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Report error Found 27 Enz. Inhib. hit(s) with Target = 'cAMP-dependent protein kinase type I-alpha regulatory subunit'
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81289(cid_23669773 | MLS001333136 | sodium;(4aR,6R,7R,7a...)
Affinity DataEC50:  68.0nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit [K244A](Human)
University of California San Diego

LigandPNGBDBM218808(8-[Fluo]-cAMP)
Affinity DataKd:  7.71nMAssay Description:The ability of the R subunit basic patch mutants to bind cAMP in the absence of the C subunit was tested using the fluorescent cAMP analogue, 8-[fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2017
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit [R243A](Human)
University of California San Diego

LigandPNGBDBM218808(8-[Fluo]-cAMP)
Affinity DataKd:  7.29nMAssay Description:The ability of the R subunit basic patch mutants to bind cAMP in the absence of the C subunit was tested using the fluorescent cAMP analogue, 8-[fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2017
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit [K242A](Human)
University of California San Diego

LigandPNGBDBM218808(8-[Fluo]-cAMP)
Affinity DataKd:  7.32nMAssay Description:The ability of the R subunit basic patch mutants to bind cAMP in the absence of the C subunit was tested using the fluorescent cAMP analogue, 8-[fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2017
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit [R241A](Human)
University of California San Diego

LigandPNGBDBM218808(8-[Fluo]-cAMP)
Affinity DataKd:  6.72nMAssay Description:The ability of the R subunit basic patch mutants to bind cAMP in the absence of the C subunit was tested using the fluorescent cAMP analogue, 8-[fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2017
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Human)
University of California San Diego

LigandPNGBDBM218808(8-[Fluo]-cAMP)
Affinity DataKd:  7.30nMAssay Description:The ability of the R subunit basic patch mutants to bind cAMP in the absence of the C subunit was tested using the fluorescent cAMP analogue, 8-[fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2017
Entry Details Article
PubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81290(sodium;[(4aR,6R,7R,7aR)-6-[6-(butanoylamino)purin-...)
Affinity DataEC50:  1.23E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM66980(MLS002154012 | sodium;butanoic acid [(4aS,5R,6R,7a...)
Affinity DataEC50:  6.70E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81292(8-Bromoadenosine 3',5'-cyclic monophosphat...)
Affinity DataEC50:  34.4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81291(sodium;(4aR,6R,7R,7aS)-6-[6-azanyl-8-(4-chlorophen...)
Affinity DataEC50:  32.7nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81290(sodium;[(4aR,6R,7R,7aR)-6-[6-(butanoylamino)purin-...)
Affinity DataEC50:  4.48E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81287(SMR000450983 | cid_4132952 | 6-(6-aminopurin-9-yl)...)
Affinity DataEC50:  2.68E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM51788(cid_5876309 | 5-[(2E)-2-(8-oxidanylidenequinolin-5...)
Affinity DataEC50: >1.14E+5nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81288(SMR000326870 | MLS000860011 | sodium;9-[(4aR,6R,7R...)
Affinity DataEC50:  7.83E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81287(SMR000450983 | cid_4132952 | 6-(6-aminopurin-9-yl)...)
Affinity DataEC50:  2.68E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81295(cid_23679857 | sodium;4-[[4-(dimethylamino)naphtha...)
Affinity DataEC50: >1.14E+5nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81294(MLS000328052 | SMR000168585 | 3-[(2,4-dichlorobenz...)
Affinity DataEC50: >1.14E+5nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81290(sodium;[(4aR,6R,7R,7aR)-6-[6-(butanoylamino)purin-...)
Affinity DataEC50:  1.23E+4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM66980(MLS002154012 | sodium;butanoic acid [(4aS,5R,6R,7a...)
Affinity DataEC50:  6.70E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81292(8-Bromoadenosine 3',5'-cyclic monophosphat...)
Affinity DataEC50:  34.4nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81291(sodium;(4aR,6R,7R,7aS)-6-[6-azanyl-8-(4-chlorophen...)
Affinity DataEC50:  32.7nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81290(sodium;[(4aR,6R,7R,7aR)-6-[6-(butanoylamino)purin-...)
Affinity DataEC50:  4.48E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81289(cid_23669773 | MLS001333136 | sodium;(4aR,6R,7R,7a...)
Affinity DataEC50:  68.0nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM81288(SMR000326870 | MLS000860011 | sodium;9-[(4aR,6R,7R...)
Affinity DataEC50:  7.83E+3nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Affiliation: The Scripps Research Institute, TSRI Assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/4/2011
Entry Details
PCBioAssay
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM50011236(Isoquinoline-5-sulfonic acid (2-amino-ethyl)-amide...)
Affinity DataIC50: 3.60E+3nMpH: 7.4 T: 2°CAssay Description:Casein kinase activities were determined under the conditions as described by Huang et al (1982).More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2013
Entry Details
PubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM92674(Isoquinolinesulfonamide, CKI-7)
Affinity DataIC50: 5.50E+5nMpH: 7.4 T: 2°CAssay Description:Casein kinase activities were determined under the conditions as described by Huang et al (1982).More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2013
Entry Details
PubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bovine)
The Scripps Research Institute Molecular Screening Center

Curated by PubChem BioAssay
LigandPNGBDBM92673(Isoquinolinesulfonamide, CKI-6)
Affinity DataIC50: 1.00E+6nMpH: 7.4 T: 2°CAssay Description:Casein kinase activities were determined under the conditions as described by Huang et al (1982).More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2013
Entry Details
PubMed