Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase PKH2 [1-944]'
TargetSerine/threonine-protein kinase PKH2 [1-944](Yeast)
Universit£Tsklinikum Frankfurt

LigandPNGBDBM104016(PS77)
Affinity DataEC50:  4.40E+4nMpH: 7.4Assay Description:The AlphaScreen Assay (Perkin Elmer) was performed according to the manufacturer's protocol in 384-well microtiter plates. Incubations were performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PKH2 [1-944](Yeast)
Universit£Tsklinikum Frankfurt

LigandPNGBDBM50321382(CHEMBL550259 | PS46 | 2-(3-(4-chlorophenyl)-3-oxo-...)
Affinity DataEC50:  8.50E+4nMpH: 7.4 T: 2°CAssay Description:The AlphaScreen Assay (Perkin Elmer) was performed according to the manufacturer's protocol in 384-well microtiter plates. Incubations were performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PKH2 [1-944](Yeast)
Universit£Tsklinikum Frankfurt

LigandPNGBDBM104018(PS182)
Affinity DataEC50:  6.60E+4nMpH: 7.4 T: 2°CAssay Description:The AlphaScreen Assay (Perkin Elmer) was performed according to the manufacturer's protocol in 384-well microtiter plates. Incubations were performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PKH2 [1-944](Yeast)
Universit£Tsklinikum Frankfurt

LigandPNGBDBM50399646(CHEMBL2177668 | PS210)
Affinity DataEC50:  6.00E+4nMpH: 7.4 T: 2°CAssay Description:The AlphaScreen Assay (Perkin Elmer) was performed according to the manufacturer's protocol in 384-well microtiter plates. Incubations were performe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PKH2 [1-944](Yeast)
Universit£Tsklinikum Frankfurt

LigandPNGBDBM104016(PS77)
Affinity DataIC50: 1.70E+4nMpH: 7.4 T: 2°CAssay Description:A 20ul mix containing 50mM Tris pH 7.5, 0.05mg/ml BSA, 0.1% β-mercaptoethanol, 10mM MgCl2, 100μM [γ-P32]ATP (5-50cpm/pmol), 0.003% Bri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2014
Entry Details Article
PubMed