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Report error Found 154 Enz. Inhib. hit(s) with Target = 'REST corepressor 1'
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50507295(CHEMBL1232432)
Affinity DataKd:  243nMAssay Description:Binding affinity to LSD1/CoREST (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50548037(CHEMBL2397513)
Affinity DataKd:  463nMAssay Description:Binding affinity to LSD1/CoREST (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50548038(CHEMBL3781027)
Affinity DataKd:  594nMAssay Description:Binding affinity to LSD1/CoREST (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50507295(CHEMBL1232432)
Affinity DataKd:  243nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594080(CHEMBL5208341)
Affinity DataKd:  1.56E+3nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594081(CHEMBL5199513)
Affinity DataKd:  1.49E+3nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594082(CHEMBL5197685)
Affinity DataKd:  147nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594083(CHEMBL5179091)
Affinity DataKd:  83nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594084(CHEMBL5204694)
Affinity DataKd:  84nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594085(CHEMBL5178765)
Affinity DataKd:  75nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594086(CHEMBL5170197)
Affinity DataKd:  81nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594087(CHEMBL5189687)
Affinity DataKd:  356nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594088(CHEMBL5172748)
Affinity DataKd:  2.85E+3nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594089(CHEMBL5181174)
Affinity DataKd:  975nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594090(CHEMBL5205888)
Affinity DataKd:  82nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594091(CHEMBL5183341)
Affinity DataKd:  251nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594092(CHEMBL5171992)
Affinity DataKd:  115nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594093(CHEMBL5191114)
Affinity DataKd:  228nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594094(CHEMBL5194934)
Affinity DataKd:  230nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594095(CHEMBL5178617)
Affinity DataKd:  237nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594096(CHEMBL5189695)
Affinity DataKd:  112nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594097(CHEMBL5175173)
Affinity DataKd:  162nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594098(CHEMBL5198334)
Affinity DataKd:  64nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594099(CHEMBL5186174)
Affinity DataKd:  86nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594100(CHEMBL5181017)
Affinity DataKd:  82nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594101(CHEMBL5175171)
Affinity DataKd:  68nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594102(CHEMBL5207435)
Affinity DataKd:  369nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594103(CHEMBL5194210)
Affinity DataKd:  191nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594104(CHEMBL5200394)
Affinity DataKd:  82nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594105(CHEMBL5189661)
Affinity DataKd:  1.30E+3nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594106(CHEMBL5202637)
Affinity DataKd:  67nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594107(CHEMBL5189756)
Affinity DataKd:  127nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50262048(CHEMBL3134377)
Affinity DataKd:  14nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50594108(CHEMBL5175660)
Affinity DataKd:  127nMAssay Description:Binding affinity to human LSD1/CoREST assessed as dissociation constant by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/21/2023
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50507295(CHEMBL1232432)
Affinity DataKd:  2.43E+5nMAssay Description:Inhibition of human LSD1-CoREST expressed in Escherichia coli assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50616052(CHEMBL5419693)
Affinity DataKd:  7.78E+3nMAssay Description:Inhibition of human LSD1-CoREST expressed in Escherichia coli assessed as dissociation constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50507295(CHEMBL1232432)
Affinity DataKd:  243nMAssay Description:Inhibition of human LSD1/CoREST expressed in Escherichia coli using histone H3K4me peptide as substrate by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50568523(CHEMBL4875015)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of N-terminal His-SUMO tagged human LSD1 (172 to 852 residues)/His-tagged CoREST (286 to 482 residues) expressed in Escherichia coli BL21 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50153586(CHEMBL3775474 | US10053456, 120 | US9718814, 71 | ...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues)/His-tagged human CoREST (286 to 482 residues) expressed in Escherichia coli BL21 (DE3) cel...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50410785(CHEMBL5291155)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of human recombinant LSD1/CoREST using ART(mK)QTARKSTGGKAPRKQLAGGK-biotin as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50410784(CHEMBL5280566)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of human recombinant LSD1/CoREST using ART(mK)QTARKSTGGKAPRKQLAGGK-biotin as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetREST corepressor 1 [4-485](Human)
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50155773(US9469597, 5 | CHEMBL3781751)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of human recombinant KDM1A/CoREST expressed in Escherichia coli using mono-methylated H3-K4 peptide as substrate assessed as H2O2 release ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2017
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50621408(CHEMBL5399284)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues)/His-tagged human CoREST (286 to 482 residues) expressed in Escherichia coli BL21 (DE3) cel...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50410789(CHEMBL5277056)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of human recombinant LSD1/CoREST using ART(mK)QTARKSTGGKAPRKQLAGGK-biotin as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50410788(CHEMBL5281376)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant LSD1/CoREST using ART(mK)QTARKSTGGKAPRKQLAGGK-biotin as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50621404(CHEMBL5421067)
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human LSD1 (172 to 852 residues)/His-tagged human CoREST (286 to 482 residues) expressed in Escherichia coli BL21 (DE3) cel...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/16/2024
Entry Details
PubMed
TargetREST corepressor 1 [4-485](Human)
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50155579(CHEMBL3546846)
Affinity DataIC50: 19nMAssay Description:Inhibition of human recombinant KDM1A/CoREST expressed in Escherichia coli using mono-methylated H3-K4 peptide as substrate assessed as H2O2 release ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2017
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50403543(CHEMBL5276713)
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant human LSD1/CoREST by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetREST corepressor 1 [4-485](Human)
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50155763(CHEMBL3780391)
Affinity DataIC50: 23nMAssay Description:Inhibition of human recombinant KDM1A/CoREST expressed in Escherichia coli using mono-methylated H3-K4 peptide as substrate assessed as H2O2 release ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2017
Entry Details Article
PubMed
TargetREST corepressor 1(Human)
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50410786(CHEMBL5270114)
Affinity DataIC50: 24nMAssay Description:Inhibition of human recombinant LSD1/CoREST using ART(mK)QTARKSTGGKAPRKQLAGGK-biotin as substrate incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
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