Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with Target = 'Thymidine kinase 2, mitochondrial (Predicted)'
LigandPNGBDBM50028586(1-(4-Benzyloxy-5-hydroxymethyl-tetrahydro-furan-2-...)
Affinity DataKi:  8.00E+3nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50404860(CHEMBL2111285)
Affinity DataKi:  1.10E+4nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50028587(1-(4-Ethylsulfanyl-5-hydroxymethyl-tetrahydro-fura...)
Affinity DataKi:  6.20E+4nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50000966(CHEMBL3143491)
Affinity DataKi:  7.20E+4nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50028583(1-(4-Hydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl...)
Affinity DataKi:  7.70E+4nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50028579(1-(4-Hydroxy-5-hydroxymethyl-tetrahydro-furan-2-yl...)
Affinity DataKi:  2.50E+5nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50367094(DEOXYCYTIDINE | EN300-6477283)
Affinity DataKi:  3.20E+5nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50018445(cid_5280 | 1-((2R,5S)-5-(hydroxymethyl)tetrahydrof...)
Affinity DataKi:  8.80E+5nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50028581(1-(5-Hexylaminomethyl-4-hydroxy-tetrahydro-furan-2...)
Affinity DataKi:  9.60E+5nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50000969(CHEMBL3143490)
Affinity DataKi:  1.10E+6nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50132294(1-((2R,5S)-4-Amino-5-hydroxymethyl-tetrahydro-fura...)
Affinity DataKi:  2.60E+6nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50013111(2',3'-didehydro-3'-deoxythymidine | 1-(5-Hydroxyme...)
Affinity DataKi:  3.25E+6nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50028576(1-(5-Ethylaminomethyl-4-hydroxy-tetrahydro-furan-2...)
Affinity DataKi:  1.44E+6nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
LigandPNGBDBM50132297(1-((2R,4S,5R)-5-(aminomethyl)-4-hydroxy-tetrahydro...)
Affinity DataKi:  4.60E+6nMAssay Description:Competitive inhibition against rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed