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(F)cc(c2)C(C)(C)O)c(F)c1
COCCn1cc(F)cc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CC3CC(F)(F)C3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2C(F)(F)F)C2CCNCC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CC3CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(C)cc2)c2cccn(CCO)c2=O)c(F)c1
CNC(=O)C(C)Nc1ccnc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1C(F)(F)F
COCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
COCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(cc3)C(F)(F)F)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CCN3CCOCC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nccc(N3CCN(C)CC3)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2CCCC2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(NCC(=O)NC3CC3)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nccc(N3CCN(CC3)S(C)(=O)=O)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nc(ccc2OC)N2C[C@H](C)N(C)[C@H](C)C2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)N2C[C@@H]3C[C@H]2CN3C)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(Cl)ccn(C)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(N3CCN(C)CC3)c2C#N)c(F)c1
COCCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2nc(ccc2F)N2CCCS2(=O)=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(C)c2=O)c(F)c1
COCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(C)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CC(O)C(F)(F)F)c2=O)c(F)c1 |w:33.36|
COCC(C(=O)N(C)C)n1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O |w:3.2|
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(C)cc2)c2cccn(CC(F)F)c2=O)c(F)c1
COC(Cn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O)C(F)(F)F |w:2.45|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(C3CCOC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(NC(C)=O)cn(C)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccnn2)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CCO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2OC)N2CCN(C)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(C3COC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccnc2P(C)(C)=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CCN3CCS(=O)(=O)CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CC(C)(C)O)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2CCOCC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(C)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(ccn(C)c2=O)C(F)(F)F)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CC3CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nc(ccc2F)C(C)(C)O)c(F)c1
COC(Cn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O)C(F)(F)F |w:2.44|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)C2CCOCC2)c(F)c1
COCC(C(=O)N(C)C)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nc(ccc2C#N)N2C[C@H](C)N(C)[C@H](C)C2)c(F)c1
CCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(cc3)C#N)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(cc2)C#N)c2cccn(CC(F)F)c2=O)c(F)c1
COCCn1cc(F)cc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(NC(C)=O)cn(C)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccc(C)n(C)c2=O)c(F)c1
COCC(CO)n1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O |w:3.2|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2nc(ccc2F)N2CCC(O)C2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(NC3COC3)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2OC)N2C[C@@H]3C[C@H]2CN3C)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(cc2)C#N)c2cccn(CCO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(cn(C)c2=O)C#N)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)N2CC(CO)OCC2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2C#N)N2C[C@H](C)N(C)[C@H](C)C2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nc(ccc2C(F)F)N2CCN(C)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(N3C[C@@H]4C[C@H]3CN4C)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C3CCC3)C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c(F)c1
COCCn1c(C)ccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(ccn(C)c2=O)C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccnn2)c(F)c1
COCCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COCCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(F)cccc2C#N)c(F)c1
COCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2N(C)C)C2CCOCC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)nc2)c2ncccc2C(F)(F)F)c(F)c1
CCn1cccc(N2C[C@H]([C@H](NC(=O)c3cccc(OC)c3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cncnc2O)c(F)c1
COCCn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(C)C)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2C2CC2)N2C[C@H](C)N(C)[C@H](C)C2)c(F)c1
COc1ccc2CC(CCc2c1)C(=O)N[C@H]1[C@@H](CN(C1=O)c1ncccc1C(F)(F)F)c1c(F)cc(OC)cc1F |w:12.13|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(C3CCOC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(C3CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(C3CC3)c2=O)c(F)c1
COCCN1CCC(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)C1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)(F)F)cc1)c1cccn(CC(O)C(F)(F)F)c1=O
OC(Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O)C(F)(F)F
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ccnn(CCO)c2=O)c(F)c1
CCn1nccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
CCn1nccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CC(C)O)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CC(C)O)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(CC(C)O)c2=O)c(F)c1
COCC(C(=O)N1C[C@@H]2C[C@H]1CO2)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COC(Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2F)c1=O)C(F)(F)F
COCCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2ccc(OC)cc2)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(Cl)cc1)c1c(C)ccn(CC(F)F)c1=O
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CCO)c2=O)c(F)c1
OC(Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O)C(F)(F)F
CCn1cncc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COCCn1cncc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)F)cc1)c1cccn(CC(O)C(F)(F)F)c1=O
CCN1CCC(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)C1=O
CCn1ccc(F)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
CCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2ccc(OC)cc2F)c1=O
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CCO)c2=O)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CC(F)F)c2=O)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(CC(F)F)c2=O)c(F)c1
CCn1cncc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(CC(=O)N3CCOCC3)c2=O)c(F)c1
COC(Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2ccc(OC)cc2F)c1=O)C(F)(F)F
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(C(F)F)c2=O)c(F)c1
CCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2ccc(OC)cc2)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)(F)F)cc1)c1c(C)ccn(C(F)F)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)F)cc1)c1c(C)ccn(C(F)F)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(Cl)cc1)c1c(C)ccn(CC2CC2)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(Cl)cc1)c1c(C)ccn(CCC(F)(F)F)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)F)cc1)c1c(C)ccn(CCC(F)(F)F)c1=O
CCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
COCC(CO)n1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
CCN1CCC(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)C1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(Cl)cc1)c1cccn(CC(C)O)c1=O
Cc1ccn(CCO)c(=O)c1N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)F)cc2)C1=O)c1ccc(Cl)cc1
COC(Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2ccc(OC)cc2)c1=O)C(F)(F)F
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(CCO)c2=O)c(F)c1
COC(C)Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccnc2OCCO)c(F)c1
COCC(CO)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2ccc(OC)cc2)c1=O
COCCn1nccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(C(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CC(C)O)c2=O)c(F)c1 |w:34.36|
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(CCC(F)(F)F)c2=O)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CCC(F)(F)F)c2=O)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(CC3CC3)c2=O)c(F)c1
COCCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2ccc(OC)cc2F)c1=O
COC(C)Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
COCC(CO)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COc1cc(F)c([C@@H]2[C@@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CCO)c2=O)c(F)c1
COCCOc1ncccc1N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)(F)F)cc2)C1=O)c1c(F)cc(OC)cc1F
CC(O)Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COCCNc1ccnc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1C(F)(F)F
COCCOc1ncccc1N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)F)cc2)C1=O)c1c(F)cc(OC)cc1F
COCCOc1ncccc1N1C[C@H]([C@H](NC(=O)c2ccc(Cl)cc2)C1=O)c1c(F)cc(OC)cc1F
Cc1ccn(CC(F)F)c(=O)c1N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)F)cc2)C1=O)c1ccc(Cl)cc1
COC(Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O)C(F)(F)F
COC(Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O)C(F)(F)F
COC(C)Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(NCCO)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(N3CCOCC3)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(CC(F)F)c2=O)c(F)c1
COCCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
CC(O)Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2ccc(Cl)cc2)c1=O
Cc1ccn(CC2CC2)c(=O)c1N1C[C@H]([C@H](NC(=O)c2ccc(Cl)cc2)C1=O)c1ccc(Cl)cc1
COCC(CO)n1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COCC(C(=O)N(C)C)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(CCC(F)(F)F)c2=O)c(F)c1
CCn1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1ccnc(c1)N1[C@@H](C)[C@H]([C@H](NC(=O)c2ccc(Cl)cc2)C1=O)c1c(F)cc(OC)cc1F
COC(Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O)C(F)(F)F
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)F)cc1)c1cccn(CC(C)O)c1=O
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CC(C)O)c2=O)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CC(C)O)c2=O)c(F)c1
COCC(CO)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2F)c1=O
COCC(CO)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2F)c1=O
CC(O)Cn1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(Cl)cc2)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)(F)F)cc1)c1cccn(CC(C)O)c1=O
COCC(C(=O)N1CCOCC1)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
Cc1ccn(CC2CC2)c(=O)c1N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)F)cc2)C1=O)c1ccc(Cl)cc1
Cc1ccn(CC(F)F)c(=O)c1N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)(F)F)cc2)C1=O)c1ccc(Cl)cc1
COCC(C(=O)N1CCCC1)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CCO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc3CCCCc3n(CCO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(NCC3CCCO3)c2C(F)(F)F)c(F)c1
COCC(C(=O)N1CC[C@@H](O)C1)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COCC(CO)n1ccc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(CC3CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(NCCS(C)(=O)=O)c2C(F)(F)F)c(F)c1
COCC(CO)n1nccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2ncccc2F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(c2=O)C(F)(F)CO)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CC#N)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CC3CCOCC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CC3CCOCC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(C3CCC3)c2=O)c(F)c1
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)F)cc1)c1c(C)ccn(CC2CC2)c1=O
CCn1c2CCCCc2cc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COCCn1c2CCCCc2cc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cncn(CC(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(C3COC3)c2=O)c(F)c1
CCn1c2CCCCc2cc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CC(O)C(F)(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ccnn(CC(O)C(F)(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cncn(CC(C)O)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccnn(CCC(F)(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CCS(C)(=O)=O)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CCS(C)(=O)=O)c2=O)c(F)c1
COCCn1ncc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COCCn1ncc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ccnn(CC(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccnn(CC(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccnn(CC(O)C(F)(F)F)c2=O)c(F)c1
COCC(CO)n1nccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COCC(CO)n1nccc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(C3CCOCC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(C3CCOC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(N3CCC(C)(O)C3)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(N3CCN4CCCC4C3)c2C(F)(F)F)c(F)c1
COCC(C(=O)N1CC2(COC2)C1)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(CC(O)C(F)(F)F)c2=O)c(F)c1
COCCN1CCCC(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)C1=O
COCC(C(=O)N1CCCC1)n1cccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cncn(CC(O)C(F)(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cncn(CCC(F)(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cncn(CCO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CC(O)C(F)(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(c2=O)C(F)(F)CO)c(F)c1
COCCN1CCC(CC1)c1cc(OC)cc(n1)N1[C@@H](C)[C@H]([C@H](NC(=O)c2ccc(OC(F)F)cc2)C1=O)c1c(F)cc(OC)cc1F
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)C2CCN(CCF)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccn3cc(C)nc23)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccn3cc(CO)nc23)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccn3cc(nc23)C2CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccn3cc(nc23)C(C)C)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccn3cc(nc23)C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)C2CCN(C)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(OCC3CCCO3)ncn2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)C2=CNCCC2)c(F)c1 |t:35|
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)C2CCCN(CCO)C2)c(F)c1
COc1cc(F)c([C@@H]2[C@@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cncn(CC(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)C2CCN(CCO)CC2)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)P(C)(C)=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(C3CCNCC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(C3CCN(C)C3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(OCC3CCOC3)ncn2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(C3CCN(C)C3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccc(n2)P(C)(C)=O)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)C2CCCN(C)C2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cncn(C3CCN(C)C3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)C2CCCN(CCO)C2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cncn(C(CO)C(F)(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccn3ccnc23)c(F)c1
CCn1cnc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COCCn1cnc(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ncn(CC3(C)COC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)C2CCN(C)CC2)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)C2CCN(CCO)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)C2CCN(C)CC2)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)N2C[C@@H]3C[C@H]2CN3C)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)C2CCN(CCO)CC2)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)C2CCNCC2)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)C2CCNCC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(C3CCNC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)N2C[C@@H]3C[C@H]2CN3C)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2ncn(CC(C)C)n2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ncn(CC(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)C2CCNCC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(OCC3CCOC3)ccc2F)c(F)c1 |w:30.32|
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)C2CCN(CC(F)F)CC2)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)C2CCN(C)CC2)c(F)c1
COc1cc(F)c([C@@H]2[C@@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)C2CCOCC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(CC(F)F)cc2)c2cc(OC)cc(n2)C2CCN(CCO)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2ncn(CC(F)F)n2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cncn(C3CCOCC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cncnc2OC2CCOCC2)c(F)c1
CCn1cnc(n1)N1C[C@H]([C@H](NC(=O)c2ccc(Cl)cc2)C1=O)c1c(F)cc(OC)cc1F
COc1cc(F)c([C@@H]2[C@@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccc(n2)N2CC[C@@H](O)C2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccn(C3CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cncn(CC3CCOCC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)C2CCN(CC(F)(F)F)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)C2CCN(CC(F)F)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)C2CCN(CC(F)(F)F)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2nc(ccc2C#N)C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cc(OC)cc(n2)N2C[C@@H]3C[C@H]2CO3)c(F)c1
COc1cc(F)c([C@@H]2[C@@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccn(CC(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cncn(CC(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)C2CCN(C)CC2)c(F)c1
COc1cc(F)c([C@@H]2[C@@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(OC)cc(n2)N2CCOCC2)c(F)c1
COc1cc(F)c([C@@H]2[C@@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(OC)cc(n2)C2CCN(C)CC2)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(OCCO)n2)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccn(CC(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)N2CC[C@@H](O)C2)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cc(OC)cc(n2)C2CCN(C)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)N2CCN(C)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)N2CCN(CC2)S(C)(=O)=O)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)N2CC[C@H](O)C2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccc(F)c(n2)N2C[C@@H]3C[C@H]2CN3C)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(C)cc(n2)N2C[C@@H]3C[C@H]2CN3C)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cc(C)cc(n2)N2C[C@@H]3C[C@H]2CN3C)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ccc(F)c(n2)N2C[C@@H]3C[C@H]2CN3C)c(F)c1
COc1cc(F)c([C@@H]2[C@@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccc(CO)n2)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)N2CCOCC2)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cc(OC)cc(n2)C2CC2)c(F)c1
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)F)cc1)c1c(C)ccn(C2CCC2)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)(F)F)cc1)c1c(C)ccn(C2COC2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(Cc3cc(C)no3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)N2CCOCC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(C(CO)C(F)(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cc(OC)cc(n2)C(C)(C)O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)C(C)(C)O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(CO)n2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cc(OC)cc(CO)n2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(C)n2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)C2CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nc(ccc2F)C2CCN(CCO)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)c3CCCc3n(CCO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)c3CCCc3n(CCO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)c3CCCc3n(CCO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cnn3CCCOc23)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cnn3CCCOc23)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cnn3CCCOc23)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn3c(C)nnc23)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(c2=O)C(F)(F)C(=O)N2CCOCC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(C3CCNC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(C3CCNC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccn3c(C)nnc23)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn3c(C)nnc23)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)c3CCCCc3n(CCO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)c3CCCCc3n(CCO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)c3CCCCc3n(CCO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(CC3CCO3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CC3CCO3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CC3CCO3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CC3CNC(=O)O3)c2=O)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccnn(CC(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn([C@H]3COC[C@@H]3O)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn([C@H]3COC[C@@H]3O)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn([C@H]3COC[C@@H]3O)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(C3CCS(=O)(=O)CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(C3CCS(=O)(=O)CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(C3CCS(=O)(=O)CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2nn(C3COC3)c(=O)cc2C)c(F)c1
COc1nn(C)cc1N1C[C@H]([C@H](NC(=O)c2ccc(Cl)cc2)C1=O)c1c(F)cc(OC)cc1F
COc1nn(C)cc1N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)F)cc2)C1=O)c1c(F)cc(OC)cc1F
COc1nn(C)cc1N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)(F)F)cc2)C1=O)c1c(F)cc(OC)cc1F
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)F)cc1)c1c(C)ccn(CC(F)F)c1=O
CCn1cc(C)c(C)c(N2C[C@H](C(NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COCCn1cc(C)c(C)c(N2C[C@H](C(NC(=O)c3ccc(Cl)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
CCn1cc(C)c(C)c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)F)cc1)c1ccnn(CCC(F)(F)F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c3CCCCc3cn(CCO)c2=O)c(F)c1
CCn1ccc(n1)N1C[C@H]([C@H](NC(=O)c2ccc(Cl)cc2)C1=O)c1c(F)cc(OC)cc1F
CCn1ccc(n1)N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)F)cc2)C1=O)c1c(F)cc(OC)cc1F
CCn1ccc(n1)N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)(F)F)cc2)C1=O)c1c(F)cc(OC)cc1F
COCCn1ccnc1N1C[C@H]([C@H](NC(=O)c2ccc(Cl)cc2)C1=O)c1c(F)cc(OC)cc1F
COCCn1ccnc1N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)F)cc2)C1=O)c1c(F)cc(OC)cc1F
COCCn1ccnc1N1C[C@H]([C@H](NC(=O)c2ccc(OC(F)(F)F)cc2)C1=O)c1c(F)cc(OC)cc1F
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(C3CCOC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2ccn(CC(F)F)n2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccn(CC(F)F)n2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ccn(CC(F)F)n2)c(F)c1
CCn1cc2CCCCc2c(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
CCn1cc2CCCCc2c(N2C[C@H]([C@@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2c(F)cc(OC)cc2F)c1=O
CCn1nccc(N2C[C@H]([C@H](NC(=O)c3ccc(Cl)cc3)C2=O)c2ccc(OC)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ccc3C(=O)OCCn3c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2ccc3C(=O)OCCn3c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2cccn(CC(O)CO)c2=O)c(F)c1
CCn1nccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
CCn1nccc(N2C[C@H]([C@H](NC(=O)c3ccc(OC(F)(F)F)cc3)C2=O)c2ccc(OC)cc2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(OCC(C)(C)O)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cccn(CC(O)CO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccn(CC(O)CO)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CC(O)C3CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2c(C)ccn(CC(O)C3CC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CC(O)C3CC3)c2=O)c(F)c1
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)(F)F)cc1)c1c(C)ccn(C2CCC2)c1=O
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(C3CCC3)c2=O)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(C3CCC3)c2=O)c(F)c1
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(Cl)cc1)c1ccnn(CC(F)F)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)F)cc1)c1ccnn(CC(F)F)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)(F)F)cc1)c1ccnn(CC(F)F)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CC3CCOC3)c2=O)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2ccnn(CC(F)F)c2=O)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ccnn(CC(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(CC3CCOC3)c2=O)c(F)c1
COc1ccc([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(CC3CCOCC3)c2=O)c(F)c1
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)F)cc1)c1c(C)ccn(CC2CCOCC2)c1=O
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)(F)F)cc1)c1c(C)ccn(CC2CCOCC2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(C3CCS(=O)(=O)C3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2c(C)ccn(C3CCS(=O)(=O)C3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)(F)F)cc2)c2ccc(C(O)=O)n(CCO)c2=O)c(F)c1
COc1ccc(cc1)[C@@H]1CN(C(=O)[C@H]1NC(=O)c1ccc(OC(F)(F)F)cc1)c1c(C)ccn(C2CCOC2)c1=O
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2c(C)ccn(C(CO)C(F)(F)F)c2=O)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2nccc(OC3CCOC3)c2C(F)(F)F)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cncn(C3CCNC3)c2=O)c(F)c1
COc1cc(F)c([C@@H]2[C@H](C)N(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)C2CCN(CCF)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(cn3ccnc23)C#N)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(C)cc(n2)C2CCN(CCO)CC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(C)cc(n2)C2CCNCC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(Cl)cc2)c2cc(C)cn3ccnc23)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cccc(n2)C2CCCNC2)c(F)c1
COc1cc(F)c([C@@H]2CN(C(=O)[C@H]2NC(=O)c2ccc(OC(F)F)cc2)c2cc(OC)cc(n2)C2CCN(CC(C)(C)O)CC2)c(F)c1
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(cc2)C#N)c(nn1C)-c1ccc(F)cc1)C(C)(C)C |r|
CO[C@H]1CC[C@H](CC1)c1nn(C)c(C(=O)N(C)C(C)(C)C)c1NS(=O)(=O)c1ccc(C)cc1 |r,wU:2.1,5.8,(-10.97,-28.81,;-9.44,-28.97,;-8.53,-27.73,;-9.16,-26.32,;-8.26,-25.08,;-6.72,-25.24,;-6.1,-26.64,;-7,-27.89,;-5.82,-23.99,;-6.3,-22.53,;-5.05,-21.62,;-5.05,-20.08,;-3.8,-22.53,;-2.34,-22.05,;-1.19,-23.08,;-2.02,-20.54,;-3.16,-19.51,;-.55,-20.07,;-.23,-18.56,;.59,-21.1,;-.87,-21.57,;-4.28,-23.99,;-3.37,-25.24,;-1.84,-25.08,;-2,-23.54,;-1.68,-26.61,;-.31,-24.92,;.59,-26.16,;2.13,-26,;2.75,-24.59,;4.28,-24.43,;1.85,-23.35,;.32,-23.51,)|
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(Cl)cc2)c(nn1C)C1CCOCC1)C(C)(C)C |r|
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(C)cc2)c(nn1C)C1=CCOCC1)C(C)(C)C |r,t:24|
CO[C@H]1CC[C@H](CC1)c1nn(C)c(C(=O)N[C@@H](C)C(C)(C)C)c1NS(=O)(=O)c1ccc(Cl)cc1 |r,wU:5.8,2.1,16.17,(1.79,-50.9,;3.12,-50.13,;3.12,-48.59,;1.79,-47.82,;1.79,-46.28,;3.12,-45.51,;4.46,-46.28,;4.46,-47.82,;3.12,-43.97,;1.88,-43.06,;2.35,-41.6,;1.45,-40.35,;3.89,-41.6,;4.8,-40.35,;4.17,-38.95,;6.33,-40.51,;7.27,-39.29,;6.69,-37.87,;8.8,-39.5,;9.74,-38.28,;9.38,-40.93,;10.32,-39.71,;4.37,-43.06,;5.83,-43.54,;6.15,-45.04,;5.01,-46.08,;7.62,-45.52,;6.47,-46.55,;5.33,-47.58,;5.65,-49.09,;7.12,-49.56,;7.44,-51.07,;8.26,-48.53,;7.94,-47.03,)|
CO[C@H]1CC[C@H](CC1)c1nn(C)c(C(=O)N[C@@H](C)C(C)(C)C)c1NS(=O)(=O)c1ccc(cc1)C1CC1 |r,wU:5.8,2.1,16.17,(1.8,-30.39,;3.13,-29.62,;3.13,-28.08,;1.8,-27.31,;1.8,-25.77,;3.13,-25,;4.47,-25.77,;4.47,-27.31,;3.13,-23.46,;1.89,-22.56,;2.36,-21.09,;1.46,-19.85,;3.9,-21.09,;4.81,-19.85,;4.18,-18.44,;6.34,-20.01,;7.26,-18.78,;6.66,-17.36,;8.79,-18.96,;9.4,-20.38,;9.72,-17.73,;10.32,-19.14,;4.38,-22.56,;5.84,-23.03,;6.16,-24.54,;5.02,-25.57,;7.63,-25.02,;6.48,-26.05,;5.34,-27.08,;5.66,-28.58,;7.12,-29.06,;8.27,-28.03,;7.95,-26.52,;7.44,-30.57,;6.97,-32.03,;8.47,-31.71,)|
CO[C@H]1CC[C@H](CC1)c1nn(C)c(C(=O)N[C@@H](C)C(C)(C)C)c1NS(=O)(=O)c1ccc(cc1)C#N |r,wU:5.8,2.1,16.17,(1.8,-30.37,;3.13,-29.6,;3.13,-28.06,;1.8,-27.29,;1.8,-25.75,;3.13,-24.98,;4.47,-25.75,;4.47,-27.29,;3.13,-23.44,;1.89,-22.54,;2.36,-21.07,;1.46,-19.83,;3.9,-21.07,;4.81,-19.83,;4.18,-18.42,;6.34,-19.99,;7.26,-18.76,;6.66,-17.34,;8.79,-18.94,;9.4,-20.36,;9.72,-17.71,;10.32,-19.12,;4.38,-22.54,;5.84,-23.01,;6.16,-24.52,;5.02,-25.55,;7.63,-25,;6.48,-26.03,;5.34,-27.06,;5.66,-28.56,;7.14,-29.09,;8.27,-28.01,;7.95,-26.5,;7.46,-30.6,;7.78,-32.11,)|
COC1CCC(=CC1)c1nn(C)c(C(=O)N[C@@H](C)C(C)(C)C)c1NS(=O)(=O)c1ccc(Cl)cc1 |r,c:5|
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(Cl)cc2)c(nn1C)C1CCC2(CC1)OCCO2)C(C)(C)C |r|
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(Cl)cc2)c(nn1C)C1=CCC2(CC1)OCCO2)C(C)(C)C |r,t:24|
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(cc2)C#N)c(nn1C)C1CCOCC1)C(C)(C)C |r|
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(cc2)C2CC2)c(nn1C)-c1ccc(F)cc1)C(C)(C)C |r|
COc1ccc(cc1)S(=O)(=O)Nc1c(nn(C)c1C(=O)N[C@@H](C)C(C)(C)C)-c1ccc(F)cc1 |r|
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(cc2F)C#N)c(nn1C)-c1ccc(F)cc1)C(C)(C)C |r|
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(C)cc2)c(nn1C)C1(O)CCOCC1)C(C)(C)C |r|
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(C)cc2)c(nn1C)C1=CCC(CC1)C#N)C(C)(C)C |r,t:24|
COCc1ccccc1-c1nn(C)c(C(=O)N[C@@H](C)C(C)(C)C)c1NS(=O)(=O)c1ccc(C)cc1 |r|
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(Cl)cc2)c(nn1C)C1CCC(F)(F)CC1)C(C)(C)C |r|
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(Cl)cc2)c(nn1C)-c1ccc(F)cc1)C(C)(C)C |r|
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(Cl)cc2)c(nn1C)-c1ccccc1C(F)F)C(C)(C)C |r|
COCc1cncc(c1)-c1nn(C)c(C(=O)N[C@@H](C)C(C)(C)C)c1NS(=O)(=O)c1ccc(Cl)cc1 |r|
COC(=O)c1c(N(S(=O)(=O)c2ccc(cc2)C#N)S(=O)(=O)c2ccc(cc2)C#N)c(nn1C)-c1ccc(F)cc1F
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(cc2)C#N)c(nn1C)C1=CCC(F)(F)CC1)C(C)(C)C |r,t:25|
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(cc2)C#N)c(nn1C)C1CCC(F)(F)CC1)C(C)(C)C |r|
CCCNC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O
CSCC[C@H](NC=O)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O
CSCC[C@H](NC(=O)Nc1cccc(C)c1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O
CSCC[C@H](NC(=O)NC(C)(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O
CSCC[C@H](NC(=O)NC12CC3CC(CC(C3)C1)C2)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |TLB:12:13:17:11.10.16,THB:12:11:17:13.18.14,14:13:10:15.17.16,14:15:10:13.18.12|
CCNC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O
CSCC[C@H](NC(=O)NCc1ccccc1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O
CSCC[C@H](NC(=O)NC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O
CSCC[C@H](NC(=O)NCC(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O
CCCCNC(=O)N[C@@H](CCSC)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O
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CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(N)=O)C(=O)N[C@@H](Cc1ccccc1)C(O)=O
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CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)NC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O
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COc1cccc(Cc2cc(C)nn(CC(=O)Nc3ccc(Br)cc3)c2=O)c1
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[H][C@@]1([C@H](O)[C@H](C)C\C=C\CC)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)[C@H](NC(=O)[C@H](CC(C)(C)O)N(C)C(=O)CN(C)C(=O)[C@H](CC)NC1=O)C(C)C |r|
[H][C@]1(NC(=O)[C@]([H])([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@](O)(NC(=O)[C@H](C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)[C@@]([H])(NC(=O)[C@@H](CC(C)C)N(C)C(=O)CN(C)C1=O)[C@@H](C)CC)C(C)C)[C@@H](C)O |r|
[H][C@@]1([C@@H](C)CC)N(C)C(=O)CN(C)C(=O)[C@H](CC)NC(=O)[C@]([H])([C@H](O)[C@H](C)C\C=C\CC)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)[C@H](NC1=O)C(C)C |r|
[H][C@]1(NC(=O)[C@]([H])([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@](O)(NC(=O)[C@H](C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)CNC1=O)C(C)C)[C@@H](C)O |r|
[H][C@@]1([C@H](O)[C@H](C)C\C=C\CC)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)[C@H](NC(=O)[C@@H](CC(C)C)N(C)C(=O)CN(C)C(=O)[C@H](CCC)NC1=O)C(C)C |r|
[H][C@]1(NC(=O)[C@]([H])([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@](O)(NC(=O)[C@H](C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)[C@@H](NC(=O)[C@@H](CC(C)C)N(C)C(=O)CN(C)C1=O)C(C)C)C(C)C)[C@@H](C)O |r|
[H][C@@]1([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)[C@H](NC(=O)[C@@H](CC(C)C)N(C)C(=O)CN(C)C(=O)[C@H](CCC)NC1=O)C(C)C |r|
[H][C@]1(NC(=O)[C@]([H])([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)CN(C)C1=O)[C@@H](C)O |r|
[H][C@]1(NC(=O)[C@]([H])([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)[C@@]([H])(NC(=O)[C@@H](CC(C)C)N(C)C(=O)CN(C)C1=O)[C@@H](C)CC)[C@@H](C)O |r|
[H][C@@]1([C@H](O)[C@H](C)C\C=C\CC)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)[C@H](NC(=O)[C@H](Cc2ccccc2)N(C)C(=O)CN(C)C(=O)[C@H](CC)NC1=O)C(C)C |r|
[H][C@]1(NC(=O)[C@]([H])([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)CN(C)C1=O)[C@@H](C)O |r|
[H][C@@]1([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC(C)C)N(C)C(=O)CN(C)C(=O)[C@H](CCC)NC1=O |r|
O=C(N1CCCCC1)c1cnn2CC(Nc12)c1ccccc1 |w:13.18|
CCOC(=O)c1cnn2CC(Nc12)c1ccccc1 |w:10.14|
OC(=O)c1cnn2CC(Nc12)c1ccccc1 |w:8.12|
CC(C)(C)NC(=O)c1cnn2CC(Nc12)c1ccccc1 |w:12.16|
O=C(N1CCCC1)c1cnn2CC(Nc12)c1ccccc1 |w:12.17|
O=C(NC1CC1)c1cnn2CC(Nc12)c1ccccc1 |w:11.16|
O=C(N1CCN(Cc2ccccc2)CC1)c1cnn2CC(Nc12)c1ccccc1 |w:20.26|
O=C(N1CCCCCC1)c1cnn2CC(Nc12)c1ccccc1 |w:14.19|
O=C(NCc1ccccc1)c1cnn2CC(Nc12)c1ccccc1 |w:15.20|
NC(=O)c1cnn2CC(Nc12)c1ccccc1 |w:8.12|
C1C(Nc2ccnn12)c1ccccc1 |w:1.9|
O=C(N1CCOCC1)c1cnn2CC(Nc12)c1ccccc1 |w:13.18|
CSCCC(NC(=O)c1ccccc1O)c1nc2ccccc2[nH]1
Oc1ccccc1C(=O)NC(C(=O)NC1CCCCC1)c1ccc(Cl)cc1
Oc1ccccc1C(=O)NC(C(=O)Nc1ccccc1)c1ccc(Cl)cc1
CSCCC(NC(=O)c1ccccc1)c1nc2ccccc2[nH]1
Cc1cccc(C)c1NC(=O)C(NC(=O)c1ccccc1O)C1CCCCC1
Cc1cccc(C)c1NC(=O)C(NC(=O)c1ccccc1O)c1cn(C)cn1
CSCC[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
Cc1cccc(C)c1NC(=O)C(NC(=O)c1ccccc1O)c1ccccc1
CCOc1ccc2oc(C(=O)NC(CCSC)c3nc4ccccc4[nH]3)c(C)c2c1
Cc1ccc(s1)C(NC(=O)c1ccccc1O)C(=O)Nc1c(C)cccc1C
CCC(CC)NC(=O)c1cnn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1Cl
CCC(CC)NC(=O)c1cn(nc1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1
C[C@H](NC(=O)c1c(NS(=O)(=O)c2ccc(C)cc2)n(nc1C(F)(F)F)-c1ccccc1)C(C)(C)C |r|
CCC(CC)NC(=O)c1ncn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1
C[C@@H](NC(=O)c1c(C)nn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1)C(C)(C)C |r|
CCC(CC)NC(=O)c1nnn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1
C[C@H](NC(=O)c1c(C)nn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1)C(C)(C)C |r|
Cc1ccc(cc1)S(=O)(=O)Nc1c(cnn1-c1ccccc1)C(=O)NCc1ccccc1
CCC(CC)NC(=O)c1cnn(c1NS(=O)(=O)C1CCCC1)-c1ccccc1
CN(C1CCCCC1)C(=O)c1cnn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1
CCC(CC)NC(=O)c1cnn(c1NS(=O)(=O)c1ccccc1)-c1ccccc1
Cc1ccc(cc1)S(=O)(=O)Nc1c(cnn1-c1ccccc1)C(=O)NC1CCCCC1
CCC(C)NC(=O)c1c(C)nn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1
CCC(CC)NC(=O)c1cnn(c1NS(=O)(=O)c1ccccc1C)-c1ccccc1
Cc1nn(c(NS(=O)(=O)c2ccc(C)cc2)c1C(=O)NCC(C)(C)C)-c1ccccc1
Cc1ccc(cc1)S(=O)(=O)Nc1c(cnn1-c1ccccc1)C(=O)NC1CCOCC1
CCC(CC)NC(=O)c1cnn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1
Cc1nn(c(NS(=O)(=O)c2ccc(C)cc2)c1C(=O)NC1CCOCC1)-c1ccccc1
CC1CCCCC1NC(=O)c1c(C)nn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1
CCCC(CC)NC(=O)c1cnn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1
CC1CCCCC1NC(=O)c1cnn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1
CN(C1CCCCC1)C(=O)c1c(C)nn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1
Cc1nn(c(NS(=O)(=O)c2ccc(C)cc2)c1C(=O)NC1CCCCC1)-c1ccccc1
CC(C)NC(=O)c1c(C)nn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1
CCC(CC)NC(=O)c1c(C)nn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccc1
CCN(C1CCCCC1)C(=O)c1cnn(c1NS(=O)(=O)c1ccc(cc1)-c1cnco1)-c1ccccc1
CCC(CC)NC(=O)c1cnn(c1NS(=O)(=O)c1ccc(cc1)-c1cnco1)-c1ccccc1
CCC(CC)NC(=O)c1cnn(C(C)C)c1NS(=O)(=O)c1ccc(C)cc1
CCC(CC)NC(=O)c1cnn(Cc2ccccc2)c1NS(=O)(=O)c1ccc(C)cc1
C[C@H](NC(=O)c1c(C)nn(c1NS(=O)(=O)c1ccc(cc1)C(F)(F)F)-c1ccc(F)cc1)C(C)(C)C |r|
CCC(CC)NC(=O)c1cnn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccccn1
C[C@H](NC(=O)c1c(C)nn(c1NS(=O)(=O)c1ccc(cc1)C#N)-c1ccc(F)cc1)C(C)(C)C |r|
CCC(CC)NC(=O)c1cnn(c1NS(=O)(=O)c1ccc(C)cc1)-c1ccc(cc1)C#N
C[C@H](NC(=O)c1c(C)nn(c1NS(=O)(=O)c1cccnc1)-c1ccc(F)cc1)C(C)(C)C |r|
C[C@H](NC(=O)c1c(C)nn(c1NS(=O)(=O)C1CCCCC1)-c1ccccc1)C(C)(C)C |r|
Cc1ccc(cc1)S(=O)(=O)Nc1c(cnn1-c1ccccc1)C(=O)NCc1ccc(C)cc1C
CCC(CC)n1nc(C)c(C(=O)N[C@@H](C)C(C)(C)C)c1NS(=O)(=O)c1ccc(C)cc1 |r|
C[C@H](NC(=O)c1c(C)nn(c1NS(=O)(=O)c1ccc(C)cc1)C(C)(C)C)C(C)(C)C |r|
C[C@H](NC(=O)c1c(C)nn(CC(F)(F)F)c1NS(=O)(=O)c1ccc(C)cc1)C(C)(C)C |r|
CCn1nc(C)c(C(=O)N[C@@H](C)C(C)(C)C)c1NS(=O)(=O)c1ccc(C)cc1 |r|
C[C@H](NC(=O)c1c(C)nn(C2CCN(CC(F)(F)F)CC2)c1NS(=O)(=O)c1ccc(C)cc1)C(C)(C)C |r|
CC(C)n1nc(C)c(C(=O)N[C@@H](C)C(C)(C)C)c1NS(=O)(=O)c1ccc(C)cc1 |r|
CCC(CC)NC(=O)c1c(C)nn(C(C)C)c1NS(=O)(=O)c1ccc(C)cc1
C[C@H](NC(=O)c1c(C)nn(C2CCS(=O)(=O)CC2)c1NS(=O)(=O)c1ccc(C)cc1)C(C)(C)C |r|
C[C@H](NC(=O)c1c(C)nn(C2CCSCC2)c1NS(=O)(=O)c1ccc(C)cc1)C(C)(C)C |r|
COCCC(C)n1nc(C)c(C(=O)N[C@@H](C)C(C)(C)C)c1NS(=O)(=O)c1ccc(C)cc1 |r|
COCC(C)n1nc(C)c(C(=O)N[C@@H](C)C(C)(C)C)c1NS(=O)(=O)c1ccc(C)cc1 |r|
C[C@H](NC(=O)c1c(C)nn(C2CCCCC2)c1NS(=O)(=O)c1ccc(C)cc1)C(C)(C)C |r|
C[C@H](NC(=O)c1c(C)nn(C2CCOCC2)c1NS(=O)(=O)c1ccc(cc1)C1CC1)C(C)(C)C |r|
C[C@H](NC(=O)c1c(C)nn(C2CCCC2)c1NS(=O)(=O)c1ccc(C)cc1)C(C)(C)C |r|
C[C@H](NC(=O)c1c(C)nn(C2CCC2)c1NS(=O)(=O)c1ccc(C)cc1)C(C)(C)C |r|
CO[C@H]1CC[C@H](CC1)n1nc(C)c(C(=O)N[C@@H](C)C(C)(C)C)c1NS(=O)(=O)c1ccc(C)cc1 |r,wU:5.8,16.17,2.1,(31.27,-8.16,;32.01,-6.81,;31.21,-5.49,;29.67,-5.52,;28.87,-4.21,;29.61,-2.86,;31.15,-2.82,;31.95,-4.13,;29.13,-1.41,;27.66,-.94,;27.66,.6,;26.41,1.51,;29.12,1.08,;29.59,2.55,;31.1,2.88,;28.56,3.69,;29.03,5.16,;27.99,6.3,;30.53,5.48,;31.57,4.34,;31,6.95,;32.01,5.9,;30.03,-.15,;31.57,-.15,;32.33,1.2,;30.99,1.97,;32.33,2.74,;33.88,1.2,;34.64,-.13,;36.18,-.13,;36.95,1.2,;38.49,1.2,;36.18,2.53,;34.64,2.52,)|
C[C@H](NC(=O)c1c(C)nn(C2CCOC2)c1NS(=O)(=O)c1ccc(C)cc1)C(C)(C)C |r|
C[C@H](NC(=O)c1c(C)nn(C2CCOCC2)c1NS(=O)(=O)c1ccc(C)cc1)C(C)(C)C |r|
OB(O)c1ccccc1CSc1ccc(cn1)C(=O)Nc1ccc(F)cc1
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](CC1=CCCCC1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccc(cc1)C(=O)c1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](CC1CCCCC1)C(O)=O |r,t:10|
CC(C)C[C@@H](NC(=O)[C@H](CC1=CCCCC1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccc(cc1)C(=O)c1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r,t:10|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccc(cc1)C(=O)c1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1cn(C(=O)OC(C)(C)C)c2ccccc12)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccc(OC(C)(C)C)cc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](CC1CCCCC1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)OC(C)(C)C)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](COC(C)(C)C)C(O)=O |r|
CC(C)C[C@H](NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](C(C)C)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccc(cc1)C(=O)c1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](CCCCNC(=O)OC(C)(C)C)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](CC(=O)OC(C)(C)C)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H]([C@@H](C)OC(C)(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CSCC[C@H](NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](CC1CCCCC1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](C(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](CCCCNC(=O)c1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](CCCCNC(=O)C1CCCCC1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](CCCCN)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccc(cc1)C(=O)c1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1cn(C(=O)OC(C)(C)C)c2ccccc12)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1cn(C=O)c2ccccc12)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccc(OC(C)(C)C)cc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccc(Cl)cc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](CC1CCCCC1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](COC(C)(C)C)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@@H](NC(=O)OC(C)(C)C)[C@@H](C)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](C)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](C)NC(=O)[C@@H](CC(C)C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
CC(C)C[C@@H](NC(=O)[C@H](C)NC(=O)OC(C)(C)C)C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@H](CC(C)C)C(=O)N[C@@H](Cc1ccccc1)C(O)=O |r|
COc1ccc(NC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)NCC2(CCCCC2)c2ccccn2)cc1 |r|
COc1ccc(NC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)NCC2(CCCCC2)c2ccc(OC)cn2)cc1 |r|
O=C(N[C@@H](Cc1c[nH]c2ccccc12)C(=O)NCC1(CC1)c1ccccc1)Nc1ccccc1 |r|
COc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)NCC2(CC2)c2ccc(C)c(F)c2)cc1 |r|
[O-][N+](=O)c1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)NCC2(CC2)c2ccccc2)cc1 |r|
COc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)NCC2(CC2)c2ccc(F)c(Cl)c2)cc1 |r|
[O-][N+](=O)c1ccc(NC(=O)N[C@@H](Cc2cccnc2)C(=O)NCC2(CC2)c2ccccc2)cc1 |r|
COc1ccc(NC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)NCC2(CC2)c2ccccc2)cc1 |r|
Fc1ccc(NC(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)NCC2(CC2)c2ccccc2)cc1 |r|
[O-][N+](=O)c1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)NCC2(CC2)c2ccccc2)cc1 |r|
[O-][N+](=O)c1ccc(NC(=O)N[C@H](Cc2cccnc2)C(=O)NCC2(CC2)c2ccccc2)cc1 |r|
COc1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)NCC2(CC2)c2ccc(F)c(Cl)c2)cc1 |r|
Fc1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)NCC2(CC2)c2ccc(F)c(Cl)c2)cc1 |r|
Fc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)NCC2(CC2)c2ccc(F)c(Cl)c2)cc1 |r|
Cc1ccc(cc1F)C1(CNC(=O)[C@H](Cc2ccc(cc2)C#N)NC(=O)Nc2ccc(F)cc2)CC1 |r|
CC[C@@H]1NC(=O)[C@H](C(C)C(C)C\C=C\C)N(C)C(=O)[C@@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](NC(=O)[C@H](CC(C)C)N(C)C(=O)CN(C)C1=O)C(C)C |r|
CC[C@@H]1NC(=O)[C@H]([C@H](O)[C@H](C)C\C=C\C)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)[C@H](C)NC(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](NC(=O)[C@H](CC(C)C)N(C)C(=O)CN(C)C1=O)C(C)C |r|
[H][C@]12N(CCC[C@@]1(CC)C=C(C(=O)OC)n1c2c(CCNC(=O)c2ccc(Br)cc2)c2ccccc12)C#N |r,t:10|
COc1ccc(NC(=O)Cn2nc(C)cc(Cc3ccccc3OC)c2=O)cc1
COc1cccc(Cc2cc(C)nn(CC(=O)Nc3c(F)cc(Cl)cc3F)c2=O)c1
CCCCC(C(=O)Nc1ccc(Cl)cc1)n1nc(cc(Cc2ccccc2OC)c1=O)C(F)(F)F
COc1ccc(Cc2cc(C)nn(C(C)C(=O)Nc3ccc(Br)cc3)c2=O)cc1
CCCCC(C(=O)Nc1ccc(Cl)cc1)n1nc(C)cc(Cc2cccc(OC)c2)c1=O
COc1ccccc1Cc1cc(C)nn(CC(=O)Nc2ccc(Cl)cc2F)c1=O
CCCCC(C(=O)Nc1ccc(Cl)cc1)n1nc(C)cc(Cc2ccccc2OC)c1=O
COc1cccc(Cc2cc(C)nn(CC(=O)Nc3ccc(Cl)cc3F)c2=O)c1
Cc1cc(Cc2ccc(F)cc2)c(=O)n(CC(=O)Nc2ccc(Br)cc2[N+]([O-])=O)n1
Cc1cc(Cc2ccc(F)cc2)c(=O)n(CC(=O)Nc2c(F)cc(F)cc2[N+]([O-])=O)n1
COc1cccc(Cc2cc(C)nn(CC(=O)Nc3ccc(Cl)cc3)c2=O)c1OC
COc1cccc(Cc2cc(C)nn(C(C)C(=O)Nc3ccc(Cl)cc3)c2=O)c1OC
CCC(C(=O)Nc1ccc(Cl)cc1)n1nc(C)cc(Cc2ccccc2OC)c1=O
COc1ccccc1Cc1cc(C)nn(C(C(C)C)C(=O)Nc2ccc(Cl)cc2)c1=O
CCCCC(C(=O)Nc1ccc(Br)cc1)n1nc(C)cc(Cc2ccccc2OC)c1=O
CCCCC(C(=O)Nc1ccc(Br)cc1)n1nc(C)cc(Cc2cccc(OC)c2)c1=O
CCCCC(C(=O)Nc1ccc(Br)cc1)n1nc(C)cc(Cc2cccc(OC)c2OC)c1=O
COc1ccccc1Cc1cc(C)nn(CC(=O)Nc2cccc(Cl)c2)c1=O
COc1ccccc1Cc1cc(C)nn(CC(=O)Nc2ccc(Cl)cc2)c1=O
COc1ccccc1Cc1cc(C)nn(CC(=O)Nc2ccccc2C#N)c1=O
COc1ccccc1Cc1cc(C)nn(CC(=O)Nc2ccc(cc2)C#N)c1=O
COc1ccccc1Cc1cc(C)nn(CC(=O)Nc2ccc(Cl)cc2Cl)c1=O
COc1ccccc1Cc1cc(C)nn(CC(=O)Nc2c(F)cc(Cl)cc2F)c1=O
CC(C(=O)Nc1ccc(Br)cc1)n1nc(C)cc(Cc2ccccc2F)c1=O
COc1cccc(Cc2cc(C)nn(C(C)C(=O)Nc3ccccc3Cl)c2=O)c1
COc1cccc(Cc2cc(C)nn(C(C)C(=O)Nc3ccccc3F)c2=O)c1
COc1cccc(Cc2cc(C)nn(C(C)C(=O)Nc3cccc(F)c3)c2=O)c1
CC(C(=O)Nc1ccc(Br)cc1)n1nc(C)cc(Cc2cccc(F)c2)c1=O
CC(C(=O)Nc1ccc(Br)cc1)n1nc(C)cc(Cc2ccc(F)cc2)c1=O
COc1ccc(OC)c(Cc2cc(C)nn(CC(=O)Nc3ccc(Cl)cc3)c2=O)c1
COc1ccccc1Cc1cc(C)nn(CC(=O)Nc2ccccc2Cl)c1=O
COc1ccccc1Cc1cc(C)nn(CC(=O)Nc2cccc(c2)C#N)c1=O
COc1ccccc1Cc1cc(nn(CC(=O)Nc2ccc(Cl)cc2)c1=O)C(F)(F)F
COc1ccccc1Cc1cc(C)nn(C(C)C(=O)Nc2ccc(Br)cc2)c1=O
COc1cccc(OC)c1Cc1cc(C)nn(CC(=O)Nc2ccc(Cl)cc2)c1=O
COc1ccccc1Cc1cc(C)nn(C(C2CC2)C(=O)Nc2ccc(Cl)cc2)c1=O
CC(C)C1=C(C(=O)N(N1C)c2ccccc2)NC(=O)Nc3ccc(cc3)Cl
COc1ccccc1Cc1cc(C)nn(CC(=O)Nc2ccc(OC(F)(F)F)cc2)c1=O
COc1cccc(Cc2cc(C)nn(C(C)C(=O)Nc3cccc(Cl)c3)c2=O)c1
CCCCC(C(=O)Nc1ccc(Cl)cc1)n1nc(C)cc(Cc2cccc(OC)c2OC)c1=O
CCc1ccc(NC(=O)Cn2nc(C)cc(Cc3ccccc3OC)c2=O)cc1
COc1cccc(Cc2cc(C)nn(C(C)C(=O)Nc3ccc(Cl)cc3)c2=O)c1
CCCC(C(=O)Nc1ccc(Cl)cc1)n1nc(C)cc(Cc2ccccc2OC)c1=O
COc1cccc(Cc2cc(C)nn(C(C)C(=O)Nc3ccc(F)cc3)c2=O)c1
COc1ccccc1Cc1cc(C)nn(C(C)C(=O)Nc2ccc(Cl)cc2)c1=O
COc1ccc(CC(NC(=O)Nc2ccc(Cl)cc2)C(N)=O)cc1
COc1ccc(cc1)[C@@H]1NC(=O)[C@@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
COc1ccc(cc1)[C@@H]1NC(=O)[C@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
COc1ccc(cc1)[C@@H]1CNC(=O)[C@@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
COc1ccc(cc1)[C@@H]1CNC(=O)[C@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
COc1ccc(cc1)[C@@H]1CCNC(=O)[C@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
COc1ccc(cc1)C1CNC(=O)C1NC(=O)Nc1ccc(Cl)cc1
COc1ccc(cc1)[C@H]1CNC(=O)[C@@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
COc1ccc(cc1)[C@@H]1CNC(=O)[C@H]1NC(=O)Nc1ccc(F)cc1 |r|
COc1ccc([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(F)cc2)c(F)c1 |r|
COc1ccc(cc1F)[C@@H]1CNC(=O)[C@H]1NC(=O)Nc1ccc(F)cc1 |r|
COc1ccc([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(F)cc2)c(Cl)c1 |r|
COc1ccc([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(F)cc2)c(C)c1 |r|
Fc1ccc(NC(=O)N[C@H]2[C@@H](CNC2=O)c2ccc(Cl)cc2F)cc1 |r|
COc1cc(F)c(cc1F)[C@@H]1CNC(=O)[C@H]1NC(=O)Nc1ccc(F)cc1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(F)cc2)c(F)c1 |r|
COc1cnc([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(F)cc2)c(F)c1 |r|
CCc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(F)cc2)c(F)c1 |r|
Fc1ccc(NC(=O)N[C@H]2[C@@H](CNC2=O)c2c(F)cc(cc2F)C#N)cc1 |r|
CNc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(F)cc2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2cccc(F)c2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccccc2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(Br)cc2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(cc2)C#N)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(C)cc2)c(F)c1 |r|
COc1ccc(NC(=O)N[C@H]2[C@@H](CNC2=O)c2c(F)cc(OC)cc2F)cc1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(F)c(F)c2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(F)c(O)c2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(Cl)c(O)c2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(C)c(O)c2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(Cl)cn2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2ccc(Cl)s2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2cc(C)ns2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)Nc2cc3ccccc3s2)c(F)c1 |r|
Brc1ccc(NC(=O)NC2CCN(C2=O)c2ccccc2)cc1
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2Nc2nc3ccccc3[nH]2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2c2nc3ccccc3[nH]2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2Nc2nnc(o2)-c2ccccc2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2Nc2nnc(o2)-c2ccc(Cl)cc2)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2Nc2cc(on2)-c2ccc(Cl)cc2)c(F)c1 |r|
Fc1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)NC2CCCCNC2=O)cc1 |r|
Fc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)NC2CCCCNC2=O)cc1 |r|
Fc1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)N2CCCCC2)cc1 |r|
Fc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)N2CCCCC2)cc1 |r|
Fc1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)N2CCCC2)cc1 |r|
Fc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)N2CCCC2)cc1 |r|
Fc1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)N2Cc3ccccc3C2)cc1 |r|
Fc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)N2Cc3ccccc3C2)cc1 |r|
Fc1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)N2CCc3ccccc23)cc1 |r|
Fc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)N2CCc3ccccc23)cc1 |r|
Fc1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)N2CCc3ccccc3C2)cc1 |r|
Fc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)N2CCc3ccccc3C2)cc1 |r|
Fc1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)N2CCCc3ccccc23)cc1 |r|
Fc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)N2CCCc3ccccc23)cc1 |r|
Fc1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)N2Cc3ccc(F)cc3C2)cc1 |r|
Fc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)N2Cc3ccc(F)cc3C2)cc1 |r|
CC1(C)CN(C(=O)[C@@H](Cc2ccc(cc2)C#N)NC(=O)Nc2ccc(F)cc2)c2ccccc12 |r|
CC1(C)CN(C(=O)[C@H](Cc2ccc(cc2)C#N)NC(=O)Nc2ccc(F)cc2)c2ccccc12 |r|
Fc1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)N2CCc3cc(F)ccc23)cc1 |r|
Fc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)N2CCc3cc(F)ccc23)cc1 |r|
Fc1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)N2CCc3ccc(F)cc23)cc1 |r|
Fc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)N2CCc3ccc(F)cc23)cc1 |r|
Fc1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)N2CCc3cccnc23)cc1 |r|
Fc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)N2CCc3cccnc23)cc1 |r|
Fc1ccc(NC(=O)N[C@H](Cc2ccc(cc2)C#N)C(=O)N2CCc3ccc(F)cc3C2)cc1 |r|
Fc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)N2CCc3ccc(F)cc3C2)cc1 |r|
CC1(C)CN(Cc2cc(F)ccc12)C(=O)[C@H](Cc1ccc(cc1)C#N)NC(=O)Nc1ccc(F)cc1 |r|
CC(C)C(C(C)NC(=O)Nc1ccc(Br)cc1)C(O)=O
CC(C)C[C@H](NC(=O)CNC(=O)Nc1ccc(Br)cc1)C(O)=O |r|
CC(C)C[C@H](NC(=O)CCNC(=O)Nc1ccc(Br)cc1)C(O)=O |r|
OC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)Nc1ccc(Br)cc1 |r|
CCC[C@H](NC(=O)CNC(=O)Nc1ccc(Br)cc1)C(O)=O |r|
COc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)NCC2(CC2)c2ccc(O)cc2)cc1 |r|
COc1ccc(NC(=O)N[C@@H](Cc2ccc(cc2)C#N)C(=O)NCC2(CC2)c2cccc(O)c2)cc1 |r|
COc1ccc(NC(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)NCC2(CC2)c2ccccc2)cc1 |r|
COc1ccc(NC(=O)N[C@H](Cc2ccc(O)cc2)C(=O)NCC2(CC2)c2ccccc2)cc1 |r|
COc1cccc(c1)-c1cc(C#N)c(C)n(CC(=O)Nc2ccc(Br)cc2)c1=O
Brc1ccc(NC(=O)Cn2c(=O)[nH]cc(-c3ccccc3)c2=O)cc1
COc1cccc(Cc2c(C)c(C)nn(CC(=O)Nc3ccc(Br)cc3)c2=O)c1
COc1ccc(Cc2c(C)c(C)nn(CC(=O)Nc3ccc(Br)cc3)c2=O)cc1
COc1ccc2cc(ccc2c1)C1(CC1)NC(=O)N[C@H]1[C@@H](CNC1=O)c1c(F)cc(OC)cc1F |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2NC(=O)NC2(CC2)c2cccc(c2)C(F)(F)F)c(F)c1 |r|
CP(C)(=O)c1ccccc1-c1ccc(N2CC[C@@H](NC(=O)Nc3ccc(Cl)cc3)C2=O)c(F)c1F |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2Nc2cc(on2)-c2ccc(cc2)C(F)F)c(F)c1 |r|
COc1cc(F)c([C@@H]2CNC(=O)[C@H]2Nc2nnc(o2)-c2ccc(Oc3ccc(nc3)C(F)(F)F)cc2)c(F)c1 |r|
Cn1c(c(NC(=O)Nc2ccc(Cl)cc2)c(=O)n1-c1ccccc1)C(C)(C)C
COc1ccc(cc1)[C@H]1CCNC(=O)[C@@H]1NC(=O)Nc1ccc(Cl)cc1 |r|
COc1cc(F)c([C@H]2CCN(CC3CC3)C(=O)[C@@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1 |r|
COc1cc(F)c([C@H]2CCN(CCC(F)F)C[C@@H]2NC(=O)Nc2ccc(Cl)cc2)c(F)c1 |r|
COc1ccc(cc1)[C@H]1CCN(C[C@@H]1NC(=O)Nc1ccc(Cl)cc1)c1ccnnc1 |r|
COc1ccc(cc1)[C@@H]1CCN(Cc2ccccn2)C(=O)[C@@H]1NC(=O)Nc1ccc(F)cc1 |r|
COc1ccc(cc1)[C@H]1CCN(Cc2ccccn2)C(=O)[C@@H]1NC(=O)Nc1ccc(F)cc1 |r|
COc1ccc(cc1)[C@H]1CCN(Cc2cccnc2)C(=O)[C@@H]1NC(=O)Nc1ccc(F)cc1 |r|
CCCCCCc1cc2c(cc1OC(C)=O)oc(C)c(-c1ccccc1OC)c2=O |(-8.65,,;-7.36,-.77,;-6.03,,;-4.69,-.77,;-3.36,,;-2.03,-.77,;-.69,,;.64,-.77,;1.98,,;1.98,1.54,;.64,2.31,;-.69,1.54,;-2.03,2.31,;-2.03,3.85,;-3.36,4.62,;-.69,4.62,;3.31,2.31,;4.64,1.54,;5.98,2.31,;4.64,,;5.98,-.77,;7.31,,;8.65,-.77,;8.65,-2.31,;7.31,-3.08,;5.98,-2.31,;4.64,-3.08,;4.64,-4.62,;3.31,-.77,;3.31,-2.31,)|
CCCCCCc1cc2c(cc1OC(C)=O)oc(C)c(-c1cccc(OC)c1)c2=O
CCCCCCc1cc2c(cc1OC(C)=O)oc(C)c(-c1ccc(OC)cc1)c2=O
CCCCCCc1cc2c(cc1OC(C)=O)oc(c(-c1ccccc1OC)c2=O)C(F)(F)F |(-8.65,0,;-7.36,-.77,;-6.03,0,;-4.7,-.77,;-3.36,0,;-2.03,-.77,;-.69,0,;.64,-.77,;1.98,0,;1.98,1.54,;.64,2.31,;-.69,1.54,;-2.03,2.31,;-2.03,3.85,;-3.36,4.62,;-.69,4.62,;3.31,2.31,;4.64,1.54,;4.64,0,;5.98,-.77,;7.31,0,;8.65,-.77,;8.65,-2.31,;7.31,-3.08,;5.98,-2.31,;4.64,-3.08,;4.64,-4.62,;3.31,-.77,;3.31,-2.31,;5.98,2.31,;5.98,3.85,;7.31,1.54,;7.31,3.08,)|
CCCCCCc1cc2c(cc1OC(C)=O)oc(c(-c1cccc(OC)c1)c2=O)C(F)(F)F
CCCCCCc1cc2c(cc1OC(C)=O)oc(c(-c1ccc(OC)cc1)c2=O)C(F)(F)F
CCCc1cc2c(cc1OC(C)=O)oc(C)c(-c1ccccc1OC)c2=O |(-6.67,-.77,;-5.34,0,;-4,-.77,;-2.67,0,;-1.33,-.77,;,0,;,1.54,;-1.33,2.31,;-2.67,1.54,;-4,2.31,;-4,3.85,;-5.34,4.62,;-2.67,4.62,;1.33,2.31,;2.67,1.54,;4,2.31,;2.67,0,;4,-.77,;5.34,0,;6.67,-.77,;6.67,-2.31,;5.34,-3.08,;4,-2.31,;2.67,-3.08,;2.67,-4.62,;1.33,-.77,;1.33,-2.31,)|
CCCc1cc2c(cc1OC(C)=O)oc(C)c(-c1cccc(OC)c1)c2=O
CCCc1cc2c(cc1OC(C)=O)oc(C)c(-c1ccc(OC)cc1)c2=O
CCc1cc2c(cc1OC(C)=O)oc(C)c(-c1ccccc1OC)c2=O |(-6,0,;-4.67,-.77,;-3.33,0,;-2,-.77,;-.67,0,;-.67,1.54,;-2,2.31,;-3.33,1.54,;-4.67,2.31,;-4.67,3.85,;-6,4.62,;-3.33,4.62,;.67,2.31,;2,1.54,;3.33,2.31,;2,0,;3.33,-.77,;4.67,0,;6,-.77,;6,-2.31,;4.67,-3.08,;3.33,-2.31,;2,-3.08,;2,-4.62,;.67,-.77,;.67,-2.31,)|
CCCCc1cc2c(cc1OC(C)=O)oc(C)c(-c1ccccc1OC)c2=O |(-7.34,0,;-6,-.77,;-4.67,0,;-3.34,-.77,;-2,0,;-.67,-.77,;.67,0,;.67,1.54,;-.67,2.31,;-2,1.54,;-3.34,2.31,;-3.34,3.85,;-4.67,4.62,;-2,4.62,;2,2.31,;3.33,1.54,;4.67,2.31,;3.33,0,;4.67,-.77,;6,0,;7.34,-.77,;7.34,-2.31,;6,-3.08,;4.67,-2.31,;3.33,-3.08,;3.33,-4.62,;2,-.77,;2,-2.31,)|
CCCCCc1cc2c(cc1OC(C)=O)oc(C)c(-c1ccccc1OC)c2=O |(-8,-.77,;-6.67,0,;-5.34,-.77,;-4,0,;-2.67,-.77,;-1.33,0,;-0,-.77,;1.33,0,;1.33,1.54,;-0,2.31,;-1.33,1.54,;-2.67,2.31,;-2.67,3.85,;-4,4.62,;-1.33,4.62,;2.67,2.31,;4,1.54,;5.34,2.31,;4,0,;5.34,-.77,;6.67,0,;8,-.77,;8,-2.31,;6.67,-3.08,;5.34,-2.31,;4,-3.08,;4,-4.62,;2.67,-.77,;2.67,-2.31,)|
CCCCCCC(=O)Oc1cc2oc(C)c(-c3cccc(OC)c3)c(=O)c2cc1C
CCCc1cc2c(cc1OC(=O)N(C)C)oc(C)c(-c1ccccc1OC)c2=O |(-4.67,-2.69,;-3.34,-1.93,;-3.34,-.39,;-2,.38,;-.67,-.39,;.67,.38,;.67,1.92,;-.67,2.69,;-2,1.92,;-3.34,2.69,;-4.67,1.92,;-4.67,.38,;-6,2.69,;-7.34,1.92,;-6,4.23,;2,2.69,;3.33,1.92,;4.67,2.69,;3.33,.38,;4.67,-.39,;6,.38,;7.34,-.39,;7.34,-1.92,;6,-2.69,;4.67,-1.92,;3.33,-2.69,;3.33,-4.23,;2,-.39,;2,-1.92,)|
CCCCCCc1cc2c(cc1OC(C)=O)oc(C)c(-c1nc3ccccc3n1C)c2=O |(-7.76,-4.62,;-7.76,-3.08,;-6.43,-2.31,;-6.43,-.77,;-5.09,-0,;-5.09,1.54,;-3.76,2.31,;-2.42,1.55,;-1.1,2.31,;-1.1,3.85,;-2.43,4.62,;-3.76,3.85,;-5.09,4.62,;-6.43,3.85,;-7.76,4.62,;-6.43,2.31,;.24,4.62,;1.57,3.85,;2.9,4.62,;1.57,2.31,;2.9,1.54,;4.24,2.31,;5.39,1.25,;6.88,1.4,;7.76,.18,;7.15,-1.19,;5.66,-1.35,;4.77,-.12,;3.24,.05,;2.15,-1.04,;.24,1.54,;.24,0,)|
Cc1oc2cc(OC(=O)c3ccco3)ccc2c(=O)c1-c1nc2ccccc2n1C |(1.59,-3.99,;.82,-2.66,;-.72,-2.66,;-1.49,-1.32,;-3.03,-1.32,;-3.8,.01,;-5.34,.01,;-6.11,1.34,;-5.34,2.68,;-7.65,1.34,;-8.56,.1,;-10.02,.57,;-10.02,2.11,;-8.56,2.59,;-3.03,1.34,;-1.49,1.34,;-.72,.01,;.82,.01,;1.59,1.34,;1.59,-1.32,;3.13,-1.32,;4.03,-.08,;5.5,-.55,;6.83,.22,;8.16,-.55,;8.16,-2.09,;6.83,-2.86,;5.5,-2.09,;4.03,-2.57,;3.56,-4.03,)|
OC(=O)c1ccc(c2C3C=CCC3C(Nc12)c1ccc(Cl)cc1)[N+]([O-])=O |c:9|
CCCCC[C@H](O)[C@H](O)/C=C/C=C/C=CC=C[C@@H](O)CCCC(=O)O
Cc1c(nc2ccc(Br)cc2c1C(=O)NC[C@H](CC(O)=O)c1ccccc1Cl)-c1ccccc1 |r|