Compile Data Set for Download or QSAR
Report error Found 212 Enz. Inhib. hit(s) with Target = 'Protein ENL'
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459744(CHEMBL4204744)
Affinity DataKd:  57nMAssay Description:Binding affinity to MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) by Bio-layer interferometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50466617(CHEMBL4287247)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to recombinant C-terminal His6-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in expressed Escherichia coli ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50466618(CHEMBL4280015)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to recombinant C-terminal His6-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in expressed Escherichia coli ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50466619(CHEMBL4290656)
Affinity DataKd:  2.30E+3nMAssay Description:Binding affinity to recombinant C-terminal His6-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in expressed Escherichia coli ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50466620(CHEMBL4283481)
Affinity DataKd:  800nMAssay Description:Binding affinity to recombinant C-terminal His6-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in expressed Escherichia coli ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50466621(CHEMBL4295184)
Affinity DataKd:  1.10E+3nMAssay Description:Binding affinity to recombinant C-terminal His6-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in expressed Escherichia coli ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529555(CHEMBL4524997)
Affinity DataKd:  1.71E+4nMAssay Description:Binding affinity to C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by isotherma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529557(CHEMBL4588022)
Affinity DataKd:  1.81E+4nMAssay Description:Binding affinity to C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by isotherma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50466617(CHEMBL4287247)
Affinity DataKd:  6.10E+3nMAssay Description:Binding affinity to C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by isotherma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50466619(CHEMBL4290656)
Affinity DataKd:  3.50E+3nMAssay Description:Binding affinity to C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by isotherma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529556(CHEMBL4552313)
Affinity DataKd:  113nMAssay Description:Binding affinity to human MLLT1 by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529558(CHEMBL4456056)
Affinity DataKd:  5.50E+3nMAssay Description:Binding affinity to C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by isotherma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529559(CHEMBL4444396)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to C-terminal His6-tagged MLLT1 YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli Rosetta by isotherma...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50566877(CHEMBL4863719)
Affinity DataKd:  45nMAssay Description:Binding affinity to human His-ENL YEATS domain assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50566890(CHEMBL4865432)
Affinity DataKd:  46nMAssay Description:Binding affinity to human His-ENL YEATS domain assessed as dissociation constant by SPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50596391(CHEMBL5171384)
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity to His6-tagged ENL YEATS domain (unknown origin) expressed in Escherichia coli BL21 DE3 assessed as dissociation constant by surface...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625619(CHEMBL4752253)
Affinity DataKd:  110nMAssay Description:Binding affinity to MLLT1 YD domain (unknown origin) assessed as dissociation constant by biolayer interferometry assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625619(CHEMBL4752253)
Affinity DataKd:  82nMAssay Description:Binding affinity to MLLT1 YD domain (unknown origin) assessed as dissociation constant by isothermal calorimetry assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529556(CHEMBL4552313)
Affinity DataKd:  25nMAssay Description:Binding affinity to C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617561(CHEMBL5438748)
Affinity DataKd:  17nMAssay Description:Binding affinity to C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells asses...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617566(CHEMBL5418051)
Affinity DataKd:  1.40E+4nMAssay Description:Binding affinity toC-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) assessed as dissociation constant by BLI assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617567(CHEMBL5395794)
Affinity DataKd:  119nMAssay Description:Binding affinity to 3xFLAG-HA-tagged wild-type human ENL YEATS domain assessed as dissociation constant by ITC titration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50576674(CHEMBL4850575)
Affinity DataKd:  1.41E+4nMAssay Description:Binding affinity to ENL YEATS domain (unknown origin) assessed as dissociation constant by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617568(CHEMBL5408148)
Affinity DataKd:  754nMAssay Description:Binding affinity to C-terminal ENL YEATS domain (unknown origin) (M1 to A148 residues) assessed as dissociation constant by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617569(CHEMBL5418436)
Affinity DataKd:  30nMAssay Description:Binding affinity to C-terminal 6-His tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21 cells assessed a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529556(CHEMBL4552313)
Affinity DataKd:  129nMAssay Description:Binding affinity to wild type human ENL YEATS domain assessed as dissociation constant by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529556(CHEMBL4552313)
Affinity DataKd:  100nMAssay Description:Binding affinity to ENL YEATS domain (unknown origin) at 100 uM by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50623073(CHEMBL5410133)
Affinity DataKd:  160nMAssay Description:Binding affinity to ENL YEATS domain (unknown origin) at 100 uM by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617567(CHEMBL5395794)
Affinity DataKd:  120nMAssay Description:Binding affinity to ENL YEATS domain (unknown origin) at 100 uM by ITC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617558(CHEMBL5400413)
Affinity DataIC50: 11nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529556(CHEMBL4552313)
Affinity DataIC50: 14nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617550(CHEMBL5423431)
Affinity DataIC50: 15nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617561(CHEMBL5438748)
Affinity DataIC50: 15nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617544(CHEMBL5397340)
Affinity DataIC50: 17nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617549(CHEMBL5411777)
Affinity DataIC50: 17nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529556(CHEMBL4552313)
Affinity DataIC50: 18nMAssay Description:Inhibition of His6-tagged ENL YEATS domain (unknown origin) expressed in Escherichia coli BL21 DE3 and biotinylated H3K27ac peptide interaction using...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617542(CHEMBL5404010)
Affinity DataIC50: 19nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617551(CHEMBL5427068)
Affinity DataIC50: 19nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617556(CHEMBL5416453)
Affinity DataIC50: 22nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617563(CHEMBL5430847)
Affinity DataIC50: 22nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617569(CHEMBL5418436)
Affinity DataIC50: 25nMAssay Description:Inhibition of recombinant C-terminal 6-His tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21 cells usin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617569(CHEMBL5418436)
Affinity DataIC50: 25nMAssay Description:Inhibition of N-terminal StrepII-SUMO or SUMO-AviTag/Cterminal 6xHis tagged ENL (unknown origin) (1 to 148 residues) expressed in Escherichia coli BL...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617548(CHEMBL5400474)
Affinity DataIC50: 28nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617555(CHEMBL5414763)
Affinity DataIC50: 32nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617564(CHEMBL5421344)
Affinity DataIC50: 32nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617545(CHEMBL5395585)
Affinity DataIC50: 35nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617552(CHEMBL5438461)
Affinity DataIC50: 35nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617543(CHEMBL5429534)
Affinity DataIC50: 37nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50617547(CHEMBL5417838)
Affinity DataIC50: 38nMAssay Description:Inhibition of C-terminal 6xHis-tagged ENL YEATS domain (1 to 148 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cells using bioti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetProtein ENL(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50623091(CHEMBL5437942)
Affinity DataIC50: 40nMAssay Description:Inhibition of 5x6His-tagged ENL YEATS domain (unknown origin) using biotinylated peptide H3K9cr (1 to 20 residues) preincubated for 15 mins followed ...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
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