Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with Target = 'TAR DNA-binding protein 43'
TargetTAR DNA-binding protein 43(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50544713(CHEMBL4638490)
Affinity DataKd:  8.90E+4nMAssay Description:Binding affinity to TDP-43 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetTAR DNA-binding protein 43(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  176nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetTAR DNA-binding protein 43(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50652792(CHEMBL3752910)
Affinity DataKd:  814nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetTAR DNA-binding protein 43(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50544711(CHEMBL4647070)
Affinity DataIC50: 100nMAssay Description:Inhibition of TDP-43 (unknown origin) binding to RNAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetTAR DNA-binding protein 43(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50544712(CHEMBL4635203)
Affinity DataIC50: 100nMAssay Description:Inhibition of TDP-43 (unknown origin) binding to RNAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetTAR DNA-binding protein 43(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM67690(SMR000058480 | DHAD | 1,4-bis[2-(2-hydroxyethylami...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of TDP-43 (unknown origin) binding to RNAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetTAR DNA-binding protein 43(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM16435(5-(1,2-dithiolan-3-yl)pentanamide | Thioctamide | ...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of TDP-43 (unknown origin) binding to RNAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetTAR DNA-binding protein 43(Human)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50106731((R)-(+)-lipoic acid | (R)-1,2-Dithiolane-3-pentano...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of TDP-43 (unknown origin) binding to RNAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed