Report error Found 105 Enz. Inhib. hit(s) with Target = 'Sodium/potassium-transporting ATPase subunit alpha-1'
TargetSodium/potassium-transporting ATPase subunit alpha-1(Human)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Ligand Info
TargetSodium/potassium-transporting ATPase subunit alpha-1(Human)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Ligand Info
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 8.30nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 45.5nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
Affinity DataIC50: 68nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of Beagle dog kidney NA+/K+ ATPase alpha 1 by measuring 32P-ATP hydrolysis preincubated for 10 mins followed by addition of 32P-ATP measur...More data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Human)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataIC50: 290nMAssay Description:Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric methodMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Human)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric methodMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Human)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric methodMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 660nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 1.25E+3nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 1.58E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 1.58E+3nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 1.89E+3nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Ligand Info
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 3.22E+3nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 3.98E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
Affinity DataIC50: 4.08E+3nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1/beta-1(Rat)
University of Minnesota
Curated by ChEMBL
University of Minnesota
Curated by ChEMBL
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibition of recombinant rat Na+/K+-ATPase alpha1/beta1 expressed in baculovirus infected insect Sf9 cell membranes using [gamma-32P]ATP as substrat...More data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 4.73E+3nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 6.30E+3nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 6.31E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Rat)
Albert-Ludwigs-University of Freiburg
Curated by ChEMBL
Albert-Ludwigs-University of Freiburg
Curated by ChEMBL
Affinity DataIC50: 8.23E+3nMAssay Description:Inhibition of Wistar rat kidney Na+,K+-ATPase alpha1 after 2 hrsMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Human)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataIC50: 9.80E+3nMAssay Description:Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric methodMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Human)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.21E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Dog)
University of Manitoba
Curated by ChEMBL
University of Manitoba
Curated by ChEMBL
Affinity DataIC50: 4.00E+4nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair



3D Structure (crystal)







































