Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with Target = 'Proteasome subunit alpha type-2'
TargetProteasome subunit alpha type-2(Baker's yeast)
University of California San Diego

LigandPNGBDBM154579((2S)-2-[(2S)-2-hexanamido-3-methylbutanamido]-N,N-...)
Affinity DataIC50: 1.20nMpH: 7.5Assay Description:One nanomolar of proteasome was incubated with different inhibitor concentrations in Tris 25 mM pH 7.5; SDS 0.03%; EDTA 0.5 mM for 15 min at 37 °C in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2015
Entry Details Article
PubMed
TargetProteasome subunit alpha type-2(Baker's yeast)
University of California San Diego

LigandPNGBDBM154578(Carmaphycin A (1))
Affinity DataIC50: 1.5nMpH: 7.5Assay Description:One nanomolar of proteasome was incubated with different inhibitor concentrations in Tris 25 mM pH 7.5; SDS 0.03%; EDTA 0.5 mM for 15 min at 37 °C in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2015
Entry Details Article
PubMed
TargetProteasome subunit alpha type-2(Baker's yeast)
University of California San Diego

LigandPNGBDBM154578(Carmaphycin A (1))
Affinity DataIC50: 46.2nMpH: 7.5Assay Description:One nanomolar of proteasome was incubated with different inhibitor concentrations in Tris 25 mM pH 7.5; SDS 0.03%; EDTA 0.5 mM for 15 min at 37 °C in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2015
Entry Details Article
PubMed
TargetProteasome subunit alpha type-2(Baker's yeast)
University of California San Diego

LigandPNGBDBM154579((2S)-2-[(2S)-2-hexanamido-3-methylbutanamido]-N,N-...)
Affinity DataIC50: 112nMpH: 7.5Assay Description:One nanomolar of proteasome was incubated with different inhibitor concentrations in Tris 25 mM pH 7.5; SDS 0.03%; EDTA 0.5 mM for 15 min at 37 °C in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2015
Entry Details Article
PubMed
TargetProteasome subunit alpha type-2(Baker's yeast)
University of California San Diego

LigandPNGBDBM154579((2S)-2-[(2S)-2-hexanamido-3-methylbutanamido]-N,N-...)
Affinity DataIC50: 165nMpH: 7.5Assay Description:One nanomolar of proteasome was incubated with different inhibitor concentrations in Tris 25 mM pH 7.5; SDS 0.03%; EDTA 0.5 mM for 15 min at 37 °C in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2015
Entry Details Article
PubMed
TargetProteasome subunit alpha type-2(Baker's yeast)
University of California San Diego

LigandPNGBDBM154579((2S)-2-[(2S)-2-hexanamido-3-methylbutanamido]-N,N-...)
Affinity DataIC50: 5.00E+4nMpH: 7.5Assay Description:One nanomolar of proteasome was incubated with different inhibitor concentrations in Tris 25 mM pH 7.5; SDS 0.03%; EDTA 0.5 mM for 15 min at 37 °C in...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2015
Entry Details Article
PubMed