Report error Found 347 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase haspin'
Displayed 1 to 50 (of 347 total ) | Next | Last >>
Affinity DataIC50: 0.00200nMAssay Description:Inhibition of human haspin preincubated for 30 mins followed by ATP and ULight-histone H3 peptide/ULight-eIF4E binding protein addition and measured ...More data for this Ligand-Target Pair
Affinity DataKd: 0.0190nMpH: 7.5Assay Description:All measurements were performed in HEPES (50 mm, pH 7.5) containing NaCl (150 mm), Tween-20 (0.005%) and DTT (5 mm) according to a previously publish...More data for this Ligand-Target Pair
Affinity DataKd: 0.0190nMAssay Description:Binding affinity to haspin (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 0.0190nMAssay Description:Binding affinity to a TEV-cleavable N-terminal His6-tagged human recombinant haspin (470 to 798 residues) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0350nMAssay Description:Inhibition of human haspin preincubated for 30 mins followed by ATP and ULight-histone H3 peptide/ULight-eIF4E binding protein addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0840nMAssay Description:Inhibition of human haspin preincubated for 30 mins followed by ATP and ULight-histone H3 peptide/ULight-eIF4E binding protein addition and measured ...More data for this Ligand-Target Pair
Affinity DataKd: 0.100nMpH: 7.5Assay Description:Association kinetics (Kon): All measurements were performed in HEPES (50 mM, pH 7.5) containing NaCl (150 mM), Tween-20 (0.005%) and DTT (5 mM) accor...More data for this Ligand-Target Pair
Affinity DataKd: 0.120nMpH: 7.5Assay Description:All measurements were performed in HEPES (50 mm, pH 7.5) containing NaCl (150 mm), Tween-20 (0.005%) and DTT (5 mm) according to a previously publish...More data for this Ligand-Target Pair
Affinity DataKd: 0.140nMpH: 7.5Assay Description:All measurements were performed in HEPES (50 mm, pH 7.5) containing NaCl (150 mm), Tween-20 (0.005%) and DTT (5 mm) according to a previously publish...More data for this Ligand-Target Pair
Affinity DataIC50: 0.155nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged haspin (470 to end residues) expressed in baculovirus infected Sf9 cells using histone H3 pepti...More data for this Ligand-Target Pair
Affinity DataKd: <0.170nMAssay Description:Inhibition of haspin (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 0.420nMAssay Description:Binding affinity to N-terminal his6-tagged human recombinant Haspin (470 to 798 residues) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataKd: 0.5nMpH: 7.5Assay Description:All measurements were performed in HEPES (50 mm, pH 7.5) containing NaCl (150 mm), Tween-20 (0.005%) and DTT (5 mm) according to a previously publish...More data for this Ligand-Target Pair
Affinity DataKd: 0.550nMAssay Description:Inhibition of haspin (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
Ligand InfoSimilars
Affinity DataIC50: 1nMAssay Description:Inhibition of human haspin preincubated for 30 mins followed by ATP and ULight-histone H3 peptide/ULight-eIF4E binding protein addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of recombinant human Haspin kinase domain (470 to 798 residues) expressed in bacteria using histone H3 (1 to 21) peptide as substrate incu...More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of haspin (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of haspin (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 2.84nMpH: 7.5Assay Description:Association kinetics (Kon): All measurements were performed in HEPES (50 mM, pH 7.5) containing NaCl (150 mM), Tween-20 (0.005%) and DTT (5 mM) accor...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human Haspin (470 to 798 residues) expressed in bacterial expression system using ARTKQTARKSTGGKAPRKQLA as substrate measur...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of recombinant human Haspin (470 to 798 residues) expressed in bacterial expression system using ARTKQTARKSTGGKAPRKQLA as substrate measur...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of human haspin preincubated for 30 mins followed by ATP and ULight-histone H3 peptide/ULight-eIF4E binding protein addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of recombinant N-terminal His6-tagged human haspin (471 end residues) expressed in baculovirus infected Sf21 insect cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of human haspin preincubated for 30 mins followed by ATP and ULight-histone H3 peptide/ULight-eIF4E binding protein addition and measured ...More data for this Ligand-Target Pair
Affinity DataKd: 4nMAssay Description:Binding affinity to a TEV-cleavable N-terminal His6-tagged human recombinant haspin (470 to 798 residues) assessed as dissociation constantMore data for this Ligand-Target Pair
Affinity DataIC50: 4.80nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of haspin (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of human haspin preincubated for 30 mins followed by ATP and ULight-histone H3 peptide/ULight-eIF4E binding protein addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of human Haspin kinase domain using histone H3 biotin peptide as substrate preincubated with enzyme for 30 mins followed by substrate and ...More data for this Ligand-Target Pair
Affinity DataIC50: 5.03nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
Affinity DataIC50: 5.10nMAssay Description:Inhibition of human Haspin using histone H3 as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition and measured after 120 mins by...More data for this Ligand-Target Pair
Affinity DataIC50: 5.87nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
Affinity DataIC50: 5.87nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of human haspin preincubated for 30 mins followed by ATP and ULight-histone H3 peptide/ULight-eIF4E binding protein addition and measured ...More data for this Ligand-Target Pair
Affinity DataIC50: 6.37nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
Affinity DataIC50: 6.37nMAssay Description:The biochemical assay to measure HASPIN activity relies on the ADP-Glo assay kit (Promega) that determines the amount of ADP as direct product of the...More data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of human haspin preincubated for 30 mins followed by ATP and ULight-histone H3 peptide/ULight-eIF4E binding protein addition and measured ...More data for this Ligand-Target Pair
Affinity DataKd: 8.40nMpH: 7.5Assay Description:All measurements were performed in HEPES (50 mm, pH 7.5) containing NaCl (150 mm), Tween-20 (0.005%) and DTT (5 mm) according to a previously publish...More data for this Ligand-Target Pair
Affinity DataIC50: 8.82nMAssay Description:The kinase assay relies on ADP-GloKM biochemical kinase assay (Promega). This is a luminescent kinase assay that measures ADP formed from a kinase re...More data for this Ligand-Target Pair
Affinity DataIC50: 8.91nMAssay Description:The kinase assay relies on ADP-GloKM biochemical kinase assay (Promega). This is a luminescent kinase assay that measures ADP formed from a kinase re...More data for this Ligand-Target Pair
Affinity DataIC50: 9.56nMAssay Description:The kinase assay relies on ADP-GloKM biochemical kinase assay (Promega). This is a luminescent kinase assay that measures ADP formed from a kinase re...More data for this Ligand-Target Pair
Affinity DataIC50: 9.80nMAssay Description:The kinase assay relies on ADP-GloKM biochemical kinase assay (Promega). This is a luminescent kinase assay that measures ADP formed from a kinase re...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of haspin (V473 to K798) (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of haspin (V473 to K798) (unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 10nMAssay Description:Binding affinity to human HASPINMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Haspin (unknown origin) in presence of [gamma-33P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of haspin (V473 to K798) (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of haspin (V473 to K798) (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of haspin (unknown origin)More data for this Ligand-Target Pair