Compile Data Set for Download or QSAR
Report error Found 247 Enz. Inhib. hit(s) with Target = 'Vasopressin V1a/V1b receptor'
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016312(CHEMBL265119 | [Sar7D-Arg8]VP (Vasopressin ))
Affinity DataKd:  650nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016314(CHEMBL269715 | [MeAla7D-Arg8]VP (Vasopressin ))
Affinity DataKd:  280nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016314(CHEMBL269715 | [MeAla7D-Arg8]VP (Vasopressin ))
Affinity DataKd:  440nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016312(CHEMBL265119 | [Sar7D-Arg8]VP (Vasopressin ))
Affinity DataKd:  420nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016311(CHEMBL413249 | [Mpa1Sar7,Drg8]VP (Vasopressin ))
Affinity DataKd:  160nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016315(CHEMBL437631 | [Val4MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  310nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016315(CHEMBL437631 | [Val4MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  480nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016317(CHEMBL2371674 | [Mpa1Val4MeAla7]AVP (Arginine-vaso...)
Affinity DataKd:  53nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016311(CHEMBL413249 | [Mpa1Sar7,Drg8]VP (Vasopressin ))
Affinity DataKd:  240nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016317(CHEMBL2371674 | [Mpa1Val4MeAla7]AVP (Arginine-vaso...)
Affinity DataKd:  82nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016309(CHEMBL410025 | [Phe2Sar7]AVP (Arginine-vasopressin...)
Affinity DataKd:  170nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016318(CHEMBL411357 | [Mpa1,MeAla7,D-Arg8]VP (Vasopressin...)
Affinity DataKd:  290nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016309(CHEMBL410025 | [Phe2Sar7]AVP (Arginine-vasopressin...)
Affinity DataKd:  260nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016310(CHEMBL406303 | [Mpa1Val4Sar7]AVP (Arginine-vasopre...)
Affinity DataKd:  42nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016316(CHEMBL413706 | [Phe2MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  110nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016316(CHEMBL413706 | [Phe2MeAla7]AVP (Arginine-vasopress...)
Affinity DataKd:  170nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016310(CHEMBL406303 | [Mpa1Val4Sar7]AVP (Arginine-vasopre...)
Affinity DataKd:  27nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016318(CHEMBL411357 | [Mpa1,MeAla7,D-Arg8]VP (Vasopressin...)
Affinity DataKd:  450nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016313(CHEMBL217517 | [Val4Sar7]AVP (Arginine-vasopressin...)
Affinity DataKd:  110nMAssay Description:Binding affinity against plasma membrane from rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016313(CHEMBL217517 | [Val4Sar7]AVP (Arginine-vasopressin...)
Affinity DataKd:  170nMAssay Description:Binding affinity against plasma membrane from rat liver using [3H]-AVP as a radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075817(Mpa-Car-lle-Gln-Asn-Cys-Sar-Arg-Gly-NH2 | CHEMBL23...)
Affinity DataKd:  18nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075816(Mca1,D-Trp2,Sar7AVT | CHEMBL264208)
Affinity DataKd:  3.80nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50403723(CHEMBL2110163)
Affinity DataKd:  1.76E+4nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075817(Mpa-Car-lle-Gln-Asn-Cys-Sar-Arg-Gly-NH2 | CHEMBL23...)
Affinity DataKd:  17.8nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataKd:  0.650nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075818(Mpa1,D-Phe2,Sar7AVT | CHEMBL157988)
Affinity DataKd:  50nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50403724(CHEMBL2110297)
Affinity DataKd:  2.64E+3nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075820(Mpa-D-Trp-lle-Gln-Asn-Cys-Sar-Arg-Gly-NH2 | CHEMBL...)
Affinity DataKd:  888nMAssay Description:Compound was evaluated for its dissociation constant (Kd) to rat liver Vasopressin V1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/30/2012
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137948(Biphenyl-2-carboxylic acid [2-[3-(4-methyl-[1,4]di...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50137948(Biphenyl-2-carboxylic acid [2-[3-(4-methyl-[1,4]di...)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50137945(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-piperaz...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137940(Biphenyl-2-carboxylic acid [2-[4-(4-dimethylamino-...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137953(Biphenyl-2-carboxylic acid [2-[4-(4-diethylamino-p...)
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50137953(Biphenyl-2-carboxylic acid [2-[4-(4-diethylamino-p...)
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137945(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-piperaz...)
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137951(Biphenyl-2-carboxylic acid [2-{4-[(2-dimethylamino...)
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50137940(Biphenyl-2-carboxylic acid [2-[4-(4-dimethylamino-...)
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291329(8-arginine vasopressin trisulphide | CHEMBL267405)
Affinity DataIC50: 9.5nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM35667([3H]Argipressin tannate | AVP | [3H]Arginine vasop...)
Affinity DataIC50: 10nMAssay Description:Tested for the TYR(Me)2 arginine-vasopressin as radioligand at 0.3 nM in A7r5 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137942(Biphenyl-2-carboxylic acid [2-(4-[1,4']bipiperidin...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137956(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-piperaz...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50137949(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-[1,4]di...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50137951(Biphenyl-2-carboxylic acid [2-{4-[(2-dimethylamino...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50137946(Biphenyl-2-carboxylic acid [2-[2-(4-dimethylamino-...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50137942(Biphenyl-2-carboxylic acid [2-(4-[1,4']bipiperidin...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50137956(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-piperaz...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in rat liverMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137949(Biphenyl-2-carboxylic acid [2-[4-(4-methyl-[1,4]di...)
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50137946(Biphenyl-2-carboxylic acid [2-[2-(4-dimethylamino-...)
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Human)
Central Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50204026(CHEMBL369150)
Affinity DataIC50: 60nMAssay Description:Inhibitory activity against arginine vasopressin V1 receptor using [3H]AVP as radioligand in human plateletMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V1a/V1b receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50043204(1N-[2-hydroxy-7,7-dimethyl-1-spiro[1H-indene-1,4'-...)
Affinity DataIC50: 67nMAssay Description:Inhibition of radioligand [3H]AVP binding to the vasopressin V1 receptor in rat liver tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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