Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with Target = 'Protein arginine N-methyltransferase 7'
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50089221(CHEMBL3577854)
Affinity DataKd:  3.70E+4nMAssay Description:Binding affinity to human full length PRMT7 by Surface plasmon resonance methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50597884(CHEMBL5185202)
Affinity DataIC50: 2.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50597884(CHEMBL5185202)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of PRMT7 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50637569(CHEMBL5562211)
Affinity DataIC50: 2.5nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50637570(CHEMBL5562317)
Affinity DataIC50: 2.5nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant human PRMT7 using GST-GAR as substrate by hotspot assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50598017(CHEMBL5206272)
Affinity DataIC50: 220nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50598020(CHEMBL5202088)
Affinity DataIC50: 226nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50637570(CHEMBL5562317)
Affinity DataIC50: 294nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50598015(CHEMBL5199380)
Affinity DataIC50: 320nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50598018(CHEMBL5180108)
Affinity DataIC50: 410nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50628241(CHEMBL5408585)
Affinity DataIC50: 540nMAssay Description:Inhibition of N-terminal/C-terminal His-tagged human recombinant full-length PRMT7 (2 to 692 residues) using histone GST-GAR as substrate and 3H-SAM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50598016(CHEMBL5170047)
Affinity DataIC50: 550nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50648951(CHEMBL5613785)
Affinity DataIC50: 555nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50598019(CHEMBL5186617)
Affinity DataIC50: 631nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50294572(5'-(Aminopropylthio)-5'-deoxy-adenosine | (2R,3R,4...)
Affinity DataIC50: 1.00E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50598022(CHEMBL5173678)
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50637574(CHEMBL5561462)
Affinity DataIC50: 2.10E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50637572(CHEMBL5563222)
Affinity DataIC50: 2.30E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Mus musculus)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50637571(CHEMBL5562427)
Affinity DataIC50: 2.40E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50637575(CHEMBL5560678)
Affinity DataIC50: 2.40E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50648945(CHEMBL5613745)
Affinity DataIC50: 2.40E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50637573(CHEMBL5527953)
Affinity DataIC50: 2.50E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/11/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50598021(CHEMBL5191769)
Affinity DataIC50: 4.68E+3nMAssay Description:Inhibition of human full length recombinant his-tagged PRMT7 (2 to 692 residues) using GST-GAR as substrate incubated for 20 mins in presence of [3H]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50628242(CHEMBL5396270)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of N-terminal/C-terminal His-tagged human recombinant full-length PRMT7 (2 to 692 residues) using histone GST-GAR as substrate and 3H-SAM ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2024
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50089221(CHEMBL3577854)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human full length PRMT7 expressed in Sf9 cells assessed as inhibition of H2B[23-37] methylationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50396023(CHEMBL2169919)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of human full length PRMT7 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50648950(CHEMBL5613744)
Affinity DataIC50: 8.30E+3nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM378654(US10266526, Compound 792 | N-{1-[(1-benzyl-1H-pyra...)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50652922(CHEMBL5678791)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50462572(CHEMBL4249337)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM378802(US10266526, Compound 985 | N-(1-((1-(4-chlorobenzy...)
Affinity DataIC50: 1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50247634(CHEMBL4067973)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of PRMT7 (unknown origin) using [3H]-SAM as co-factor by scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/3/2019
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50550092(CHEMBL4740128)
Affinity DataIC50: 2.33E+4nMAssay Description:Inhibition of recombinant GST-tagged PRMT7 (unknown origin) expressed in Escherichia coli using biotin-labeled SMD1 as substrate incubated for 120 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50550091(CHEMBL4648477)
Affinity DataIC50: 2.36E+4nMAssay Description:Inhibition of recombinant GST-tagged PRMT7 (unknown origin) expressed in Escherichia coli using biotin-labeled SMD1 as substrate incubated for 120 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50525201(CHEMBL4463124)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of recombinant full-length human PRMT7 expressed in Sf9 insect cells using Ac-KKDGKKRKRSRKESYK-biotin as substrate measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50609300(CHEMBL5266562)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of PRMT7 (unknown origin) by radioisotope based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/20/2024
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50089221(CHEMBL3577854)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human full length PRMT7 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human full length PRMT7 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2016
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50551136(CHEMBL4757320)
Affinity DataIC50: 6.15E+4nMAssay Description:Inhibition of recombinant human PRMT7 using GST-GAR as substrate by hotspot assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50551131(CHEMBL4787257)
Affinity DataIC50: 6.94E+4nMAssay Description:Inhibition of recombinant human PRMT7 using GST-GAR as substrate by hotspot assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM223137(P5i-6)
Affinity DataIC50: 1.00E+5nMT: 2°CAssay Description:All in vitro enzymatic assays were carried out by Shanghai ChemPartner Co. (998 Halei Road, Pudong New Area, Shanghai, 201203, China). To measure the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/26/2017
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50238541(CHEMBL4092336)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human N-terminal His-tagged full length PRMT7 expressed in baculovirus using of histone H4 as substrate preincubated for 15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/8/2019
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532859(CHEMBL4436627)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT7 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50532859(CHEMBL4436627)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of PRMT7 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50643958(CHEMBL5566004)
Affinity DataIC50: 1.00E+5nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/12/2025
Entry Details
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50529897(CHEMBL4468383)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant full length human N-terminal FLAG-tagged PRMT7 expressed in Sf9 insect cells preincubated for 15 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50529897(CHEMBL4468383)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant full length human N-terminal FLAG-tagged PRMT7 expressed in Sf9 insect cells preincubated for 15 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50550095(CHEMBL4792295)
Affinity DataIC50: 1.26E+5nMAssay Description:Inhibition of recombinant GST-tagged PRMT7 (unknown origin) expressed in Escherichia coli using biotin-labeled SMD1 as substrate incubated for 120 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetProtein arginine N-methyltransferase 7(Human)
University of Toronto

Curated by ChEMBL
LigandPNGBDBM50550093(CHEMBL4755950)
Affinity DataIC50: 2.48E+5nMAssay Description:Inhibition of recombinant GST-tagged PRMT7 (unknown origin) expressed in Escherichia coli using biotin-labeled SMD1 as substrate incubated for 120 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
Displayed 1 to 50 (of 52 total ) | Next | Last >>
Jump to: