Report error Found 328 Enz. Inhib. hit(s) with Target = 'Thymidine kinase, cytosolic'
Displayed 1 to 50 (of 328 total ) | Next | Last >>
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against HSV-1 Thymidine kinase in OST-TK-/HSV-1 TK+ cell line in combination with gancicclovirMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against HSV-1 Thymidine kinase in OST-TK-/HSV-1 TK+ cell line in combination with BVAraUMore data for this Ligand-Target Pair
Affinity DataKd: 15nMAssay Description:Binding affinity to human TK1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibitory activity (50 uM) against HSV-1 Thymidine kinase in OST-TK-/HSV-1 TK+ cell line in combination with BVAraUMore data for this Ligand-Target Pair
Affinity DataIC50: 26nMAssay Description:Inhibitory activity (50 uM) against HSV-1 Thymidine kinase in OST-TK-/HSV-1 TK+ cell line in combination with gancicclovirMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Binding affinity towards HSV-1 thymidine kinase was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Compound was evaluated for Kinetic constant for viral thymidine kinase of Herpes simplex virus (HSV) -1More data for this Ligand-Target Pair
Affinity DataKi: 90nMAssay Description:Binding affinity constant against HSV-1 thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity constant against HSV-1 thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:Compound was evaluated for Kinetic constant for viral thymidine kinase of Herpes simplex virus (HSV) -1More data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Compound was evaluated for Kinetic constant for viral thymidine kinase of Herpes simplex virus (HSV) -1More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibitory activity against HSV-1 Thymidine kinase in OST-TK-/HSV-1 TK+ cell line in combination with gancicclovirMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity constant against HSV-1 thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Binding affinity constant against HSV-1 thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:Binding affinity constant against HSV-1 thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 230nMAssay Description:Inhibitory activity against HSV-1 Thymidine kinase in OST-TK-/HSV-1 TK+ cell line in combination with gancicclovirMore data for this Ligand-Target Pair
Affinity DataIC50: 390nMAssay Description:Inhibitory concentration against HSV-1 TK (WT) catalyzed [3H]-GCV phosphorylationMore data for this Ligand-Target Pair
Affinity DataKi: 440nMAssay Description:Compound was evaluated for Kinetic constant for viral thymidine kinase of Herpes simplex virus (HSV) -2More data for this Ligand-Target Pair
Affinity DataKi: 950nMAssay Description:Compound was evaluated for Kinetic constant for viral thymidine kinase of Herpes simplex virus (HSV) -2More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Compound was evaluated for inhibitory effect against phosphorylation of [methyl-3H]dThd by HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Compound was evaluated for Kinetic constant for viral thymidine kinase of Herpes simplex virus (HSV) -2More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory concentration on phosphorylation of [methyl-3H]-dTh by human Thymidine Kinase 2More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibitory effect against phosphorylation of [methyl-3H]dThd by Thymidine Kinase 2 (TK-2)More data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibitory concentration against HSV-1 TK (WT) catalyzed [3H]-GCV phosphorylationMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity against HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of HSV-1 thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Compound was tested for the binding affinity to thymidine kinase from HSV-1 infected HeLa BuMore data for this Ligand-Target Pair
Affinity DataKi: 2.06E+3nMAssay Description:Binding affinity towards HSV-1 thymidine kinase was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibitory activity against HSV-1 Thymidine kinase in OST-TK-/HSV-1 TK+ cell line in combination with BVAraUMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibitory concentration on phosphorylation of [methyl-3H]-dTh by human Thymidine Kinase 2More data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Competitive inhibition against rat Mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Binding affinity against HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.90E+3nMAssay Description:Inhibitory affect against rabbit thymus thymidine kinase and represented as molt/4F kinase.More data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human TK1 by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Compound was evaluated for inhibitory effect against phosphorylation of [methyl-3H]dThd by HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Compound was evaluated for inhibitory effect against phosphorylation of [methyl-3H]dThd by HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibitory activity against HSV-1 Thymidine kinase in OST-TK-/HSV-1 TK+ cell line in combination with BVAraUMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibitory effect against phosphorylation of [methyl-3H]dThd by Thymidine Kinase 2 (TK-2)More data for this Ligand-Target Pair
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibitory concentration on phosphorylation of [methyl-3H]-dTh by human Thymidine Kinase 2More data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory effect against phosphorylation of [methyl-3H]dThd by Thymidine Kinase 2 (TK-2)More data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Evaluated for the mixed objective Non-competitive inhibition constant Ki against TdR varied rat mitochondrial thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.90E+3nMAssay Description:Competitive inhibition against rat cytoplasmic Thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.90E+3nMAssay Description:Competitive inhibition against rat cytoplasmic Thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nMAssay Description:Compound was tested for the binding affinity to thymidine kinase from Varicella zoster virus infected human cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibitory concentration on phosphorylation of [methyl-3H]-dTh by human Thymidine Kinase 2More data for this Ligand-Target Pair
Affinity DataKi: 4.30E+3nMAssay Description:Binding affinity against HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibitory effect against phosphorylation of [methyl-3H]dThd by Thymidine Kinase 2 (TK-2)More data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibitory effect against phosphorylation of [methyl-3H]dThd by Thymidine Kinase 2 (TK-2)More data for this Ligand-Target Pair
Affinity DataKi: 4.70E+3nMAssay Description:In Vitro inhibition of Thymidine Monophosphatase Kinase (TMPKh)More data for this Ligand-Target Pair






























