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Report error Found 10 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ABL1 [Y253F]'
TargetTyrosine-protein kinase ABL1 [Y253F](Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM332698(US10196378, Compound C01)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
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TargetTyrosine-protein kinase ABL1 [Y253F](Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM332699(US10196378, Compound C02)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
Go to US Patent

TargetTyrosine-protein kinase ABL1 [Y253F](Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM332700(US10196378, Compound C03)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
Go to US Patent

TargetTyrosine-protein kinase ABL1 [Y253F](Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM332702(US10196378, Compound C05)
Affinity DataKi: <1nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
Go to US Patent

TargetTyrosine-protein kinase ABL1 [Y253F](Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM332706(US10196378, Compound C10 | US10196378, Compound C0...)
Affinity DataKi:  2.5nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
Go to US Patent

TargetTyrosine-protein kinase ABL1 [Y253F](Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM332705(US10196378, Compound C08)
Affinity DataKi:  3.40nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
Go to US Patent

TargetTyrosine-protein kinase ABL1 [Y253F](Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM332703(US10196378, Compound C06)
Affinity DataKi:  6.20nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
Go to US Patent

TargetTyrosine-protein kinase ABL1 [Y253F](Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM332706(US10196378, Compound C10 | US10196378, Compound C0...)
Affinity DataKi:  7.60nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
Go to US Patent

TargetTyrosine-protein kinase ABL1 [Y253F](Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM332701(US10196378, Compound C04)
Affinity DataKi:  50nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
Go to US Patent

TargetTyrosine-protein kinase ABL1 [Y253F](Human)
The Regents of The University of Michigan

US Patent
LigandPNGBDBM332704(US10196378, Compound C07)
Affinity DataKi: >9.00E+3nMAssay Description:The biochemical assays were carried out using the non-phosphorylated kinase domain of c-Abl, Bcr-Abl in Ba/F3 cells is in the phosphorylated state.More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2019
Entry Details
Go to US Patent